SA516371037B1 - معدلات مستقبل nmda وعقاقير أولية منها وأملاح منها واستخداماتها - Google Patents
معدلات مستقبل nmda وعقاقير أولية منها وأملاح منها واستخداماتها Download PDFInfo
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- SA516371037B1 SA516371037B1 SA516371037A SA516371037A SA516371037B1 SA 516371037 B1 SA516371037 B1 SA 516371037B1 SA 516371037 A SA516371037 A SA 516371037A SA 516371037 A SA516371037 A SA 516371037A SA 516371037 B1 SA516371037 B1 SA 516371037B1
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- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Ophthalmology & Optometry (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Gastroenterology & Hepatology (AREA)
- Epidemiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361896308P | 2013-10-28 | 2013-10-28 | |
| PCT/US2014/062367 WO2015065891A1 (en) | 2013-10-28 | 2014-10-27 | Nmda receptor modulators and prodrugs, salts, and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SA516371037B1 true SA516371037B1 (ar) | 2018-05-16 |
Family
ID=53004986
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SA516371037A SA516371037B1 (ar) | 2013-10-28 | 2016-04-28 | معدلات مستقبل nmda وعقاقير أولية منها وأملاح منها واستخداماتها |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US9745342B2 (ja) |
| EP (2) | EP3564256A1 (ja) |
| JP (1) | JP6603668B2 (ja) |
| KR (1) | KR20160077153A (ja) |
| CN (2) | CN105764522A (ja) |
| AU (2) | AU2014342624A1 (ja) |
| BR (1) | BR112016009443A8 (ja) |
| CA (1) | CA2928701A1 (ja) |
| CL (2) | CL2016001001A1 (ja) |
| IL (1) | IL245302B (ja) |
| MX (2) | MX2016005510A (ja) |
| RU (1) | RU2016119830A (ja) |
| SA (1) | SA516371037B1 (ja) |
| SG (2) | SG11201603376UA (ja) |
| WO (1) | WO2015065891A1 (ja) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102257284B1 (ko) | 2013-01-22 | 2021-05-28 | 비스타젠 쎄라퓨틱스, 인크. | L-4-클로로키뉴레닌의 투여형 및 치료적 용도 |
| CN116082461B (zh) * | 2022-10-14 | 2023-11-14 | 浙江大学 | 一种具有抗菌活性的小分子肽及其应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1801118A4 (en) | 2004-09-14 | 2009-09-02 | Shionogi & Co | METHOD FOR SYNTHESIS OF MUCIN-TYPE PEPTIDES AND GLUCKOPEPTIDES RELATED TO MUC1 |
| CA2686827C (en) * | 2006-12-14 | 2014-09-16 | Aileron Therapeutics, Inc. | Bis-sulfhydryl macrocyclization systems |
| WO2008104000A2 (en) * | 2007-02-23 | 2008-08-28 | Aileron Therapeutics, Inc. | Triazole macrocycle systems |
| AU2009293164B2 (en) * | 2008-09-18 | 2015-07-09 | Northwestern University | NMDA receptor modulators and uses thereof |
| CA2737921C (en) * | 2008-09-22 | 2019-01-15 | Aileron Therapeutics, Inc. | Methods for preparing purified alpha-helical peptidomimetic macrocycle compositions with low metal ppm levels |
| BR112012020142A2 (pt) * | 2010-02-11 | 2020-08-18 | Northwestern University | moduladores do receptor de nmda com estrutura secundária estabilizada e usos dos mesmos. |
| KR101692275B1 (ko) * | 2010-02-11 | 2017-01-04 | 노오쓰웨스턴 유니버시티 | ２차 구조 안정화된 ｎｍｄａ 수용체 조절제 및 그의 용도 |
| EA201790653A1 (ru) * | 2011-04-27 | 2017-07-31 | Нортвестерн Юниверсити | Способ лечения болезни альцгеймера и других расстройств |
-
2014
- 2014-10-27 SG SG11201603376UA patent/SG11201603376UA/en unknown
- 2014-10-27 EP EP19159957.0A patent/EP3564256A1/en not_active Withdrawn
- 2014-10-27 AU AU2014342624A patent/AU2014342624A1/en not_active Abandoned
- 2014-10-27 CA CA2928701A patent/CA2928701A1/en not_active Abandoned
- 2014-10-27 JP JP2016552196A patent/JP6603668B2/ja not_active Expired - Fee Related
- 2014-10-27 RU RU2016119830A patent/RU2016119830A/ru unknown
- 2014-10-27 KR KR1020167013971A patent/KR20160077153A/ko not_active Application Discontinuation
- 2014-10-27 CN CN201480064349.XA patent/CN105764522A/zh active Pending
- 2014-10-27 BR BR112016009443A patent/BR112016009443A8/pt not_active IP Right Cessation
- 2014-10-27 CN CN202010688442.5A patent/CN112321678A/zh active Pending
- 2014-10-27 US US15/033,031 patent/US9745342B2/en active Active
- 2014-10-27 SG SG10201810496XA patent/SG10201810496XA/en unknown
- 2014-10-27 WO PCT/US2014/062367 patent/WO2015065891A1/en active Application Filing
- 2014-10-27 EP EP14858298.4A patent/EP3062810A4/en not_active Withdrawn
- 2014-10-27 MX MX2016005510A patent/MX2016005510A/es unknown
-
2016
- 2016-04-25 IL IL245302A patent/IL245302B/en active IP Right Grant
- 2016-04-27 MX MX2021000029A patent/MX2021000029A/es unknown
- 2016-04-27 CL CL2016001001A patent/CL2016001001A1/es unknown
- 2016-04-28 SA SA516371037A patent/SA516371037B1/ar unknown
-
2017
- 2017-07-24 US US15/658,107 patent/US10590167B2/en not_active Expired - Fee Related
-
2020
- 2020-02-17 AU AU2020201109A patent/AU2020201109A1/en not_active Abandoned
- 2020-08-31 CL CL2020002247A patent/CL2020002247A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20180127466A1 (en) | 2018-05-10 |
| IL245302B (en) | 2020-05-31 |
| EP3062810A4 (en) | 2017-05-03 |
| CN112321678A (zh) | 2021-02-05 |
| CL2020002247A1 (es) | 2021-02-05 |
| WO2015065891A1 (en) | 2015-05-07 |
| EP3564256A1 (en) | 2019-11-06 |
| US10590167B2 (en) | 2020-03-17 |
| AU2014342624A1 (en) | 2016-06-02 |
| AU2020201109A1 (en) | 2020-03-05 |
| MX2021000029A (es) | 2021-03-25 |
| US9745342B2 (en) | 2017-08-29 |
| BR112016009443A8 (pt) | 2020-03-24 |
| RU2016119830A3 (ja) | 2018-07-02 |
| JP6603668B2 (ja) | 2019-11-06 |
| IL245302A0 (en) | 2016-06-30 |
| EP3062810A1 (en) | 2016-09-07 |
| CA2928701A1 (en) | 2015-05-07 |
| RU2016119830A (ru) | 2017-12-04 |
| CL2016001001A1 (es) | 2016-12-16 |
| SG10201810496XA (en) | 2018-12-28 |
| MX2016005510A (es) | 2017-01-06 |
| US20160244485A1 (en) | 2016-08-25 |
| JP2016537413A (ja) | 2016-12-01 |
| KR20160077153A (ko) | 2016-07-01 |
| SG11201603376UA (en) | 2016-05-30 |
| CN105764522A (zh) | 2016-07-13 |
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