DK139944B - Optisk aktive syrer til anvendelse ved adskillelse af isomere af visse kemiske forbindelser. - Google Patents
Optisk aktive syrer til anvendelse ved adskillelse af isomere af visse kemiske forbindelser.Info
- Publication number
- DK139944B DK139944B DK127372AA DK127372A DK139944B DK 139944 B DK139944 B DK 139944B DK 127372A A DK127372A A DK 127372AA DK 127372 A DK127372 A DK 127372A DK 139944 B DK139944 B DK 139944B
- Authority
- DK
- Denmark
- Prior art keywords
- isomers
- separation
- optically active
- chemical compounds
- certain chemical
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000007513 acids Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- SYSQUGFVNFXIIT-UHFFFAOYSA-N n-[4-(1,3-benzoxazol-2-yl)phenyl]-4-nitrobenzenesulfonamide Chemical class C1=CC([N+](=O)[O-])=CC=C1S(=O)(=O)NC1=CC=C(C=2OC3=CC=CC=C3N=2)C=C1 SYSQUGFVNFXIIT-UHFFFAOYSA-N 0.000 title 1
- 238000000926 separation method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6571—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
- C07F9/6574—Esters of oxyacids of phosphorus
- C07F9/65744—Esters of oxyacids of phosphorus condensed with carbocyclic or heterocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Pyridine Compounds (AREA)
- Braiding, Manufacturing Of Bobbin-Net Or Lace, And Manufacturing Of Nets By Knotting (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT49167/71A IT951631B (it) | 1971-03-18 | 1971-03-18 | Composti utili per la separazione di isomeri ottici geometrici e strutturali e relativo procedimen to di sintesi |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK139944B true DK139944B (da) | 1979-05-21 |
| DK139944C DK139944C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1979-10-22 |
Family
ID=11269830
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK127372AA DK139944B (da) | 1971-03-18 | 1972-03-17 | Optisk aktive syrer til anvendelse ved adskillelse af isomere af visse kemiske forbindelser. |
Country Status (18)
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4143028A (en) * | 1977-12-05 | 1979-03-06 | Ciba-Geigy Corporation | Alkylated 1,1'-biphenyl-2,2'-diyl phosphonites and stabilized compositions |
| US5288914A (en) * | 1984-08-27 | 1994-02-22 | The Dow Chemical Company | Poly(arylcyclobutenes) |
| NL8403224A (nl) * | 1984-10-24 | 1986-05-16 | Oce Andeno Bv | Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen. |
| DE3940765A1 (de) * | 1989-12-09 | 1991-06-13 | Hoechst Ag | Verfahren zur herstellung reiner cyclischer phosphorsaeurediarylester |
| PT759904E (pt) * | 1994-05-16 | 2000-10-31 | Merrell Pharma Inc | Processo e sais diastereomericos uteis para a resolucao optica de alfa-¬4-(1,1-dimetiletil)-fenil|-4-(hidroxidifenilmetil)-1-piperidinobutanol racemico e compostos derivados |
| JP4725757B2 (ja) * | 1999-03-24 | 2011-07-13 | 東ソー株式会社 | ビナフトールリン酸誘導体及びその利用 |
| US6274745B1 (en) | 1999-03-24 | 2001-08-14 | Tosoh Corporation | Binaphthol monophosphoric acid derivative and its use |
| ATE320420T1 (de) * | 1999-10-22 | 2006-04-15 | Takeda Pharmaceutical | Verfahren zur herstellung von optisch aktiven naphthalinderivaten und darin eingesetzte optische resolver |
| AU1303001A (en) * | 1999-11-10 | 2001-06-06 | Takeda Chemical Industries Ltd. | Process for the production of optically active cyclic enaminone derivatives |
| US6391926B2 (en) | 2000-03-13 | 2002-05-21 | Tosoh Corporation | Optically active phosphate derivative |
| CN1289075C (zh) | 2001-07-09 | 2006-12-13 | 佐纳根有限公司 | 富含反式克罗米酚的克罗米酚组合物的用途 |
| US7517828B2 (en) * | 2003-04-25 | 2009-04-14 | Toagosei Co., Ltd. | Chiral broensted acid catalyst for asymmetric synthesis and method of asymmetric synthesis with the catalyst |
| US7229557B2 (en) * | 2004-02-04 | 2007-06-12 | Konec, Inc. | Method to separate stereoisomers |
| US8420822B2 (en) * | 2009-10-09 | 2013-04-16 | Hetero Research Foundation | Optical resolution of substituted 2-(2-pyridinylmethylsulphinyl)-1H-benzimidazoles |
| UA113291C2 (xx) | 2011-08-04 | 2017-01-10 | Метаболіти транскломіфену і їх застосування | |
| SG10201704820SA (en) | 2012-08-21 | 2017-07-28 | Repros Therapeutics Inc | Trans-clomiphene formulations and uses thereof |
