RU2005108667A - Производные n-биарилметиламиноциклоалканкарбоксамида - Google Patents
Производные n-биарилметиламиноциклоалканкарбоксамида Download PDFInfo
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- RU2005108667A RU2005108667A RU2005108667/04A RU2005108667A RU2005108667A RU 2005108667 A RU2005108667 A RU 2005108667A RU 2005108667/04 A RU2005108667/04 A RU 2005108667/04A RU 2005108667 A RU2005108667 A RU 2005108667A RU 2005108667 A RU2005108667 A RU 2005108667A
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- optionally substituted
- halogen
- hydrogen
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- YXFVVABEGXRONW-UHFFFAOYSA-N Cc1ccccc1 Chemical compound Cc1ccccc1 YXFVVABEGXRONW-UHFFFAOYSA-N 0.000 description 1
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Vascular Medicine (AREA)
- Obesity (AREA)
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- Hospice & Palliative Care (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40674202P | 2002-08-29 | 2002-08-29 | |
| US60/406,742 | 2002-08-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RU2005108667A true RU2005108667A (ru) | 2005-08-27 |
Family
ID=31978351
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2005108667/04A RU2005108667A (ru) | 2002-08-29 | 2003-08-25 | Производные n-биарилметиламиноциклоалканкарбоксамида |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US7163951B2 (enExample) |
| EP (1) | EP1545538A2 (enExample) |
| JP (1) | JP2005537323A (enExample) |
| KR (1) | KR20050033660A (enExample) |
| CN (1) | CN1678320A (enExample) |
| AU (1) | AU2003265674B2 (enExample) |
| BR (1) | BR0313239A (enExample) |
| CA (1) | CA2495914A1 (enExample) |
| IL (1) | IL166426A0 (enExample) |
| MX (1) | MXPA05002245A (enExample) |
| NO (1) | NO20051539L (enExample) |
| PL (1) | PL374529A1 (enExample) |
| RU (1) | RU2005108667A (enExample) |
| WO (1) | WO2004019868A2 (enExample) |
| ZA (1) | ZA200500471B (enExample) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1654232A4 (en) * | 2003-08-07 | 2008-11-12 | Merck & Co Inc | SULPHONYL SUBSTITUTED N- (BIARYLMETHYL) AMINOCYCLOPROPANCARBOXYLIC ACID AMIDE |
| AU2005211733A1 (en) | 2004-02-11 | 2005-08-25 | Shionogi & Co., Ltd | HIV integrase inhibitors |
| ATE423114T1 (de) * | 2004-03-02 | 2009-03-15 | Merck & Co Inc | Aminocyclopropancarbonsäureamidderivate als bradykininantagonisten |
| US7429604B2 (en) * | 2004-06-15 | 2008-09-30 | Bristol Myers Squibb Company | Six-membered heterocycles useful as serine protease inhibitors |
| US20060217362A1 (en) * | 2004-12-29 | 2006-09-28 | Tung Jay S | Novel compounds useful for bradykinin B1 receptor antagonism |
| ES2422197T3 (es) | 2005-06-03 | 2013-09-09 | Merck Sharp & Dohme | Derivados 1-hidroxicicloalcanocarboxamida como antagonistas de la bradiquinina |
| US8163749B2 (en) | 2005-12-14 | 2012-04-24 | Bristol-Myers Squibb Company | Six-membered heterocycles useful as serine protease inhibitors |
| JP5238812B2 (ja) | 2007-08-29 | 2013-07-17 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 新規ブラジキニンb1アンタゴニスト |
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| WO2010031577A1 (en) * | 2008-09-18 | 2010-03-25 | Jerini Ag | Use of bradykinin b1 receptor antagonists in intestinal fibrosis treatment |
| WO2010097373A1 (de) * | 2009-02-26 | 2010-09-02 | Boehringer Ingelheim International Gmbh | Verbindungen als bradykinin b1 antagonisten |
| GEP20135933B (en) * | 2009-02-26 | 2013-10-10 | Boehringer Ingelheim Int | Compounds as bradykinin b1 antagonists |
| WO2010141273A1 (en) * | 2009-06-02 | 2010-12-09 | Boehringer Ingelheim International Gmbh | DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES |
| KR101628132B1 (ko) * | 2010-01-25 | 2016-06-08 | 주식회사 바이오씨에스 | 신규한 바이아릴아미드 유도체 및 이를 유효성분으로 함유하는 조성물 |
