RU2296763C2 - Амид 8-амино-[1.2.4]триазоло-[1.5-а]пиридин-6-карбоновой кислоты и содержащее его лекарственное средство - Google Patents

Амид 8-амино-[1.2.4]триазоло-[1.5-а]пиридин-6-карбоновой кислоты и содержащее его лекарственное средство Download PDF

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RU2296763C2
RU2296763C2 RU2004114278/04A RU2004114278A RU2296763C2 RU 2296763 C2 RU2296763 C2 RU 2296763C2 RU 2004114278/04 A RU2004114278/04 A RU 2004114278/04A RU 2004114278 A RU2004114278 A RU 2004114278A RU 2296763 C2 RU2296763 C2 RU 2296763C2
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amino
triazolo
pyridin
bromofuran
formula
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RU2004114278/04A
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Russian (ru)
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RU2004114278A (ru
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Маттиас Генрих НЕТТЕКОВЕН (DE)
Маттиас Генрих Неттековен
Себастьен ШМИТТ (FR)
Себастьен ШМИТТ
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Ф.Хоффманн-Ля Рош Аг
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P25/00—Drugs for disorders of the nervous system
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Psychology (AREA)
  • Immunology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Addiction (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
RU2004114278/04A 2001-10-08 2002-10-04 Амид 8-амино-[1.2.4]триазоло-[1.5-а]пиридин-6-карбоновой кислоты и содержащее его лекарственное средство RU2296763C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01123948 2001-10-08
EP01123948.0 2001-10-08

Publications (2)

Publication Number Publication Date
RU2004114278A RU2004114278A (ru) 2005-10-27
RU2296763C2 true RU2296763C2 (ru) 2007-04-10

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RU2004114278/04A RU2296763C2 (ru) 2001-10-08 2002-10-04 Амид 8-амино-[1.2.4]триазоло-[1.5-а]пиридин-6-карбоновой кислоты и содержащее его лекарственное средство

Country Status (13)

Country Link
US (1) US6689790B2 (enExample)
EP (1) EP1435952A1 (enExample)
JP (1) JP4101755B2 (enExample)
KR (1) KR100614486B1 (enExample)
CN (1) CN1564686A (enExample)
AR (1) AR036734A1 (enExample)
AU (1) AU2002347055B2 (enExample)
BR (1) BR0213172A (enExample)
CA (1) CA2462806A1 (enExample)
MX (1) MXPA04003277A (enExample)
PL (1) PL370067A1 (enExample)
RU (1) RU2296763C2 (enExample)
WO (1) WO2003030904A1 (enExample)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2538963C2 (ru) * 2009-07-17 2015-01-10 Джапан Тобакко Инк. Триазолопиридиновое соединение и его действие в качестве ингибитора пролилгидроксилазы и индуктора выработки эритропоэтина
RU2552642C2 (ru) * 2008-09-08 2015-06-10 СИГНАЛ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи Аминотриазолопиридины и их применение в качестве ингибиторов киназ
RU2620379C2 (ru) * 2012-02-09 2017-05-25 Ф.Хоффманн-Ля Рош Аг СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ 2-ФЕНИЛ[1,2,4]ТРИАЗОЛО[1,5-а]ПИРИДИНА
RU2681941C2 (ru) * 2013-05-31 2019-03-14 Ниссан Кемикал Индастриз, Лтд. Гетероциклическое амидное соединение

