SE8006119L - Tripeptidderivat och forfarande for framstellning derav - Google Patents

Tripeptidderivat och forfarande for framstellning derav

Info

Publication number
SE8006119L
SE8006119L SE8006119A SE8006119A SE8006119L SE 8006119 L SE8006119 L SE 8006119L SE 8006119 A SE8006119 A SE 8006119A SE 8006119 A SE8006119 A SE 8006119A SE 8006119 L SE8006119 L SE 8006119L
Authority
SE
Sweden
Prior art keywords
amino
alkylamino
lower alkyl
derivatives
formula
Prior art date
Application number
SE8006119A
Other languages
English (en)
Inventor
A A Failli
H U Immer
M K Gotz
Original Assignee
Ayerst Mckenna & Harrison
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ayerst Mckenna & Harrison filed Critical Ayerst Mckenna & Harrison
Publication of SE8006119L publication Critical patent/SE8006119L/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C07K5/0823—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Claims (1)

1. PATENTKRAV Aminoskyddade derivat av en fdrening, corn her formeln H - L - Pro - N - CH - C - Y - R3 (I) 11 R12 ,1 R van i R1 Sr vate, lagre alkyl eller NR4R5, van i R4 och R5 vardera Sr lagre alkyl, R2 Sr vats eller lagre alkyl, R3 Sr amino, lagre alkylamino, di(lagre alkyl)-amino eller amino-(lagre alkyl)-amino och Y Sr aminosyraresten Gly eller 0-Ala, med det fOrbehillet att nar R1 an NR4R5, Mr R3 lagre alkylamino, di(lagre alkyl)-amino eller amino-(lagre alkyl)-amino, corn Sr anvAndbara fOr framstallning av peptidderivat enligt formeln I.
SE8006119A 1975-07-28 1980-09-02 Tripeptidderivat och forfarande for framstellning derav SE8006119L (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/599,450 US4018912A (en) 1975-07-28 1975-07-28 Tripeptide derivatives with central nervous system activity and preparation thereof

Publications (1)

Publication Number Publication Date
SE8006119L true SE8006119L (sv) 1980-09-02

Family

ID=24399667

Family Applications (2)

Application Number Title Priority Date Filing Date
SE7608484A SE431330B (sv) 1975-07-28 1976-07-27 Forfarande for framstellning av tripeptidderivat, vilka har cns-aktivitet
SE8006119A SE8006119L (sv) 1975-07-28 1980-09-02 Tripeptidderivat och forfarande for framstellning derav

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SE7608484A SE431330B (sv) 1975-07-28 1976-07-27 Forfarande for framstellning av tripeptidderivat, vilka har cns-aktivitet

Country Status (10)

Country Link
US (1) US4018912A (sv)
JP (1) JPS6033854B2 (sv)
BE (1) BE844603A (sv)
CA (1) CA1062250A (sv)
CH (1) CH621111A5 (sv)
DE (1) DE2633976A1 (sv)
FR (1) FR2319378A1 (sv)
GB (1) GB1523685A (sv)
SE (2) SE431330B (sv)
SU (1) SU632299A3 (sv)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4093713A (en) * 1977-02-28 1978-06-06 Ayerst Mckenna & Harrison Ltd. Dipeptide derivatives with central nervous system activity and preparation thereof
DE3226242A1 (de) * 1982-07-14 1984-01-26 Basf Ag, 6700 Ludwigshafen N-acylderivate von dipeptiden, ihre herstellung und verwendung bei der therapie von krankheiten und mittel dafuer
DE3226241A1 (de) * 1982-07-14 1984-01-26 Basf Ag, 6700 Ludwigshafen N-acylderivate von peptiden, ihre herstellung und verwendung bei der bekaempfung von krankheiten und mittel dafuer
US5190924A (en) * 1991-02-13 1993-03-02 Boc Health Care, Inc. Peptide amides and amide dimers useful as muscle relaxants
US6767897B2 (en) * 1994-05-04 2004-07-27 Innapharma, Inc. Therapeutic uses of tri-, tetra-, penta-, and polypeptides
US5767083A (en) * 1994-05-04 1998-06-16 Innapharma, Inc. Tri-, tetra-, penta-, and polypeptides and their therapeutic use as an antidepressant agent
US5589460A (en) * 1994-05-04 1996-12-31 Innapharma, Inc. Tri-, tetra-, penta-, and polypeptides and their therapeutic use as an antidepressant agent
US6489300B1 (en) * 1997-07-31 2002-12-03 Eugene D. Thorsett Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4
DE19813849A1 (de) * 1998-03-27 1999-09-30 Degussa Verfahren zur einstufigen Umsalzung und Aufreinigung von Oligopeptiden

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1033906A (en) * 1962-03-30 1966-06-22 Geigy Ag J R Process for the production of a new tetrapeptide
NL6707845A (sv) * 1966-06-11 1967-12-12
BE787908A (fr) * 1971-08-24 1973-02-23 Abbott Lab Medicament antidepressif et antiparkinsonien
US3888840A (en) * 1973-02-07 1975-06-10 American Home Prod Novel hydrazinocarboxamide derivatives and preparation thereof

Also Published As

Publication number Publication date
JPS6033854B2 (ja) 1985-08-05
US4018912A (en) 1977-04-19
JPS5223070A (en) 1977-02-21
DE2633976A1 (de) 1977-02-10
CA1062250A (en) 1979-09-11
SU632299A3 (ru) 1978-11-05
BE844603A (fr) 1977-01-28
SE431330B (sv) 1984-01-30
GB1523685A (en) 1978-09-06
FR2319378A1 (fr) 1977-02-25
FR2319378B1 (sv) 1979-05-04
CH621111A5 (sv) 1981-01-15

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