RU2472497C2 - Титрование тапентадола - Google Patents
Титрование тапентадола Download PDFInfo
- Publication number
- RU2472497C2 RU2472497C2 RU2009142940/15A RU2009142940A RU2472497C2 RU 2472497 C2 RU2472497 C2 RU 2472497C2 RU 2009142940/15 A RU2009142940/15 A RU 2009142940/15A RU 2009142940 A RU2009142940 A RU 2009142940A RU 2472497 C2 RU2472497 C2 RU 2472497C2
- Authority
- RU
- Russia
- Prior art keywords
- dose
- administration
- tapentadol
- period
- day
- Prior art date
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07008218A EP1985292A1 (en) | 2007-04-23 | 2007-04-23 | Titration of tapentadol |
| EP07008218.5 | 2007-04-23 | ||
| PCT/EP2008/003178 WO2008128740A1 (en) | 2007-04-23 | 2008-04-21 | Titration of tapentadol |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2009142940A RU2009142940A (ru) | 2011-05-27 |
| RU2472497C2 true RU2472497C2 (ru) | 2013-01-20 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2009142940/15A RU2472497C2 (ru) | 2007-04-23 | 2008-04-21 | Титрование тапентадола |
Country Status (21)
| Country | Link |
|---|---|
| US (4) | US20090012180A1 (https=) |
| EP (5) | EP1985292A1 (https=) |
| JP (4) | JP5933176B2 (https=) |
| KR (3) | KR102078999B1 (https=) |
| CN (1) | CN101730530B (https=) |
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| EP1985292A1 (en) | 2007-04-23 | 2008-10-29 | Grünenthal GmbH | Titration of tapentadol |
| RU2673882C1 (ru) * | 2008-10-30 | 2018-12-03 | Грюненталь Гмбх | Новые и эффективные лекарственные формы тапентадола |
| US8870876B2 (en) * | 2009-02-13 | 2014-10-28 | Tarsus Medical Inc. | Methods and devices for treating hallux valgus |
| US8277459B2 (en) * | 2009-09-25 | 2012-10-02 | Tarsus Medical Inc. | Methods and devices for treating a structural bone and joint deformity |
| US8652141B2 (en) | 2010-01-21 | 2014-02-18 | Tarsus Medical Inc. | Methods and devices for treating hallux valgus |
| EP2566461A2 (de) * | 2010-05-05 | 2013-03-13 | Ratiopharm GmbH | Festes tapentadol in nicht-kristalliner form |
| US8696719B2 (en) | 2010-06-03 | 2014-04-15 | Tarsus Medical Inc. | Methods and devices for treating hallux valgus |
| DK2588093T3 (en) * | 2010-06-30 | 2016-08-29 | Gruenenthal Gmbh | Tapentadol FOR USE IN THE TREATMENT OF irritable bowel syndrome |
| CN110015955A (zh) * | 2010-07-23 | 2019-07-16 | 格吕伦塔尔有限公司 | 3-(3-二甲基氨基-1-乙基-2-甲基-丙基)-苯酚的盐或共晶体 |
| CN101948397A (zh) * | 2010-09-07 | 2011-01-19 | 天津泰普药品科技发展有限公司 | 镇痛药他喷他多重要中间体的制备方法 |
| ES2910085T3 (es) | 2011-03-04 | 2022-05-11 | Gruenenthal Gmbh | Composición farmacéutica acuosa semisólida que contiene tapentadol |
| CN103501775A (zh) * | 2011-03-04 | 2014-01-08 | 格吕伦塔尔有限公司 | 他喷他多的胃肠外给药 |
| MX388963B (es) | 2011-03-04 | 2025-03-20 | Gruenenthal Gmbh | Formulacion farmaceutica acuosa de tapentadol para administracion oral |
| EP3607943B1 (en) * | 2011-04-05 | 2024-09-11 | Grünenthal GmbH | Tapentadol for use in treating pain associated with trigeminal neuralgia |
| ES2703282T3 (es) | 2011-04-05 | 2019-03-07 | Gruenenthal Gmbh | Tapentadol para prevenir la cronificación del dolor |
| US20120277319A1 (en) | 2011-04-29 | 2012-11-01 | Gruenenthal Gmbh | Use of Tapentadol for Inhibiting and/or Treating Depression and Anxiety |
| CA2901802C (en) * | 2013-03-15 | 2021-03-02 | Mallinckrodt Llc | Abuse deterrent solid dosage form for immediate release with functional score |
| EP2845625A1 (en) * | 2013-09-04 | 2015-03-11 | Grünenthal GmbH | Tapentadol for use in the treatment of fibromyalgia and chronic fatigue syndrome |
| PE20171651A1 (es) | 2015-03-27 | 2017-11-13 | Gruenenthal Chemie | Formulacion estable para administracion parenteral de tapentadol |
| PT3302454T (pt) * | 2015-05-26 | 2021-04-01 | Technophage Investig E Desenvolvimento Em Biotecnologia Sa | Composições para utilização no tratamento da doença de parkinson e distúrbios associados |
| JP7373904B2 (ja) * | 2016-02-29 | 2023-11-06 | パーク・セラピューティクス・インコーポレイテッド | セブラノパドールの滴定 |
| EP3515412B1 (en) | 2016-09-23 | 2025-04-23 | Grünenthal GmbH | Stable formulation for parenteral administration of tapentadol |
| ES3010208T3 (en) | 2020-03-16 | 2025-04-01 | Gruenenthal Gmbh | Scored tablet comprising tapentadol |
| WO2022194941A1 (en) * | 2021-03-17 | 2022-09-22 | Actelion Pharmaceuticals Ltd | Pharmaceutical dosage system |
| EP4333820A1 (en) * | 2021-05-07 | 2024-03-13 | Grünenthal GmbH | Tapentadol for treating neuropathic pain in covid-19 patients |
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| RU2150465C1 (ru) * | 1994-07-23 | 2000-06-10 | Грюненталь Гмбх | 1-фенил-3-диметиламино-пропановые соединения, способ их получения (варианты) и болеутоляющее лекарственное средство |
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| US4783337A (en) | 1983-05-11 | 1988-11-08 | Alza Corporation | Osmotic system comprising plurality of members for dispensing drug |
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| DE102007019417A1 (de) | 2007-04-23 | 2008-11-13 | Grünenthal GmbH | Tapentadol zur Schmerzbehandlung bei Arthrose |
| EP1985292A1 (en) * | 2007-04-23 | 2008-10-29 | Grünenthal GmbH | Titration of tapentadol |
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