RU2002126272A - Производные азолов в качестве терапевтических агентов против грибковых инфекций - Google Patents

Производные азолов в качестве терапевтических агентов против грибковых инфекций Download PDF

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Publication number
RU2002126272A
RU2002126272A RU2002126272/04A RU2002126272A RU2002126272A RU 2002126272 A RU2002126272 A RU 2002126272A RU 2002126272/04 A RU2002126272/04 A RU 2002126272/04A RU 2002126272 A RU2002126272 A RU 2002126272A RU 2002126272 A RU2002126272 A RU 2002126272A
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RU
Russia
Prior art keywords
group
hydroxy
amino
alkoxy
compound
Prior art date
Application number
RU2002126272/04A
Other languages
English (en)
Russian (ru)
Inventor
Ашвани Кумар ВЕРМА (IN)
Ашвани Кумар ВЕРМА
Судершан К. АРОРА (IN)
Судершан К. АРОРА
Джасбир Сингх АРОРА (IN)
Джасбир Сингх АРОРА
Ашок РАТТАН (IN)
Ашок РАТТАН
Original Assignee
Рэнбакси Лабораториз Лимитед (In)
Рэнбакси Лабораториз Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IN198DE2000 external-priority patent/IN191188B/en
Application filed by Рэнбакси Лабораториз Лимитед (In), Рэнбакси Лабораториз Лимитед filed Critical Рэнбакси Лабораториз Лимитед (In)
Publication of RU2002126272A publication Critical patent/RU2002126272A/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
RU2002126272/04A 2000-03-07 2001-03-01 Производные азолов в качестве терапевтических агентов против грибковых инфекций RU2002126272A (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
IN198/DEL/2000 2000-03-07
IN198DE2000 IN191188B (fr) 2000-03-07 2000-03-07
US09/575,578 2000-05-22
US09/575,578 US6670363B1 (en) 2000-03-07 2000-05-22 Azole compounds as therapeutic agents for fungal infections

Publications (1)

Publication Number Publication Date
RU2002126272A true RU2002126272A (ru) 2004-08-10

Family

ID=26324879

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2002126272/04A RU2002126272A (ru) 2000-03-07 2001-03-01 Производные азолов в качестве терапевтических агентов против грибковых инфекций

Country Status (8)

Country Link
EP (1) EP1278755A2 (fr)
JP (1) JP2004501867A (fr)
AU (1) AU3402301A (fr)
CA (1) CA2402345A1 (fr)
NZ (1) NZ521241A (fr)
PL (1) PL365072A1 (fr)
RU (1) RU2002126272A (fr)
WO (1) WO2001066551A2 (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002218505A1 (en) * 2000-11-30 2002-06-11 Senju Pharmaceutical Co. Ltd. Pancreatitis remedies and medicines for prevention and therapy of reflux esophagitis
US6710049B2 (en) 2000-12-26 2004-03-23 Ranbaxy Laboratories Limited Azole compounds as anti-fungal agents
DE60234812D1 (de) 2001-01-29 2010-02-04 Shionogi & Co Arzneipräparat, das als wirkstoff 5-methyl-1-phenyl-2-(1h)-pyridon enthält
HUP0303249A3 (en) 2001-02-22 2007-03-28 Sankyo Co Water-soluble triazole fungicide compounds and pharmaceutical compositions containing them
IN192526B (fr) * 2001-09-25 2004-04-24 Ranbaxy Lab
AU2002328176A1 (en) * 2002-08-26 2004-03-11 Ranbaxy Laboratories Limited Azole derivatives as antifungal agents
EP1413301A1 (fr) * 2002-10-24 2004-04-28 Bayer CropScience SA Médicaments antifongiques à base de dérivés d'arylamidine
WO2007020888A1 (fr) 2005-08-12 2007-02-22 Takeda Pharmaceutical Company Limited Agent protegeant des cellules du cerveau/neuronales et agent therapeutique pour des troubles du sommeil
EP2709609B1 (fr) 2011-05-17 2017-10-04 Shionogi & Co., Ltd. Composés hétérocycliques
US9907812B2 (en) 2011-06-22 2018-03-06 Vyome Biosciences Pvt. Ltd. Conjugate-based antifungal and antibacterial prodrugs
CN102617494B (zh) * 2012-03-15 2014-10-29 南京工业大学 一种含有烯醚结构的三唑类化合物及其制备方法和用途
NZ714817A (en) 2013-06-04 2017-07-28 Vyome Biosciences Pvt Ltd Coated particles and compositions comprising same
MY188541A (en) 2014-01-29 2021-12-21 Vyome Therapeutics Ltd Besifloxacin for the treatment of resistant acne
CA2937365C (fr) 2016-03-29 2018-09-18 F. Hoffmann-La Roche Ag Formulation en granules de 5-methyl-1-phenyl-2-(1h)-pyridone et methode de fabrication associee
AR109545A1 (es) 2016-09-29 2018-12-19 Bayer Cropscience Ag Derivados de triazol

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW218017B (fr) * 1992-04-28 1993-12-21 Takeda Pharm Industry Co Ltd
CA2134417A1 (fr) * 1993-12-22 1995-06-23 Katsumi Itoh Derives azotes optiquement actifs leur production et leur utilisation
US5639754A (en) * 1994-07-12 1997-06-17 Janssen Pharmaceutica N.V. Urea and thiourea derivatives of azolones
EP0957101A1 (fr) * 1998-05-14 1999-11-17 Janssen Pharmaceutica N.V. Azoles solubles dans l'eau, antifongiques à large spectre

Also Published As

Publication number Publication date
CA2402345A1 (fr) 2001-09-13
AU3402301A (en) 2001-09-17
WO2001066551A8 (fr) 2003-06-26
NZ521241A (en) 2004-02-27
WO2001066551A2 (fr) 2001-09-13
PL365072A1 (en) 2004-12-27
JP2004501867A (ja) 2004-01-22
EP1278755A2 (fr) 2003-01-29
WO2001066551A3 (fr) 2002-03-07

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Legal Events

Date Code Title Description
FA92 Acknowledgement of application withdrawn (lack of supplementary materials submitted)

Effective date: 20051115