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2009259853A1 (en) * 2008-06-20 2009-12-23 Genentech, Inc. Triazolopyridine JAK inhibitor compounds and methods
EP2296475A4 (en) * 2008-06-20 2014-03-05 Genentech Inc TRIAZOLOPYRIDINE COMPOUNDS JAK KINASE INHIBITORS AND METHODS
US9048427B2 (en) * 2013-03-06 2015-06-02 National Tsing Hua University Thin film fabrication of rubber material with piezoelectric characteristics
CN104370807B (zh) * 2014-11-13 2016-10-05 安徽星宇化工有限公司 一种6-羟基-5-硝基烟酸的合成方法及其分离提纯方法
CA3095839A1 (en) 2018-04-08 2019-10-17 Beigene, Ltd. Pyrazolotriazolopyrimidine derivatives as a2a receptor antagonist
CN110742893B (zh) * 2018-07-23 2024-04-05 百济神州(北京)生物科技有限公司 A2a受体拮抗剂治疗癌症的方法
WO2020054712A1 (ja) * 2018-09-12 2020-03-19 日本化薬株式会社 有害生物防除剤

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2097382C1 (ru) * 1991-02-22 1997-11-27 Эгиш Дьедьсердьяр Производные 5-(замещенный амино)-1,2,4-триазол-[1,5а]-пиримидина, их фармацевтически приемлемые кислотно-аддитивные соли, фармацевтическая композиция, обладающая кардиотоническим и коронарорасширяющим действием, и способ кардиотонического и/или коронарорасширяющегося воздействия на сердце
RU2135498C1 (ru) * 1994-06-16 1999-08-27 Пфайзер Инк. Пиразоло- и пирролопиридины

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE287263C (enExample) *
JP4195729B2 (ja) * 1997-03-24 2008-12-10 協和醗酵工業株式会社 ［１，２，４］トリアゾロ［１，５−ｃ］ピリミジン誘導体
US6355653B1 (en) * 1999-09-06 2002-03-12 Hoffmann-La Roche Inc. Amino-triazolopyridine derivatives
US6506772B1 (en) * 2000-12-15 2003-01-14 Hoffmann-La Roche Inc. Substituted [1,2,4]triazolo[1,5a]pyridine derivatives with activity as adenosine receptor ligands

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2097382C1 (ru) * 1991-02-22 1997-11-27 Эгиш Дьедьсердьяр Производные 5-(замещенный амино)-1,2,4-триазол-[1,5а]-пиримидина, их фармацевтически приемлемые кислотно-аддитивные соли, фармацевтическая композиция, обладающая кардиотоническим и коронарорасширяющим действием, и способ кардиотонического и/или коронарорасширяющегося воздействия на сердце
RU2135498C1 (ru) * 1994-06-16 1999-08-27 Пфайзер Инк. Пиразоло- и пирролопиридины

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2552642C2 (ru) * 2008-09-08 2015-06-10 СИГНАЛ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи Аминотриазолопиридины и их применение в качестве ингибиторов киназ
RU2538963C2 (ru) * 2009-07-17 2015-01-10 Джапан Тобакко Инк. Триазолопиридиновое соединение и его действие в качестве ингибитора пролилгидроксилазы и индуктора выработки эритропоэтина
RU2620379C2 (ru) * 2012-02-09 2017-05-25 Ф.Хоффманн-Ля Рош Аг СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ 2-ФЕНИЛ[1,2,4]ТРИАЗОЛО[1,5-а]ПИРИДИНА
RU2681941C2 (ru) * 2013-05-31 2019-03-14 Ниссан Кемикал Индастриз, Лтд. Гетероциклическое амидное соединение

Also Published As

Publication number Publication date
US20030207911A1 (en) 2003-11-06
US6689790B2 (en) 2004-02-10
JP4101755B2 (ja) 2008-06-18
KR20040048940A (ko) 2004-06-10
BR0213172A (pt) 2004-09-14
EP1435952A1 (en) 2004-07-14
CN1564686A (zh) 2005-01-12
KR100614486B1 (ko) 2006-08-22
CA2462806A1 (en) 2003-04-17
AR036734A1 (es) 2004-09-29
MXPA04003277A (es) 2004-07-23
RU2004114278A (ru) 2005-10-27
AU2002347055B2 (en) 2006-10-12
WO2003030904A1 (en) 2003-04-17
JP2005508942A (ja) 2005-04-07
PL370067A1 (en) 2005-05-16

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