RU99100084A - Применение ингибиторов клеточного натрий-водородного обмена для получения лекарственного средства для нормализации уровня липидов сыворотки - Google Patents
Применение ингибиторов клеточного натрий-водородного обмена для получения лекарственного средства для нормализации уровня липидов сывороткиInfo
- Publication number
- RU99100084A RU99100084A RU99100084/14A RU99100084A RU99100084A RU 99100084 A RU99100084 A RU 99100084A RU 99100084/14 A RU99100084/14 A RU 99100084/14A RU 99100084 A RU99100084 A RU 99100084A RU 99100084 A RU99100084 A RU 99100084A
- Authority
- RU
- Russia
- Prior art keywords
- normalization
- application
- serum lipids
- metabolism inhibitors
- cellular sodium
- Prior art date
Links
- 230000036740 Metabolism Effects 0.000 title 1
- 210000002966 Serum Anatomy 0.000 title 1
- 230000001413 cellular Effects 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 150000002632 lipids Chemical class 0.000 title 1
- 230000004060 metabolic process Effects 0.000 title 1
- 230000035786 metabolism Effects 0.000 title 1
- XONPDZSGENTBNJ-UHFFFAOYSA-N molecular hydrogen;sodium Chemical compound [Na].[H][H] XONPDZSGENTBNJ-UHFFFAOYSA-N 0.000 title 1
- 238000010606 normalization Methods 0.000 title 1
Images
Claims (1)
- Текст формулы заявки в факсимильном виде (см. чертижи).
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19622222.2 | 1996-06-03 | ||
DE19622222A DE19622222A1 (de) | 1996-06-03 | 1996-06-03 | Verwendung von Inhibitoren des zellulären Na·+·/H·+·-Exchangers (NHE) zur Herstellung eines Medikament zur Normalisierung der Serumlipide |
DE19712636A DE19712636A1 (de) | 1997-03-26 | 1997-03-26 | Verwendung von Inhibitoren des zellulären Na+/H+Exchangers (NHE) zur Herstellung eines Medikament zur Normalisierung der Serumlipide |
DE19712636.7 | 1997-03-26 |
Publications (2)
Publication Number | Publication Date |
---|---|
RU99100084A true RU99100084A (ru) | 2000-11-10 |
RU2211032C2 RU2211032C2 (ru) | 2003-08-27 |
Family
ID=26026256
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU99100084/14A RU2211032C2 (ru) | 1996-06-03 | 1997-05-20 | Применение ингибиторов клеточного натрий-водородного обмена для получения лекарственного средства для нормализации уровня липидов сыворотки |
Country Status (23)
Country | Link |
---|---|
EP (1) | EP0918515B1 (ru) |
JP (1) | JP4527811B2 (ru) |
KR (1) | KR100511711B1 (ru) |
CN (1) | CN1221339A (ru) |
AR (1) | AR007353A1 (ru) |
AT (1) | ATE293965T1 (ru) |
AU (1) | AU722166B2 (ru) |
BR (1) | BR9709516A (ru) |
CA (1) | CA2257299A1 (ru) |
DE (2) | DE19622222A1 (ru) |
DK (1) | DK0918515T3 (ru) |
ES (1) | ES2241049T3 (ru) |
IL (1) | IL126935A0 (ru) |
NO (1) | NO985480L (ru) |
NZ (1) | NZ333095A (ru) |
PL (1) | PL189950B1 (ru) |
PT (1) | PT918515E (ru) |
RU (1) | RU2211032C2 (ru) |
SI (1) | SI0918515T1 (ru) |
SK (1) | SK165898A3 (ru) |
TR (1) | TR199802505T2 (ru) |
WO (1) | WO1997046226A2 (ru) |
ZA (1) | ZA974828B (ru) |
Families Citing this family (37)
Publication number | Priority date | Publication date | Assignee | Title |
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US6011059A (en) * | 1997-12-24 | 2000-01-04 | Bristol-Myers Squibb Company | Acyl guanidine sodium/proton exchange inhibitors and method |
US6160134A (en) * | 1997-12-24 | 2000-12-12 | Bristol-Myers Squibb Co. | Process for preparing chiral cyclopropane carboxylic acids and acyl guanidines |
DE19859727A1 (de) * | 1998-12-23 | 2000-06-29 | Aventis Pharma Gmbh | Die Verwendung von Hemmern des Natrium-Wasserstoff-Austauschers zur Herstellung eines Medikaments zur Verhinderung von altersbedingten Organ-Dysfunktionen, altersbedingten Erkrankungen zur Lebensverlängerung |
CA2370607A1 (en) | 1999-04-23 | 2000-11-02 | Bristol-Myers Squibb Company | Bicyclic acyl guanidine sodium/proton exchange inhibitors and method |
