SE382058B - Forfarande for framstellning av nya alfa aryl-4-substituerade piperidinoalkanolderivat - Google Patents

Forfarande for framstellning av nya alfa aryl-4-substituerade piperidinoalkanolderivat

Info

Publication number
SE382058B
SE382058B SE7300974A SE7300974A SE382058B SE 382058 B SE382058 B SE 382058B SE 7300974 A SE7300974 A SE 7300974A SE 7300974 A SE7300974 A SE 7300974A SE 382058 B SE382058 B SE 382058B
Authority
SE
Sweden
Prior art keywords
piperidinoal
aryl
substituted
procedure
preparing new
Prior art date
Application number
SE7300974A
Other languages
English (en)
Swedish (sv)
Inventor
A A Carr
C R Kinsolvning
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22829539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE382058(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of SE382058B publication Critical patent/SE382058B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/70Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SE7300974A 1972-01-28 1973-01-24 Forfarande for framstellning av nya alfa aryl-4-substituerade piperidinoalkanolderivat SE382058B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22182172A 1972-01-28 1972-01-28

Publications (1)

Publication Number Publication Date
SE382058B true SE382058B (sv) 1976-01-12

Family

ID=22829539

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7300974A SE382058B (sv) 1972-01-28 1973-01-24 Forfarande for framstellning av nya alfa aryl-4-substituerade piperidinoalkanolderivat

Country Status (26)

Country Link
JP (1) JPS5115035B2 (xx)
AR (1) AR195314A1 (xx)
AT (2) AT323742B (xx)
AU (1) AU467361B2 (xx)
BE (1) BE794597A (xx)
CA (1) CA978946A (xx)
CH (2) CH587820A5 (xx)
CS (1) CS177834B2 (xx)
DD (1) DD103239A5 (xx)
DE (1) DE2303306C3 (xx)
DK (1) DK136713B (xx)
ES (1) ES410731A1 (xx)
FR (1) FR2181690B1 (xx)
GB (1) GB1413138A (xx)
HU (1) HU166477B (xx)
IE (1) IE36983B1 (xx)
IL (1) IL41060A (xx)
LU (1) LU66916A1 (xx)
NL (1) NL175410C (xx)
NO (1) NO140057C (xx)
PH (1) PH10264A (xx)
PL (1) PL89095B1 (xx)
SE (1) SE382058B (xx)
SU (1) SU464997A3 (xx)
YU (1) YU36013B (xx)
ZA (1) ZA728544B (xx)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3941795A (en) 1974-02-08 1976-03-02 Richardson-Merrell Inc. α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES
US4254129A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
US4254130A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
IT1200123B (it) * 1985-09-27 1989-01-05 Ind Chimica Srl Procedimento per la preparazione di alfa-(p-terbutilfenil)-4-(idrossidifenilmetil)-1-piperidinobutanolo
US4742175A (en) * 1986-05-07 1988-05-03 Merrell Dow Pharmaceuticals Inc. Preparation of polymorphically pure terfenadine
JPS63101760U (xx) * 1986-12-19 1988-07-02
IT1205685B (it) * 1987-05-26 1989-03-31 Erregierre Spa Processo per la preparazione di alfa-(alchilfenil)-4-(idrossi difenilmetil)-1-piperidina butanolo
ZA901360B (en) * 1989-02-28 1990-11-28 Merrell Dow Pharma Preparation of the low-melting polymorphic form of terfenadine
CA2015390A1 (en) * 1989-05-01 1990-11-01 Frederick J. Mccarty Process for the preparation of the high melting polymorphic of terfenadine
DE3917241A1 (de) * 1989-05-26 1990-11-29 Schaper & Bruemmer Gmbh 4-(hydroxydiphenylmethyl)-1-piperidyl-phenylalkan-derivate
US5466691A (en) * 1991-08-09 1995-11-14 Yoshitomi Pharmaceutical Industries, Ltd. Thiophene compound
JPH11504650A (ja) * 1995-05-08 1999-04-27 ヘキスト・マリオン・ルセル・インコーポレイテツド アルファ−(置換アルキルフェニル)−4−(ヒドロキシジフェニルメチル)−1−ピペリジンブタノール誘導体、その製造および抗ヒスタミン剤、抗アレルギー剤および気管支拡張剤としてのその使用
ES2216191T3 (es) * 1997-03-11 2004-10-16 Aventis Pharmaceuticals Inc. Procedimiento para preparar acido 4-(4-(hidroxidifenil)-1-piperidinil)-1-hidroxibutil)-alfa,alfa-dimetilfenilacetico y derivados fosforilados.
US7498345B2 (en) * 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of piperidine derivatives
US8153385B2 (en) 2004-10-18 2012-04-10 Reverse Proteomics Research Institute Co., Ltd. Target protein and target gene in drug designing and screening method

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3081303A (en) * 1961-10-13 1963-03-12 Searle & Co 1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols
GB1242169A (en) * 1969-04-09 1971-08-11 Ucb Sa Piperidine derivatives

Also Published As

Publication number Publication date
CS177834B2 (xx) 1977-08-31
CH587820A5 (xx) 1977-05-13
DE2303306C3 (de) 1979-05-31
NO140057B (no) 1979-03-19
IE36983L (en) 1973-07-28
FR2181690B1 (xx) 1976-05-14
NL175410C (nl) 1984-11-01
IL41060A (en) 1975-06-25
IE36983B1 (en) 1977-04-13
DK136713B (da) 1977-11-14
PH10264A (en) 1976-10-20
JPS5115035B2 (xx) 1976-05-13
PL89095B1 (xx) 1976-10-30
FR2181690A1 (xx) 1973-12-07
SU464997A3 (ru) 1975-03-25
ZA728544B (en) 1974-02-27
NO140057C (no) 1979-07-04
DK136713C (xx) 1978-05-01
NL175410B (nl) 1984-06-01
YU3473A (en) 1981-02-28
LU66916A1 (xx) 1973-07-27
AR195314A1 (es) 1973-09-28
JPS4885578A (xx) 1973-11-13
CH593259A5 (xx) 1977-11-30
CA978946A (en) 1975-12-02
YU36013B (en) 1981-11-13
DE2303306A1 (de) 1973-08-02
DE2303306B2 (de) 1978-09-28
HU166477B (xx) 1975-03-28
ES410731A1 (es) 1976-04-01
AU4989372A (en) 1974-06-13
AU467361B2 (en) 1975-11-27
NL7300873A (xx) 1973-07-31
GB1413138A (en) 1975-11-05
AT321917B (de) 1975-04-25
IL41060A0 (en) 1973-02-28
DD103239A5 (xx) 1974-01-12
BE794597A (fr) 1973-05-16
AT323742B (de) 1975-07-25

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Legal Events

Date Code Title Description
SPCF Application for supplementary protection certificate filed

Free format text: 7300974

SPCG Supplementary protection certificate granted

Free format text: 7300974, EXPIRES: 19990523