SE409323B - Anvendning av en optisk isomer av bi-(4,5,6,7-tetrahydronaftyl)-fosforsyraderivat for kemisk upplosning av basiska optiska cis- och trans-isomerer - Google Patents
Anvendning av en optisk isomer av bi-(4,5,6,7-tetrahydronaftyl)-fosforsyraderivat for kemisk upplosning av basiska optiska cis- och trans-isomererInfo
- Publication number
- SE409323B SE409323B SE7203303A SE330372A SE409323B SE 409323 B SE409323 B SE 409323B SE 7203303 A SE7203303 A SE 7203303A SE 330372 A SE330372 A SE 330372A SE 409323 B SE409323 B SE 409323B
- Authority
- SE
- Sweden
- Prior art keywords
- afthyl
- tetrahydrone
- isomers
- trans
- phosphoric acid
- Prior art date
Links
- 230000003287 optical effect Effects 0.000 title 2
- 238000004090 dissolution Methods 0.000 title 1
- 150000003013 phosphoric acid derivatives Chemical class 0.000 title 1
- 239000000126 substance Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6571—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
- C07F9/6574—Esters of oxyacids of phosphorus
- C07F9/65744—Esters of oxyacids of phosphorus condensed with carbocyclic or heterocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Pyridine Compounds (AREA)
- Braiding, Manufacturing Of Bobbin-Net Or Lace, And Manufacturing Of Nets By Knotting (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT49167/71A IT951631B (it) | 1971-03-18 | 1971-03-18 | Composti utili per la separazione di isomeri ottici geometrici e strutturali e relativo procedimen to di sintesi |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SE409323B true SE409323B (sv) | 1979-08-13 |
Family
ID=11269830
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7203303A SE409323B (sv) | 1971-03-18 | 1972-03-15 | Anvendning av en optisk isomer av bi-(4,5,6,7-tetrahydronaftyl)-fosforsyraderivat for kemisk upplosning av basiska optiska cis- och trans-isomerer |
Country Status (18)
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4143028A (en) * | 1977-12-05 | 1979-03-06 | Ciba-Geigy Corporation | Alkylated 1,1'-biphenyl-2,2'-diyl phosphonites and stabilized compositions |
| US5288914A (en) * | 1984-08-27 | 1994-02-22 | The Dow Chemical Company | Poly(arylcyclobutenes) |
| NL8403224A (nl) * | 1984-10-24 | 1986-05-16 | Oce Andeno Bv | Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen. |
| DE3940765A1 (de) * | 1989-12-09 | 1991-06-13 | Hoechst Ag | Verfahren zur herstellung reiner cyclischer phosphorsaeurediarylester |
| AU689578B2 (en) * | 1994-05-16 | 1998-04-02 | Aventisub Ii Inc. | Process and diastereomeric salts useful for the optical resolution of racemic alpha-(4-(1,1-dimethylethyl)phenyl)-4-(hydroxydiphenylmethyl )-1-piperidinebutanol and derivative compounds |
| JP4725757B2 (ja) * | 1999-03-24 | 2011-07-13 | 東ソー株式会社 | ビナフトールリン酸誘導体及びその利用 |
| DE60008807T2 (de) | 1999-03-24 | 2005-01-13 | Tosoh Corp., Shinnanyo | Binaphtol-monophosphorsäurederivate und deren Verwendung |
| US6800778B1 (en) | 1999-10-22 | 2004-10-05 | Takeda Chemical Industries, Ltd. | Process for producing optically active naphthalene derivative and optical resolver therefor |
| WO2001034557A1 (fr) * | 1999-11-10 | 2001-05-17 | Takeda Chemical Industries, Ltd. | Procede de production de derives d'enaminone cycliques optiquement actifs |
| US6391926B2 (en) | 2000-03-13 | 2002-05-21 | Tosoh Corporation | Optically active phosphate derivative |
| NZ530491A (en) | 2001-07-09 | 2007-08-31 | Repros Therapeutics Inc | Composition comprising 0-29% cis-clomiphene and 79-100% trans-clomiphene testosterone deficiency in men |
| WO2004096753A1 (ja) * | 2003-04-25 | 2004-11-11 | Toagosei Co., Ltd. | キラルなブレンステッド酸による不斉合成用触媒および当該触媒を用いた不斉合成方法 |
| US7229557B2 (en) * | 2004-02-04 | 2007-06-12 | Konec, Inc. | Method to separate stereoisomers |
| WO2011042910A2 (en) * | 2009-10-09 | 2011-04-14 | Hetero Research Foundation | Optical resolution of substituted 2-(2- pyridinylmethylsulphinyl)-1h-benzimidazoles |
| UA113291C2 (xx) | 2011-08-04 | 2017-01-10 | Метаболіти транскломіфену і їх застосування | |
| JP2015527360A (ja) | 2012-08-21 | 2015-09-17 | レプロス セラピューティクス インコーポレイティド | トランス−クロミフェン製剤およびその使用 |