DE19945302A1 (de) * | 1999-09-22 | 2001-03-29 | Merck Patent Gmbh | Biphenylderivate als NHE-3-Inhibitoren |
US6423705B1 (en) | 2001-01-25 | 2002-07-23 | Pfizer Inc. | Combination therapy |
AU2002348276A1 (en) | 2001-11-16 | 2003-06-10 | Bristol-Myers Squibb Company | Dual inhibitors of adipocyte fatty acid binding protein and keratinocyte fatty acid binding protein |
US7230007B2 (en) | 2003-06-12 | 2007-06-12 | Sanofi-Aventis Deutschland Gmbh | Derivatives of 3-(Guanidinocarbonyl) heterocycle, methods of preparation and intermediates thereof, their use as medicaments, and pharmaceutical compositions therefrom |
FR2856062B1 (fr) * | 2003-06-12 | 2005-11-11 | Aventis Pharma Sa | Derives 3-guanidinocarbonyl-heterocycle, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant |
EP1646371A4 (en) * | 2003-06-26 | 2010-09-22 | Biotron Ltd | ANTIVIRAL COMPOSITIONS AND METHODS |
US7371759B2 (en) | 2003-09-25 | 2008-05-13 | Bristol-Myers Squibb Company | HMG-CoA reductase inhibitors and method |
US7420059B2 (en) | 2003-11-20 | 2008-09-02 | Bristol-Myers Squibb Company | HMG-CoA reductase inhibitors and method |
US7572805B2 (en) | 2004-07-14 | 2009-08-11 | Bristol-Myers Squibb Company | Pyrrolo(oxo)isoquinolines as 5HT ligands |
US7517991B2 (en) | 2004-10-12 | 2009-04-14 | Bristol-Myers Squibb Company | N-sulfonylpiperidine cannabinoid receptor 1 antagonists |
US7314882B2 (en) | 2005-01-12 | 2008-01-01 | Bristol-Myers Squibb Company | Bicyclic heterocycles as cannabinoid receptor modulators |
WO2006076569A2 (en) | 2005-01-12 | 2006-07-20 | Bristol-Myers Squibb Company | Bicyclic heterocycles as cannabinoid receptor modulators |
US20060160850A1 (en) | 2005-01-18 | 2006-07-20 | Chongqing Sun | Bicyclic heterocycles as cannabinoid receptor modulators |
ATE421518T1 (de) | 2005-02-10 | 2009-02-15 | Bristol Myers Squibb Co | Dihydrochinazolinone als 5ht-modulatoren |
US7452892B2 (en) | 2005-06-17 | 2008-11-18 | Bristol-Myers Squibb Company | Triazolopyrimidine cannabinoid receptor 1 antagonists |
US7632837B2 (en) | 2005-06-17 | 2009-12-15 | Bristol-Myers Squibb Company | Bicyclic heterocycles as cannabinoid-1 receptor modulators |
TW200726765A (en) | 2005-06-17 | 2007-07-16 | Bristol Myers Squibb Co | Triazolopyridine cannabinoid receptor 1 antagonists |
US7317012B2 (en) | 2005-06-17 | 2008-01-08 | Bristol-Myers Squibb Company | Bicyclic heterocycles as cannabinoind-1 receptor modulators |
US7629342B2 (en) | 2005-06-17 | 2009-12-08 | Bristol-Myers Squibb Company | Azabicyclic heterocycles as cannabinoid receptor modulators |
US7795436B2 (en) | 2005-08-24 | 2010-09-14 | Bristol-Myers Squibb Company | Substituted tricyclic heterocycles as serotonin receptor agonists and antagonists |
AR056155A1 (es) | 2005-10-26 | 2007-09-19 | Bristol Myers Squibb Co | Antagonistas del receptor 1 de la hormona de concentracion de melanina no basica |
US7553836B2 (en) | 2006-02-06 | 2009-06-30 | Bristol-Myers Squibb Company | Melanin concentrating hormone receptor-1 antagonists |
US20090011994A1 (en) | 2007-07-06 | 2009-01-08 | Bristol-Myers Squibb Company | Non-basic melanin concentrating hormone receptor-1 antagonists and methods |
PE20091928A1 (es) | 2008-05-29 | 2009-12-31 | Bristol Myers Squibb Co | Tienopirimidinas hidroxisustituidas como antagonistas de receptor-1 de hormona concentradora de melanina no basicos |
US10517839B2 (en) | 2008-06-09 | 2019-12-31 | Cornell University | Mast cell inhibition in diseases of the retina and vitreous |
AU2010229653A1 (en) | 2009-03-27 | 2011-10-20 | Astrazeneca Ab | Methods for preventing major adverse cardiovascular events with DPP-IV inhibitors |
AU2011210765A1 (en) | 2010-01-28 | 2012-09-13 | President And Fellows Of Harvard College | Compositions and methods for enhancing proteasome activity |
ES2724531T3 (es) | 2011-05-12 | 2019-09-11 | Proteostasis Therapeutics Inc | Reguladores de proteostasis |