| MX2015005160A (es) | 2012-11-02 | 2015-07-17 | Repros Therapeutics Inc | Trans-clomifeno para uso en terapia de cancer. |
| CN106068121A (zh) * | 2014-03-11 | 2016-11-02 | 利普生物药剂公司 | 使用单一溶剂进行克罗米芬合成 |
| WO2016014812A1 (en) | 2014-07-24 | 2016-01-28 | Aspen Park Pharmaceuticals, Inc. | Treating androgen deprivation therapy induced hot flashes and bone loss using cis-clomiphene |
| EP3015454A1 (en) * | 2014-10-28 | 2016-05-04 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Stable solid form of trans-Clomiphene citrate |
| EP3015453B1 (en) | 2014-10-28 | 2016-10-12 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Process for the preparation of Clomiphene |
| US10364212B2 (en) | 2016-04-22 | 2019-07-30 | F.I.S.—Fabbrica Italiana Sintetici S.p.A. | Process for the preparation of enclomiphene citrate having needle shaped crystal habit |
| WO2019051416A1 (en) | 2017-09-11 | 2019-03-14 | Atossa Genetics Inc. | METHODS FOR THE MANUFACTURE AND USE OF ENDOXIFEN |
| FR3082842A1 (fr) * | 2018-06-21 | 2019-12-27 | Veru Inc. | Polymorphe de cis-clomiphene (zuclomiphene) et procedes d'utilisation de celui-ci |
| KR20220042352A (ko) | 2019-07-03 | 2022-04-05 | 아토사 테라퓨틱스, 인크. | 엔독시펜의 서방성 조성물 |
| CA3098552A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Processes for the preparation of zuclomiphene and intermediates thereof |
| CA3098725A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Zuclpomiphene salts and crystalline forms thereof |
| CA3105944A1 (en) | 2020-01-22 | 2021-07-22 | Apotex Inc. | Crystalline forms of zuclomiphene citrate |
| EP3907213A1 (en) | 2020-05-04 | 2021-11-10 | Pcas | Processes for the production of isomerically pure or enriched cis-clomiphene |
| US11578025B2 (en) | 2020-10-19 | 2023-02-14 | Apotex Inc. | Processes for the preparation of zuclomiphene intermediates |
-
1971
- 1971-03-18 IT IT49167/71A patent/IT951631B/it active
-
1972
- 1972-02-28 ZA ZA721297A patent/ZA721297B/xx unknown
- 1972-02-29 IL IL38860A patent/IL38860A/xx unknown
- 1972-03-03 AU AU39611/72A patent/AU462431B2/en not_active Expired
- 1972-03-03 PH PH13312A patent/PH10768A/en unknown
- 1972-03-09 GB GB1104172A patent/GB1360946A/en not_active Expired
- 1972-03-09 CA CA136,671A patent/CA961500A/en not_active Expired
- 1972-03-10 US US00233793A patent/US3848030A/en not_active Expired - Lifetime
- 1972-03-15 SE SE7203303A patent/SE409323B/xx unknown
- 1972-03-16 DE DE2212660A patent/DE2212660C3/de not_active Expired
- 1972-03-17 NO NO880/72A patent/NO136357C/no unknown
- 1972-03-17 BE BE780887A patent/BE780887A/xx unknown
- 1972-03-17 NL NL7203574A patent/NL7203574A/xx not_active Application Discontinuation
- 1972-03-17 ES ES400862A patent/ES400862A1/es not_active Expired
- 1972-03-17 FR FR7209350A patent/FR2129741A5/fr not_active Expired
- 1972-03-17 JP JP2661472A patent/JPS5547013B1/ja active Pending
- 1972-03-17 DK DK127372AA patent/DK139944B/da unknown
- 1972-03-17 CH CH395572A patent/CH576921A5/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| IT951631B (it) | 1973-07-10 |
| AU462431B2 (en) | 1975-06-09 |
| ES400862A1 (es) | 1976-04-16 |
| IL38860A0 (en) | 1972-04-27 |
| CA961500A (en) | 1975-01-21 |
| GB1360946A (en) | 1974-07-24 |
| US3848030A (en) | 1974-11-12 |
| NL7203574A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1972-09-20 |
| DE2212660B2 (de) | 1980-07-10 |
| DK139944C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1979-10-22 |
| FR2129741A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1972-10-27 |
| SE409323B (sv) | 1979-08-13 |
| NO136357B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-05-16 |
| BE780887A (fr) | 1972-07-17 |
| DE2212660A1 (de) | 1972-09-28 |
| DE2212660C3 (de) | 1981-09-24 |
| CH576921A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1976-06-30 |
| JPS5547013B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1980-11-27 |
| NO136357C (no) | 1977-08-24 |
| AU3961172A (en) | 1973-09-06 |
| PH10768A (en) | 1977-09-05 |
| ZA721297B (en) | 1973-03-28 |
| IL38860A (en) | 1975-06-25 |
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