RU2549899C2 - Кристаллические формы гидрохлорида финголимода - Google Patents
Кристаллические формы гидрохлорида финголимода Download PDFInfo
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- RU2549899C2 RU2549899C2 RU2011123371/04A RU2011123371A RU2549899C2 RU 2549899 C2 RU2549899 C2 RU 2549899C2 RU 2011123371/04 A RU2011123371/04 A RU 2011123371/04A RU 2011123371 A RU2011123371 A RU 2011123371A RU 2549899 C2 RU2549899 C2 RU 2549899C2
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- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2627691C1 (ru) * | 2016-07-06 | 2017-08-10 | Олег Ростиславович Михайлов | Кристаллическая η-модификация 2-амино-2-(2-(4-октилфенил)этил)пропан-1,3-диол гидрохлорида, способ её получения и фармацевтическая композиция на её основе |
| RU2663833C2 (ru) * | 2013-03-05 | 2018-08-10 | Биокон Лимитед | Способ получения соединений 2-амино-1,3-пропандиола и их солей |
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| EP2621889B1 (en) | 2010-10-01 | 2019-07-17 | Synthon BV | Process for making fingolimod hydrochloride crystals |
| PL2632889T3 (pl) | 2010-10-28 | 2019-04-30 | Mapi Pharma Ltd | Związki pośrednie i sposób wytwarzania fingolimodu |
| WO2012071524A1 (en) | 2010-11-24 | 2012-05-31 | Ratiopharm Gmbh | Arylsulfonate salts of fingolimod and processes for preparation thereof |
| US9266816B2 (en) | 2010-11-25 | 2016-02-23 | Shilpa Medicare Limited | Fingolimod polymorphs and their processes |
| EP2658840B1 (en) | 2010-12-28 | 2019-07-03 | Synthon BV | Process for making fingolimod hydrochloride crystals |
| WO2012097330A2 (en) * | 2011-01-14 | 2012-07-19 | University Of Washington | Compositions and methods for treating degenerative muscle conditions |
| EP2702034A4 (en) | 2011-04-29 | 2015-03-25 | Reddys Lab Ltd Dr | PREPARATION OF FINGOLIMOD AND ITS SALTS |
| US9751834B2 (en) | 2011-05-26 | 2017-09-05 | Gri Bio, Inc. | Oxygenated amino- or ammonium-containing sulfonic acid, phosphonic acid and carboxylic acid derivatives and their medical use |
| EP2739606B1 (en) | 2011-05-26 | 2016-04-27 | Jado Technologies GmbH | Hydroxy-substituted amino and ammonium derivatives and their medical use |
| DK2809318T3 (da) | 2011-05-26 | 2019-07-22 | Gri Bio Inc | Ammoniumholdige sulfonsyre-, phosphonsyre- og carboxylsyrederivater og disses medicinske anvendelse |
| WO2013019872A1 (en) | 2011-08-01 | 2013-02-07 | Teva Pharmaceutical Industries Ltd. | Process for preparing pharmaceutical compositions comprising fingolimod |
| WO2013091704A1 (en) * | 2011-12-22 | 2013-06-27 | Synthon Bv | Pharmaceutical composition comprising fingolimod |
| CN102887829B (zh) * | 2012-09-05 | 2014-07-02 | 中国科学院上海药物研究所 | 芬戈莫德粘酸盐及其晶体的制备方法和用途 |
| EP2945927A4 (en) * | 2013-01-17 | 2017-01-18 | Shilpa Medicare Limited | Process for preparation of fingolimod and its salts |
| EP3027174B1 (en) | 2013-07-29 | 2019-07-24 | Aizant Drug Research Solutions Private Limited | Pharmaceutical compositions of fingolimod |
| WO2016042493A1 (en) * | 2014-09-19 | 2016-03-24 | Aizant Drug Research Pvt. Ltd | Pharmaceutical compositions of fingolimod |
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| RU2663833C2 (ru) * | 2013-03-05 | 2018-08-10 | Биокон Лимитед | Способ получения соединений 2-амино-1,3-пропандиола и их солей |
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| WO2010055028A3 (en) | 2010-07-08 |
| WO2010055028A2 (en) | 2010-05-20 |
| EP2356090A2 (en) | 2011-08-17 |
| ES2643161T3 (es) | 2017-11-21 |
| AU2009315736A1 (en) | 2010-05-20 |
| PL2356090T3 (pl) | 2017-12-29 |
| US20110229501A1 (en) | 2011-09-22 |
| JP2014139179A (ja) | 2014-07-31 |
| JP2016028056A (ja) | 2016-02-25 |
| KR101393994B1 (ko) | 2014-05-14 |
| PT2356090T (pt) | 2017-10-16 |
| AU2009315736B2 (en) | 2013-08-29 |
| RU2011123371A (ru) | 2012-12-20 |
| JP2012508216A (ja) | 2012-04-05 |
| CA2743232C (en) | 2015-12-29 |
| JP2018035160A (ja) | 2018-03-08 |
| CN104788325A (zh) | 2015-07-22 |
| BRPI0921826A2 (pt) | 2016-01-12 |
| KR20130109254A (ko) | 2013-10-07 |
| CN107233336A (zh) | 2017-10-10 |
| US8530522B2 (en) | 2013-09-10 |
| CN102209705A (zh) | 2011-10-05 |
| MX2011004962A (es) | 2011-05-30 |
| RU2015111229A3 (https=) | 2018-11-08 |
| US20140051766A1 (en) | 2014-02-20 |
| CA2743232A1 (en) | 2010-05-20 |
| RU2015111229A (ru) | 2015-11-20 |
| EP2356090B1 (en) | 2017-07-05 |
| KR20110069156A (ko) | 2011-06-22 |
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