SA07280027B1 - مركبات سبيرو [إميدازوليدين -4، 3' - إندول] -2، 2'، 5(1'h) – ترايون جديدة لمعالجة الحالات المصاحبة لمستقبل فانيلويد 1 - Google Patents
مركبات سبيرو [إميدازوليدين -4، 3' - إندول] -2، 2'، 5(1'h) – ترايون جديدة لمعالجة الحالات المصاحبة لمستقبل فانيلويد 1 Download PDFInfo
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- SA07280027B1 SA07280027B1 SA07280027A SA07280027A SA07280027B1 SA 07280027 B1 SA07280027 B1 SA 07280027B1 SA 07280027 A SA07280027 A SA 07280027A SA 07280027 A SA07280027 A SA 07280027A SA 07280027 B1 SA07280027 B1 SA 07280027B1
- Authority
- SA
- Saudi Arabia
- Prior art keywords
- pain
- compound
- indole
- salt
- imidazolidine
- Prior art date
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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Applications Claiming Priority (1)
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| US77111906P | 2006-02-07 | 2006-02-07 |
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| EP2781521A4 (en) | 2011-10-19 | 2015-03-04 | Kowa Co | NEW SPIROINDOLIN COMPOUND AND MEDICAL AGENT THEREFOR |
| TWI586668B (zh) * | 2012-09-06 | 2017-06-11 | 第一三共股份有限公司 | 二螺吡咯啶衍生物之結晶 |
| CN108409746B (zh) * | 2018-05-15 | 2021-08-24 | 中山大学 | 一种含吡咯或吲哚并氮杂环烷结构的手性氧代螺环吲哚类化合物及其消旋体和制备方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU532110B2 (en) | 1979-11-13 | 1983-09-15 | Ici Ltd. | Spiro(imidazolidine-4,3:-indoline)-2,2:5-trione derivatives |
| ZA806623B (en) * | 1979-11-13 | 1981-12-30 | Ici Ltd | Substituted indoline-2-one derivatives |
| IE52879B1 (en) | 1981-05-12 | 1988-03-30 | Ici Plc | Pharmaceutical spiro-hydantoin derivatives |
| GB8331194D0 (en) | 1982-12-20 | 1983-12-29 | Ici Plc | Chemical process |
| US4611062A (en) * | 1984-03-26 | 1986-09-09 | Imperial Chemical Industries Plc | Process for resolving certain spiro compounds |
| WO1992007830A2 (en) | 1990-10-29 | 1992-05-14 | Pfizer Inc. | Oxindole peptide antagonists |
| HUP0203548A3 (en) * | 1999-07-21 | 2003-04-28 | Astrazeneca Ab | New spirooxindole derivatives, process for their preparation, pharmaceutical compositions containing them and their use |
| US7248802B2 (en) | 2002-11-27 | 2007-07-24 | Nokia Corporation | Distribution of a synchronization signal in an optical communication system |
| TW200508197A (en) | 2003-03-31 | 2005-03-01 | Ucb Sa | Indolone-acetamide derivatives, processes for preparing them and their uses |
| SE0301446D0 (sv) * | 2003-05-16 | 2003-05-16 | Astrazeneca Ab | New Compounds |
| US7585878B2 (en) | 2003-06-12 | 2009-09-08 | Astellas Pharma Inc. | Benzamide derivative or salt thereof |
| GB0326633D0 (en) * | 2003-11-14 | 2003-12-17 | Merck Sharp & Dohme | Therapeutic agents |
| US7879866B2 (en) | 2004-07-19 | 2011-02-01 | Dorte Xenia Gram | Inhibition of the activity of the capsaicin receptor in the treatment of obesity or obesity-related diseases and disorders |
| WO2007091948A2 (en) * | 2006-02-07 | 2007-08-16 | Astrazeneca Ab | Novel spiro [imidazolidine-4, 3´-indole] 2, 2´,5´(1h) triones for treatment of conditions associated with vanilloid receptor 1 |
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2007
- 2007-01-31 AR ARP070100412A patent/AR059265A1/es not_active Application Discontinuation
- 2007-01-31 TW TW096103591A patent/TW200801011A/zh unknown
- 2007-02-05 US US11/671,153 patent/US20070185179A1/en not_active Abandoned
- 2007-02-06 AU AU2007212786A patent/AU2007212786B2/en not_active Ceased
- 2007-02-06 SG SG201100854-7A patent/SG169387A1/en unknown
- 2007-02-06 KR KR1020087019272A patent/KR20080094906A/ko not_active Withdrawn
- 2007-02-06 SA SA07280027A patent/SA07280027B1/ar unknown
- 2007-02-06 RU RU2008131905/04A patent/RU2421457C2/ru not_active IP Right Cessation
- 2007-02-06 UY UY30132A patent/UY30132A1/es not_active Application Discontinuation
- 2007-02-06 NZ NZ571070A patent/NZ571070A/en unknown
- 2007-02-06 EP EP07709323A patent/EP2013215A4/en not_active Withdrawn
- 2007-02-06 BR BRPI0707423-9A patent/BRPI0707423A2/pt not_active IP Right Cessation
- 2007-02-06 CA CA002641632A patent/CA2641632A1/en not_active Abandoned
- 2007-02-06 JP JP2008554186A patent/JP2009526043A/ja active Pending
- 2007-02-06 CN CNA2007800125819A patent/CN101415711A/zh active Pending
- 2007-02-06 WO PCT/SE2007/000107 patent/WO2007091947A2/en not_active Ceased
- 2007-06-02 UA UAA200809311A patent/UA93226C2/ru unknown
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2008
- 2008-07-17 IL IL192890A patent/IL192890A0/en unknown
- 2008-07-23 ZA ZA200806407A patent/ZA200806407B/xx unknown
- 2008-08-14 NO NO20083547A patent/NO20083547L/no not_active Application Discontinuation
- 2008-11-20 US US12/274,837 patent/US7868181B2/en not_active Expired - Fee Related
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2009
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|---|---|
| AU2007212786A1 (en) | 2007-08-16 |
| AU2007212786A8 (en) | 2010-05-06 |
| IL192890A0 (en) | 2009-02-11 |
| NZ571070A (en) | 2011-07-29 |
| WO2007091947A8 (en) | 2008-08-07 |
| AU2007212786B2 (en) | 2011-06-02 |
| RU2008131905A (ru) | 2010-03-20 |
| EP2013215A2 (en) | 2009-01-14 |
| US7868181B2 (en) | 2011-01-11 |
| ZA200806407B (en) | 2009-04-29 |
| CN101415711A (zh) | 2009-04-22 |
| EP2013215A4 (en) | 2010-09-08 |
| CL2009000523A1 (es) | 2009-07-17 |
| BRPI0707423A2 (pt) | 2011-05-03 |
| RU2421457C2 (ru) | 2011-06-20 |
| NO20083547L (no) | 2008-11-05 |
| WO2007091947A3 (en) | 2007-10-04 |
| SG169387A1 (en) | 2011-03-30 |
| KR20080094906A (ko) | 2008-10-27 |
| JP2009526043A (ja) | 2009-07-16 |
| TW200801011A (en) | 2008-01-01 |
| UY30132A1 (es) | 2009-07-17 |
| CA2641632A1 (en) | 2007-08-16 |
| US20090137650A1 (en) | 2009-05-28 |
| AR059265A1 (es) | 2008-03-19 |
| WO2007091947A2 (en) | 2007-08-16 |
| UA93226C2 (en) | 2011-01-25 |
| US20070185179A1 (en) | 2007-08-09 |
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