RU2003104798A - Содержащие циланзетрон лекарственные средства для лечения не страдающих запорами пациентов мужского пола с синдромом раздраженного кишечника (срк) - Google Patents
Содержащие циланзетрон лекарственные средства для лечения не страдающих запорами пациентов мужского пола с синдромом раздраженного кишечника (срк) Download PDFInfo
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- RU2003104798A RU2003104798A RU2003104798/15A RU2003104798A RU2003104798A RU 2003104798 A RU2003104798 A RU 2003104798A RU 2003104798/15 A RU2003104798/15 A RU 2003104798/15A RU 2003104798 A RU2003104798 A RU 2003104798A RU 2003104798 A RU2003104798 A RU 2003104798A
- Authority
- RU
- Russia
- Prior art keywords
- use according
- ibs
- treatment
- irrital
- cylanesetron
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Claims (8)
1. Применение циланзетрона или его фармакологически приемлемых кислотно-аддитивных солей и/или сольватов для получения фармацевтических композиций, предназначенных для лечения и/или профилактики синдрома раздраженного кишечника (СРК) у не страдающих запорами пациентов мужского пола.
2. Применение по п.1, при котором используют гидрохлорид циланзетрона.
3. Применение по п.1, при котором используют моногидрат гидрохлорида циланзетрона.
4. Применение по меньшей мере одного антагониста 5НТ3-рецептора для получения фармацевтической композиции, предназначенной для лечения страдающих синдромом раздраженного кишечника пациентов обоего пола при ее приеме трижды в день.
5. Применение по п.4, при котором по меньшей мере один антагонист 5НТ3-рецептора применяют в дозе от 1 до 16 мг.
6. Применение по п.4, при котором препарат принимают трижды в день после основных приемов пищи утром, в дневное время и вечером соответственно.
7. Применение по п.4, при котором в качестве антагониста 5НТ3-рецептора применяют алозетрон, азазетрон, долазетрон, гранизетрон, индизетрон, итазетрон, леризетрон, онданзетрон, рамозетрон, тропизетрон и/или (R)-закоприд.
8. Применение по п.4, при котором в качестве антагониста 5НТ3-рецептора применяют циланзетрон или его фармакологически приемлемые кислотно-аддитивные соли и/или сольваты.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10036645 | 2000-07-26 | ||
DE10036645.7 | 2000-07-26 | ||
DE10123447.3 | 2001-05-14 | ||
DE10123447A DE10123447A1 (de) | 2000-07-26 | 2001-05-14 | Cilansetron enthaltende Arzneimittel zur Behandlung nicht-obstipativer männlicher IBS-Patienten |
Publications (1)
Publication Number | Publication Date |
---|---|
RU2003104798A true RU2003104798A (ru) | 2004-06-27 |
Family
ID=26006529
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2003104798/15A RU2003104798A (ru) | 2000-07-26 | 2001-07-18 | Содержащие циланзетрон лекарственные средства для лечения не страдающих запорами пациентов мужского пола с синдромом раздраженного кишечника (срк) |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP1307195A2 (ru) |
JP (1) | JP2004504343A (ru) |
CN (1) | CN1444479A (ru) |
AR (1) | AR028970A1 (ru) |
AU (1) | AU2001276409A1 (ru) |
BR (1) | BR0112690A (ru) |
CA (1) | CA2417677A1 (ru) |
CZ (1) | CZ2003158A3 (ru) |
HU (1) | HUP0301479A2 (ru) |
IL (1) | IL153972A0 (ru) |
MX (1) | MXPA02012917A (ru) |
NO (1) | NO20030373L (ru) |
PL (1) | PL363517A1 (ru) |
RU (1) | RU2003104798A (ru) |
SK (1) | SK1272003A3 (ru) |
WO (1) | WO2002007713A2 (ru) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0216027D0 (en) | 2002-07-10 | 2002-08-21 | Arachnova Therapeutics Ltd | New therapeutic use |
WO2005073220A1 (ja) * | 2004-01-30 | 2005-08-11 | Yamanouchi Pharmaceutical Co., Ltd. | 下痢型過敏性腸症候群治療剤 |
WO2005072730A1 (ja) * | 2004-01-30 | 2005-08-11 | Astellas Pharma Inc. | 下痢型過敏性腸症候群治療剤 |
JP4632204B2 (ja) * | 2005-09-21 | 2011-02-16 | アステラス製薬株式会社 | 下痢型過敏性腸症候群治療剤 |
US7601856B2 (en) | 2006-07-27 | 2009-10-13 | Wyeth | Benzofurans as potassium ion channel modulators |
US7662831B2 (en) | 2006-07-27 | 2010-02-16 | Wyeth Llc | Tetracyclic indoles as potassium channel modulators |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9721139D0 (en) * | 1997-10-07 | 1997-12-03 | Glaxo Group Ltd | Medicaments |
GB9930077D0 (en) * | 1999-12-20 | 2000-02-09 | Glaxo Group Ltd | Medicaments |
-
2001
- 2001-06-21 AR ARP010102958A patent/AR028970A1/es unknown
- 2001-07-18 PL PL01363517A patent/PL363517A1/xx not_active Application Discontinuation
- 2001-07-18 AU AU2001276409A patent/AU2001276409A1/en not_active Abandoned
- 2001-07-18 MX MXPA02012917A patent/MXPA02012917A/es unknown
- 2001-07-18 BR BR0112690-3A patent/BR0112690A/pt not_active Application Discontinuation
- 2001-07-18 WO PCT/EP2001/008260 patent/WO2002007713A2/de not_active Application Discontinuation
- 2001-07-18 JP JP2002513449A patent/JP2004504343A/ja active Pending
- 2001-07-18 RU RU2003104798/15A patent/RU2003104798A/ru not_active Application Discontinuation
- 2001-07-18 HU HU0301479A patent/HUP0301479A2/hu unknown
- 2001-07-18 CA CA002417677A patent/CA2417677A1/en not_active Abandoned
- 2001-07-18 EP EP01954044A patent/EP1307195A2/de not_active Withdrawn
- 2001-07-18 SK SK127-2003A patent/SK1272003A3/sk unknown
- 2001-07-18 CN CN01813307A patent/CN1444479A/zh active Pending
- 2001-07-18 CZ CZ2003158A patent/CZ2003158A3/cs unknown
- 2001-07-18 IL IL15397201A patent/IL153972A0/xx unknown
-
2003
- 2003-01-24 NO NO20030373A patent/NO20030373L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
HUP0301479A2 (hu) | 2003-09-29 |
SK1272003A3 (en) | 2003-07-01 |
CN1444479A (zh) | 2003-09-24 |
JP2004504343A (ja) | 2004-02-12 |
WO2002007713A3 (de) | 2002-11-14 |
CA2417677A1 (en) | 2003-01-27 |
IL153972A0 (en) | 2003-07-31 |
NO20030373D0 (no) | 2003-01-24 |
AR028970A1 (es) | 2003-05-28 |
MXPA02012917A (es) | 2003-05-14 |
WO2002007713A2 (de) | 2002-01-31 |
BR0112690A (pt) | 2003-06-24 |
CZ2003158A3 (cs) | 2003-08-13 |
NO20030373L (no) | 2003-01-24 |
AU2001276409A1 (en) | 2002-02-05 |
PL363517A1 (en) | 2004-11-29 |
EP1307195A2 (de) | 2003-05-07 |
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