RU2476432C2 - 6-, 7- или 8-замещенные производные хиназолинона и композиции, включающие их, и способы их использования - Google Patents

6-, 7- или 8-замещенные производные хиназолинона и композиции, включающие их, и способы их использования Download PDF

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RU2476432C2
RU2476432C2 RU2010116273/04A RU2010116273A RU2476432C2 RU 2476432 C2 RU2476432 C2 RU 2476432C2 RU 2010116273/04 A RU2010116273/04 A RU 2010116273/04A RU 2010116273 A RU2010116273 A RU 2010116273A RU 2476432 C2 RU2476432 C2 RU 2476432C2
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mmol
methyl
optionally substituted
alkyl
oxo
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RU2010116273/04A
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RU2010116273A (ru
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Джордж В. Мюллер
Хон-Вах МАН
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Селджин Корпорейшн
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Anesthesiology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
RU2010116273/04A 2007-09-26 2008-09-25 6-, 7- или 8-замещенные производные хиназолинона и композиции, включающие их, и способы их использования RU2476432C2 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US99567607P 2007-09-26 2007-09-26
US60/995,676 2007-09-26
PCT/US2008/011124 WO2009042177A1 (en) 2007-09-26 2008-09-25 6-, 7-, or 8-substituted quinazolinone derivatives and compositions comprising and methods of using the same

Publications (2)

Publication Number Publication Date
RU2010116273A RU2010116273A (ru) 2011-11-10
RU2476432C2 true RU2476432C2 (ru) 2013-02-27

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US (5) US8492395B2 (cg-RX-API-DMAC10.html)
EP (1) EP2200999B1 (cg-RX-API-DMAC10.html)
JP (1) JP5637852B2 (cg-RX-API-DMAC10.html)
KR (1) KR101593242B1 (cg-RX-API-DMAC10.html)
CN (2) CN101952272B (cg-RX-API-DMAC10.html)
AU (1) AU2008305581C1 (cg-RX-API-DMAC10.html)
BR (1) BRPI0817525A2 (cg-RX-API-DMAC10.html)
CA (1) CA2704710C (cg-RX-API-DMAC10.html)
CO (1) CO6270228A2 (cg-RX-API-DMAC10.html)
CR (1) CR11355A (cg-RX-API-DMAC10.html)
ES (1) ES2523925T3 (cg-RX-API-DMAC10.html)
IL (2) IL204763A (cg-RX-API-DMAC10.html)
MX (1) MX347987B (cg-RX-API-DMAC10.html)
MY (1) MY157495A (cg-RX-API-DMAC10.html)
NI (1) NI201000041A (cg-RX-API-DMAC10.html)
NZ (1) NZ584425A (cg-RX-API-DMAC10.html)
RU (1) RU2476432C2 (cg-RX-API-DMAC10.html)
SG (2) SG10201503486XA (cg-RX-API-DMAC10.html)
UA (1) UA102078C2 (cg-RX-API-DMAC10.html)
WO (1) WO2009042177A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201002303B (cg-RX-API-DMAC10.html)

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