EP2892897A1 (en) | 2012-09-05 | 2015-07-15 | Bristol-Myers Squibb Company | Pyrrolone or pyrrolidinone melanin concentrating hormone receptor-1 antagonists |
EP2892896B1 (en) | 2012-09-05 | 2016-06-29 | Bristol-Myers Squibb Company | Pyrrolone or pyrrolidinone melanin concentrating hormore receptor-1 antagonists |
WO2014116228A1 (en) | 2013-01-25 | 2014-07-31 | President And Fellows Of Harvard College | Usp14 inhibitors for treating or preventing viral infections |
WO2015073528A1 (en) | 2013-11-12 | 2015-05-21 | Proteostasis Therapeutics, Inc. | Proteasome activity enhancing compounds |
EP3823631A1 (en) | 2018-07-19 | 2021-05-26 | Astrazeneca AB | Methods of treating hfpef employing dapagliflozin and compositions comprising the same |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5110817A (en) * | 1988-10-21 | 1992-05-05 | Beyer Jr Karl H | Method for controlling and/or lowering serum triglyceride and/or cholesterol levels in mammals |
US4920123A (en) * | 1988-10-21 | 1990-04-24 | Beyer Jr Karl H | Method for controlling and/or lowering serum triglyceride and/or cholesterol levels in mammals |
AU7316591A (en) * | 1990-02-28 | 1991-09-18 | Upjohn Company, The | Use of 3-guanidinopropionic acid in the treatment and prevention of metabolic disorders |
ATE157351T1 (de) * | 1993-02-20 | 1997-09-15 | Hoechst Ag | Substituierte benzoylguanidine, verfahren zu ihrer herstellung, ihre verwendung als medikament, als inhibitoren des zellulären na+/h+-austauschs oder als diagnostikum sowie sie enthaltendes medikament |
DE4318658A1 (de) * | 1993-06-04 | 1994-12-08 | Hoechst Ag | Substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
DE4325822A1 (de) * | 1993-07-31 | 1995-02-02 | Hoechst Ag | Substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
IL114670A0 (en) * | 1994-08-05 | 1995-11-27 | Fujisawa Pharmaceutical Co | Guanidine derivatives pharmaceutical compositions containing the same and processes for the preparation thereof |
-
1996
- 1996-06-03 DE DE19622222A patent/DE19622222A1/de not_active Withdrawn
-
1997
- 1997-05-20 JP JP50014498A patent/JP4527811B2/ja not_active Expired - Fee Related
- 1997-05-20 WO PCT/EP1997/002548 patent/WO1997046226A2/de not_active Application Discontinuation
- 1997-05-20 AU AU29576/97A patent/AU722166B2/en not_active Ceased
- 1997-05-20 AT AT97923937T patent/ATE293965T1/de not_active IP Right Cessation
- 1997-05-20 EP EP97923937A patent/EP0918515B1/de not_active Expired - Lifetime
- 1997-05-20 SI SI9730705T patent/SI0918515T1/sl unknown
- 1997-05-20 RU RU99100084/14A patent/RU2211032C2/ru not_active IP Right Cessation
- 1997-05-20 CA CA002257299A patent/CA2257299A1/en not_active Abandoned
- 1997-05-20 BR BR9709516A patent/BR9709516A/pt not_active Application Discontinuation
- 1997-05-20 ES ES97923937T patent/ES2241049T3/es not_active Expired - Lifetime
- 1997-05-20 IL IL12693597A patent/IL126935A0/xx not_active IP Right Cessation
- 1997-05-20 TR TR1998/02505T patent/TR199802505T2/xx unknown
- 1997-05-20 SK SK1658-98A patent/SK165898A3/sk unknown
- 1997-05-20 PL PL97330412A patent/PL189950B1/pl not_active IP Right Cessation
- 1997-05-20 DE DE59712287T patent/DE59712287D1/de not_active Expired - Lifetime
- 1997-05-20 KR KR10-1998-0709811A patent/KR100511711B1/ko not_active IP Right Cessation
- 1997-05-20 DK DK97923937T patent/DK0918515T3/da active
- 1997-05-20 PT PT97923937T patent/PT918515E/pt unknown
- 1997-05-20 NZ NZ333095A patent/NZ333095A/xx unknown
- 1997-05-20 CN CN97195194A patent/CN1221339A/zh active Pending
- 1997-05-30 AR ARP970102344A patent/AR007353A1/es unknown
- 1997-06-02 ZA ZA9704828A patent/ZA974828B/xx unknown
-
1998
- 1998-11-24 NO NO985480A patent/NO985480L/no not_active Application Discontinuation
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