RU2666899C2 - Производные пиридазинон-амидов - Google Patents

Производные пиридазинон-амидов Download PDF

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RU2666899C2
RU2666899C2 RU2015137757A RU2015137757A RU2666899C2 RU 2666899 C2 RU2666899 C2 RU 2666899C2 RU 2015137757 A RU2015137757 A RU 2015137757A RU 2015137757 A RU2015137757 A RU 2015137757A RU 2666899 C2 RU2666899 C2 RU 2666899C2
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Russia
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disease
formula
compound
syndrome
pyridazin
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RU2015137757A
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Russian (ru)
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RU2015137757A (ru
Inventor
Катрин Жоран-Лебрюн
Сантош КУЛКАРНИ
Стефано ГРОСИНЬЯНИ
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Мерк Патент Гмбх
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    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • C—CHEMISTRY; METALLURGY
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Neurology (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Oncology (AREA)
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RU2015137757A 2013-02-07 2014-02-06 Производные пиридазинон-амидов RU2666899C2 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13154390.2 2013-02-07
EP13154390 2013-02-07
PCT/EP2014/000316 WO2014121931A1 (en) 2013-02-07 2014-02-06 Pyridazinone-amides derivatives

Publications (2)

Publication Number Publication Date
RU2015137757A RU2015137757A (ru) 2017-03-13
RU2666899C2 true RU2666899C2 (ru) 2018-09-13

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RU2015137757A RU2666899C2 (ru) 2013-02-07 2014-02-06 Производные пиридазинон-амидов

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US (2) US9567320B2 (cg-RX-API-DMAC7.html)
EP (1) EP2953944B1 (cg-RX-API-DMAC7.html)
JP (1) JP6483624B2 (cg-RX-API-DMAC7.html)
KR (1) KR102293952B1 (cg-RX-API-DMAC7.html)
CN (1) CN104968658B (cg-RX-API-DMAC7.html)
AU (1) AU2014214321B2 (cg-RX-API-DMAC7.html)
BR (1) BR112015018663A2 (cg-RX-API-DMAC7.html)
CA (1) CA2900431C (cg-RX-API-DMAC7.html)
DK (1) DK2953944T3 (cg-RX-API-DMAC7.html)
ES (1) ES2634627T3 (cg-RX-API-DMAC7.html)
HR (1) HRP20171076T1 (cg-RX-API-DMAC7.html)
HU (1) HUE032863T2 (cg-RX-API-DMAC7.html)
IL (1) IL240290B (cg-RX-API-DMAC7.html)
LT (1) LT2953944T (cg-RX-API-DMAC7.html)
MX (1) MX364486B (cg-RX-API-DMAC7.html)
PL (1) PL2953944T3 (cg-RX-API-DMAC7.html)
PT (1) PT2953944T (cg-RX-API-DMAC7.html)
RS (1) RS56331B1 (cg-RX-API-DMAC7.html)
RU (1) RU2666899C2 (cg-RX-API-DMAC7.html)
SG (1) SG11201506100XA (cg-RX-API-DMAC7.html)
SI (1) SI2953944T1 (cg-RX-API-DMAC7.html)
WO (1) WO2014121931A1 (cg-RX-API-DMAC7.html)

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CN113750094A (zh) 2015-04-22 2021-12-07 里格尔药品股份有限公司 吡唑化合物以及制备和使用该化合物的方法
WO2017049068A1 (en) * 2015-09-18 2017-03-23 Merck Patent Gmbh Heteroaryl compounds as irak inhibitors and uses thereof
CA3002560A1 (en) 2015-10-23 2017-04-27 Array Biopharma, Inc. 2-aryl- and 2-heteroaryl-substituted 2-pyridazin-3(2h)-one compounds as inhibitors of fgfr tyrosine kinases
JOP20180011A1 (ar) 2017-02-16 2019-01-30 Gilead Sciences Inc مشتقات بيرولو [1، 2-b]بيريدازين
WO2019060693A1 (en) 2017-09-22 2019-03-28 Kymera Therapeutics, Inc. CRBN LIGANDS AND USES THEREOF
JP7366031B2 (ja) 2017-09-22 2023-10-20 カイメラ セラピューティクス， インコーポレイテッド タンパク質分解剤およびそれらの使用
WO2019111218A1 (en) 2017-12-08 2019-06-13 Cadila Healthcare Limited Novel heterocyclic compounds as irak4 inhibitors
IL315310A (en) 2017-12-26 2024-10-01 Kymera Therapeutics Inc Irak degraders and uses thereof
WO2019140380A1 (en) 2018-01-12 2019-07-18 Kymera Therapeutics, Inc. Protein degraders and uses thereof
WO2019140387A1 (en) 2018-01-12 2019-07-18 Kymera Therapeutics, Inc. Crbn ligands and uses thereof
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