| CN103980258B (zh) | 2010-02-23 | 2016-09-07 | 贝林格尔.英格海姆国际有限公司 | 作为缓激肽b1拮抗剂的化合物 |
| US8937073B2 (en) | 2010-08-20 | 2015-01-20 | Boehringer Ingelheim International Gmbh | Disubstituted tetrahydrofuranyl compounds and their use as B1-receptor antagonists |
| HUP1000598A2 (en) * | 2010-11-05 | 2012-09-28 | Richter Gedeon Nyrt | Indole derivatives |
| US8912221B2 (en) * | 2010-12-27 | 2014-12-16 | Hoffmann-La Roche Inc. | Biaryl amide derivatives |
| US8592426B2 (en) * | 2011-01-24 | 2013-11-26 | Hoffmann—La Roche Inc. | Aryl-benzocycloalkyl amide derivatives |
| NO2686520T3 (enExample) | 2011-06-06 | 2018-03-17 | ||
| PE20160194A1 (es) | 2013-06-13 | 2016-04-20 | Akebia Therapeutics Inc | Composiciones y metodos para tratar anemia |
| AU2016209126A1 (en) | 2015-01-23 | 2017-08-10 | Akebia Therapeutics, Inc. | Solid forms of 2-(5-(3-fluorophenyl)-3-hydroxypicolinamido)acetic acid, compositions, and uses thereof |
| SG11201707994UA (en) | 2015-04-01 | 2017-10-30 | Akebia Therapeutics Inc | Compositions and methods for treating anemia |
| AU2019265629B2 (en) | 2018-05-09 | 2024-09-12 | Akebia Therapeutics, Inc. | Process for preparing 2-((5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl)amino)acetic acid |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5023265A (en) * | 1990-06-01 | 1991-06-11 | Schering Corporation | Substituted 1-H-pyrrolopyridine-3-carboxamides |
| IL99372A0 (en) | 1990-09-10 | 1992-08-18 | Ciba Geigy Ag | Azacyclic compounds |
| CA2473778A1 (en) | 2002-02-08 | 2003-08-14 | Merck & Co., Inc. | N-biphenylmethyl aminocycloalkanecarboxamide derivatives |
| AR038377A1 (es) | 2002-02-08 | 2005-01-12 | Merck & Co Inc | Derivados de n-bifenil-aminocicloalcancarboxamida (con sustitucion con metilo) |
-
2003
- 2003-08-25 US US10/523,911 patent/US7163951B2/en not_active Expired - Fee Related
- 2003-08-25 KR KR1020057003550A patent/KR20050033660A/ko not_active Withdrawn
- 2003-08-25 MX MXPA05002245A patent/MXPA05002245A/es not_active Application Discontinuation
- 2003-08-25 RU RU2005108667/04A patent/RU2005108667A/ru not_active Application Discontinuation
- 2003-08-25 IL IL16642603A patent/IL166426A0/xx unknown
- 2003-08-25 CN CNA03820293XA patent/CN1678320A/zh active Pending
- 2003-08-25 AU AU2003265674A patent/AU2003265674B2/en not_active Ceased
- 2003-08-25 PL PL03374529A patent/PL374529A1/xx not_active Application Discontinuation
- 2003-08-25 WO PCT/US2003/026628 patent/WO2004019868A2/en not_active Ceased
- 2003-08-25 BR BR0313239-0A patent/BR0313239A/pt not_active Application Discontinuation
- 2003-08-25 CA CA002495914A patent/CA2495914A1/en not_active Abandoned
- 2003-08-25 EP EP03791763A patent/EP1545538A2/en not_active Withdrawn
- 2003-08-25 JP JP2004532994A patent/JP2005537323A/ja active Pending
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2005
- 2005-01-18 ZA ZA2005/00471A patent/ZA200500471B/en unknown
- 2005-03-23 NO NO20051539A patent/NO20051539L/no unknown
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|---|---|
| MXPA05002245A (es) | 2005-06-08 |
| WO2004019868A2 (en) | 2004-03-11 |
| US20050288305A1 (en) | 2005-12-29 |
| PL374529A1 (en) | 2005-10-31 |
| AU2003265674B2 (en) | 2008-12-11 |
| AU2003265674A1 (en) | 2004-03-19 |
| NO20051539L (no) | 2005-05-25 |
| BR0313239A (pt) | 2005-06-14 |
| WO2004019868A3 (en) | 2004-04-29 |
| IL166426A0 (en) | 2006-01-15 |
| JP2005537323A (ja) | 2005-12-08 |
| KR20050033660A (ko) | 2005-04-12 |
| CA2495914A1 (en) | 2004-03-11 |
| EP1545538A2 (en) | 2005-06-29 |
| CN1678320A (zh) | 2005-10-05 |
| US7163951B2 (en) | 2007-01-16 |
| ZA200500471B (en) | 2006-07-26 |
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| FA92 | Acknowledgement of application withdrawn (lack of supplementary materials submitted) |
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