RU2599846C2 - Новые и эффективные лекарственые формы тапентадола - Google Patents

Новые и эффективные лекарственые формы тапентадола Download PDF

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RU2599846C2
RU2599846C2 RU2011121513/15A RU2011121513A RU2599846C2 RU 2599846 C2 RU2599846 C2 RU 2599846C2 RU 2011121513/15 A RU2011121513/15 A RU 2011121513/15A RU 2011121513 A RU2011121513 A RU 2011121513A RU 2599846 C2 RU2599846 C2 RU 2599846C2
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Russia
Prior art keywords
tapentadol
naltrexone
pharmaceutically acceptable
combination
acceptable salt
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RU2011121513/15A
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English (en)
Russian (ru)
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RU2011121513A (ru
Inventor
СЕША Рамеш
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Грюненталь Гмбх
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42634123&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RU2599846(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Грюненталь Гмбх filed Critical Грюненталь Гмбх
Publication of RU2011121513A publication Critical patent/RU2011121513A/ru
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    • A—HUMAN NECESSITIES
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    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
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    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Otolaryngology (AREA)
  • Transplantation (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
RU2011121513/15A 2008-10-30 2009-10-29 Новые и эффективные лекарственые формы тапентадола RU2599846C2 (ru)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US19762508P 2008-10-30 2008-10-30
US61/197,625 2008-10-30
US20531209P 2009-01-21 2009-01-21
US61/205,312 2009-01-21
US26863009P 2009-06-15 2009-06-15
US61/268,630 2009-06-15
PCT/US2009/005866 WO2010096045A1 (en) 2008-10-30 2009-10-29 Novel and potent tapentadol dosage forms

Related Child Applications (1)

Application Number Title Priority Date Filing Date
RU2015154026A Division RU2673882C1 (ru) 2008-10-30 2009-10-29 Новые и эффективные лекарственные формы тапентадола

Publications (2)

Publication Number Publication Date
RU2011121513A RU2011121513A (ru) 2012-12-10
RU2599846C2 true RU2599846C2 (ru) 2016-10-20

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ID=42634123

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RU2011121513/15A RU2599846C2 (ru) 2008-10-30 2009-10-29 Новые и эффективные лекарственые формы тапентадола
RU2015154026A RU2673882C1 (ru) 2008-10-30 2009-10-29 Новые и эффективные лекарственные формы тапентадола

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RU2015154026A RU2673882C1 (ru) 2008-10-30 2009-10-29 Новые и эффективные лекарственные формы тапентадола

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US (1) US9642801B2 (cg-RX-API-DMAC7.html)
EP (1) EP2352494B1 (cg-RX-API-DMAC7.html)
JP (2) JP6216489B2 (cg-RX-API-DMAC7.html)
KR (2) KR101712339B1 (cg-RX-API-DMAC7.html)
CN (2) CN104257600A (cg-RX-API-DMAC7.html)
AU (2) AU2009340504A1 (cg-RX-API-DMAC7.html)
BR (1) BRPI0921725A2 (cg-RX-API-DMAC7.html)
CA (1) CA2741984C (cg-RX-API-DMAC7.html)
CL (1) CL2011000967A1 (cg-RX-API-DMAC7.html)
CO (1) CO6382115A2 (cg-RX-API-DMAC7.html)
CY (1) CY1122269T1 (cg-RX-API-DMAC7.html)
DK (1) DK2352494T3 (cg-RX-API-DMAC7.html)
EC (2) ECSP11011016A (cg-RX-API-DMAC7.html)
ES (1) ES2758831T3 (cg-RX-API-DMAC7.html)
HR (1) HRP20191909T1 (cg-RX-API-DMAC7.html)
HU (1) HUE047438T2 (cg-RX-API-DMAC7.html)
IL (2) IL212523A0 (cg-RX-API-DMAC7.html)
LT (1) LT2352494T (cg-RX-API-DMAC7.html)
MX (1) MX2011004455A (cg-RX-API-DMAC7.html)
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PE (3) PE20110390A1 (cg-RX-API-DMAC7.html)
PL (1) PL2352494T3 (cg-RX-API-DMAC7.html)
PT (1) PT2352494T (cg-RX-API-DMAC7.html)
RU (2) RU2599846C2 (cg-RX-API-DMAC7.html)
SI (1) SI2352494T1 (cg-RX-API-DMAC7.html)
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Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2009340504A1 (en) 2008-10-30 2010-08-26 Grunenthal Gmbh Novel and potent tapentadol dosage forms
LT2424514T (lt) * 2009-04-30 2017-04-25 Grünenthal GmbH Tapentadolis reumatoidinio artrito skausmo gydymui
US10363251B2 (en) 2009-07-16 2019-07-30 Mallinckrodt Llc (+)-morphinans as antagonists of toll-like receptor 9 and therapeutic uses thereof
US20130116333A1 (en) * 2010-05-05 2013-05-09 Ratiopharm Gmbh Solid tapentadol in non-crystalline form
US9700508B2 (en) 2010-05-10 2017-07-11 Euro-Celtique S.A. Pharmaceutical compositions comprising hydromorphone and naloxone
US9993433B2 (en) 2010-05-10 2018-06-12 Euro-Celtique S.A. Manufacturing of active-free granules and tablets comprising the same
NZ603170A (en) 2010-05-10 2015-04-24 Euro Celtique Sa Combination of active loaded granules with additional actives
PL2593095T3 (pl) 2010-07-16 2019-12-31 Mallinckrodt Llc (+)-morfinany jako antagoniści receptora toll-podobnego 9 i ich terapeutyczne zastosowania
DK3656765T3 (da) * 2010-07-23 2021-06-14 Gruenenthal Gmbh Salte eller co-krystaller af 3-(3-dimethylamin-1-ethyl-2-methyl-propyl)-phenol
WO2012051246A1 (en) * 2010-10-12 2012-04-19 Ratiopharm Gmbh Tapentadol hydrobromide and crystalline forms thereof
BR112013022556A8 (pt) * 2011-03-04 2018-01-16 Gruenenthal Gmbh composição farmacêutica aquosa semissólida contendo tapentadol, seu uso e uso de tapentadol
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