| US9687458B2 (en) | 2012-11-02 | 2017-06-27 | Repros Therapeutics Inc. | Trans-clomiphene for use in cancer therapy |
| CA2942301A1 (en) * | 2014-03-11 | 2015-09-17 | Repros Therapeutics Inc. | Clomiphene synthesis using a single solvent |
| LT3171866T (lt) | 2014-07-24 | 2020-12-28 | Aspen Park Pharmaceuticals, Inc. | Androgenų deprivacijos terapijos sukeltų karščio bangų ir kaulų retėjimo gydymas cis-klomifenu |
| EP3015454A1 (en) * | 2014-10-28 | 2016-05-04 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Stable solid form of trans-Clomiphene citrate |
| EP3015453B1 (en) | 2014-10-28 | 2016-10-12 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Process for the preparation of Clomiphene |
| CA2989364C (en) * | 2016-04-22 | 2021-07-20 | F.I.S. - Fabbrica Italiana Sintetici S.P.A. | Process for the preparation of enclomiphene citrate having needle shaped crystal habit. |
| TWI793165B (zh) | 2017-09-11 | 2023-02-21 | 美商阿托薩醫療公司 | 製造及使用因多昔芬(endoxifen)之方法 |
| FR3082842A1 (fr) * | 2018-06-21 | 2019-12-27 | Veru Inc. | Polymorphe de cis-clomiphene (zuclomiphene) et procedes d'utilisation de celui-ci |
| US12201591B2 (en) | 2019-07-03 | 2025-01-21 | Atossa Therapeutics, Inc. | Sustained release compositions of endoxifen |
| CA3098552A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Processes for the preparation of zuclomiphene and intermediates thereof |
| CA3098725A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Zuclpomiphene salts and crystalline forms thereof |
| CA3105944A1 (en) | 2020-01-22 | 2021-07-22 | Apotex Inc. | Crystalline forms of zuclomiphene citrate |
| EP3907213A1 (en) | 2020-05-04 | 2021-11-10 | Pcas | Processes for the production of isomerically pure or enriched cis-clomiphene |
| US11578025B2 (en) | 2020-10-19 | 2023-02-14 | Apotex Inc. | Processes for the preparation of zuclomiphene intermediates |
-
1971
- 1971-03-18 IT IT49167/71A patent/IT951631B/it active
-
1972
- 1972-02-28 ZA ZA721297A patent/ZA721297B/xx unknown
- 1972-02-29 IL IL38860A patent/IL38860A/xx unknown
- 1972-03-03 AU AU39611/72A patent/AU462431B2/en not_active Expired
- 1972-03-03 PH PH13312A patent/PH10768A/en unknown
- 1972-03-09 GB GB1104172A patent/GB1360946A/en not_active Expired
- 1972-03-09 CA CA136,671A patent/CA961500A/en not_active Expired
- 1972-03-10 US US00233793A patent/US3848030A/en not_active Expired - Lifetime
- 1972-03-15 SE SE7203303A patent/SE409323B/xx unknown
- 1972-03-16 DE DE2212660A patent/DE2212660C3/de not_active Expired
- 1972-03-17 BE BE780887A patent/BE780887A/xx unknown
- 1972-03-17 CH CH395572A patent/CH576921A5/xx not_active IP Right Cessation
- 1972-03-17 FR FR7209350A patent/FR2129741A5/fr not_active Expired
- 1972-03-17 JP JP2661472A patent/JPS5547013B1/ja active Pending
- 1972-03-17 NL NL7203574A patent/NL7203574A/xx not_active Application Discontinuation
- 1972-03-17 NO NO880/72A patent/NO136357C/no unknown
- 1972-03-17 ES ES400862A patent/ES400862A1/es not_active Expired
- 1972-03-17 DK DK127372AA patent/DK139944B/da unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL38860A0 (en) | 1972-04-27 |
| NL7203574A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1972-09-20 |
| BE780887A (fr) | 1972-07-17 |
| IL38860A (en) | 1975-06-25 |
| JPS5547013B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1980-11-27 |
| DK139944C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1979-10-22 |
| CA961500A (en) | 1975-01-21 |
| DE2212660C3 (de) | 1981-09-24 |
| IT951631B (it) | 1973-07-10 |
| ES400862A1 (es) | 1976-04-16 |
| FR2129741A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1972-10-27 |
| PH10768A (en) | 1977-09-05 |
| DE2212660A1 (de) | 1972-09-28 |
| US3848030A (en) | 1974-11-12 |
| GB1360946A (en) | 1974-07-24 |
| DK139944B (da) | 1979-05-21 |
| ZA721297B (en) | 1973-03-28 |
| NO136357B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-05-16 |
| AU462431B2 (en) | 1975-06-09 |
| AU3961172A (en) | 1973-09-06 |
| CH576921A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1976-06-30 |
| NO136357C (no) | 1977-08-24 |
| DE2212660B2 (de) | 1980-07-10 |
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