RU2002126272A - Производные азолов в качестве терапевтических агентов против грибковых инфекций - Google Patents
Производные азолов в качестве терапевтических агентов против грибковых инфекций Download PDFInfo
- Publication number
- RU2002126272A RU2002126272A RU2002126272/04A RU2002126272A RU2002126272A RU 2002126272 A RU2002126272 A RU 2002126272A RU 2002126272/04 A RU2002126272/04 A RU 2002126272/04A RU 2002126272 A RU2002126272 A RU 2002126272A RU 2002126272 A RU2002126272 A RU 2002126272A
- Authority
- RU
- Russia
- Prior art keywords
- group
- hydroxy
- amino
- alkoxy
- compound
- Prior art date
Links
- 0 Cc1c(*)c(*)c(*)c(*)c1N1C*(*)CN(*N(C(*)=NN2C(C(*N3)C4C=CC(*)=C[C@@]4C3=NC=N)C=*)C2=O)CC1 Chemical compound Cc1c(*)c(*)c(*)c(*)c1N1C*(*)CN(*N(C(*)=NN2C(C(*N3)C4C=CC(*)=C[C@@]4C3=NC=N)C=*)C2=O)CC1 0.000 description 2
- VMLFEGKGYIEHLK-UHFFFAOYSA-N CC(C(c(c(F)c1)ccc1F)=O)Oc(cc1)ccc1N(CC1)CCN1C(C)=O Chemical compound CC(C(c(c(F)c1)ccc1F)=O)Oc(cc1)ccc1N(CC1)CCN1C(C)=O VMLFEGKGYIEHLK-UHFFFAOYSA-N 0.000 description 1
- YKLLQPPSMNHDKT-UHFFFAOYSA-N CN(CC(CN/C=N\C=N)(c(c(F)c1)ccc1F)O)c(cc1)ccc1[N+]([O-])=O Chemical compound CN(CC(CN/C=N\C=N)(c(c(F)c1)ccc1F)O)c(cc1)ccc1[N+]([O-])=O YKLLQPPSMNHDKT-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Virology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN198/DEL/2000 | 2000-03-07 | ||
IN198DE2000 IN191188B (fr) | 2000-03-07 | 2000-03-07 | |
US09/575,578 | 2000-05-22 | ||
US09/575,578 US6670363B1 (en) | 2000-03-07 | 2000-05-22 | Azole compounds as therapeutic agents for fungal infections |
Publications (1)
Publication Number | Publication Date |
---|---|
RU2002126272A true RU2002126272A (ru) | 2004-08-10 |
Family
ID=26324879
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2002126272/04A RU2002126272A (ru) | 2000-03-07 | 2001-03-01 | Производные азолов в качестве терапевтических агентов против грибковых инфекций |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1278755A2 (fr) |
JP (1) | JP2004501867A (fr) |
AU (1) | AU3402301A (fr) |
CA (1) | CA2402345A1 (fr) |
NZ (1) | NZ521241A (fr) |
PL (1) | PL365072A1 (fr) |
RU (1) | RU2002126272A (fr) |
WO (1) | WO2001066551A2 (fr) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2002218505A1 (en) * | 2000-11-30 | 2002-06-11 | Senju Pharmaceutical Co. Ltd. | Pancreatitis remedies and medicines for prevention and therapy of reflux esophagitis |
US6710049B2 (en) | 2000-12-26 | 2004-03-23 | Ranbaxy Laboratories Limited | Azole compounds as anti-fungal agents |
DE60234812D1 (de) | 2001-01-29 | 2010-02-04 | Shionogi & Co | Arzneipräparat, das als wirkstoff 5-methyl-1-phenyl-2-(1h)-pyridon enthält |
HUP0303249A3 (en) | 2001-02-22 | 2007-03-28 | Sankyo Co | Water-soluble triazole fungicide compounds and pharmaceutical compositions containing them |
IN192526B (fr) * | 2001-09-25 | 2004-04-24 | Ranbaxy Lab | |
AU2002328176A1 (en) * | 2002-08-26 | 2004-03-11 | Ranbaxy Laboratories Limited | Azole derivatives as antifungal agents |
EP1413301A1 (fr) * | 2002-10-24 | 2004-04-28 | Bayer CropScience SA | Médicaments antifongiques à base de dérivés d'arylamidine |
WO2007020888A1 (fr) | 2005-08-12 | 2007-02-22 | Takeda Pharmaceutical Company Limited | Agent protegeant des cellules du cerveau/neuronales et agent therapeutique pour des troubles du sommeil |
EP2709609B1 (fr) | 2011-05-17 | 2017-10-04 | Shionogi & Co., Ltd. | Composés hétérocycliques |
US9907812B2 (en) | 2011-06-22 | 2018-03-06 | Vyome Biosciences Pvt. Ltd. | Conjugate-based antifungal and antibacterial prodrugs |
CN102617494B (zh) * | 2012-03-15 | 2014-10-29 | 南京工业大学 | 一种含有烯醚结构的三唑类化合物及其制备方法和用途 |
NZ714817A (en) | 2013-06-04 | 2017-07-28 | Vyome Biosciences Pvt Ltd | Coated particles and compositions comprising same |
MY188541A (en) | 2014-01-29 | 2021-12-21 | Vyome Therapeutics Ltd | Besifloxacin for the treatment of resistant acne |
CA2937365C (fr) | 2016-03-29 | 2018-09-18 | F. Hoffmann-La Roche Ag | Formulation en granules de 5-methyl-1-phenyl-2-(1h)-pyridone et methode de fabrication associee |
AR109545A1 (es) | 2016-09-29 | 2018-12-19 | Bayer Cropscience Ag | Derivados de triazol |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW218017B (fr) * | 1992-04-28 | 1993-12-21 | Takeda Pharm Industry Co Ltd | |
CA2134417A1 (fr) * | 1993-12-22 | 1995-06-23 | Katsumi Itoh | Derives azotes optiquement actifs leur production et leur utilisation |
US5639754A (en) * | 1994-07-12 | 1997-06-17 | Janssen Pharmaceutica N.V. | Urea and thiourea derivatives of azolones |
EP0957101A1 (fr) * | 1998-05-14 | 1999-11-17 | Janssen Pharmaceutica N.V. | Azoles solubles dans l'eau, antifongiques à large spectre |
-
2001
- 2001-03-01 NZ NZ521241A patent/NZ521241A/en unknown
- 2001-03-01 PL PL01365072A patent/PL365072A1/xx not_active Application Discontinuation
- 2001-03-01 WO PCT/IB2001/000300 patent/WO2001066551A2/fr not_active Application Discontinuation
- 2001-03-01 RU RU2002126272/04A patent/RU2002126272A/ru not_active Application Discontinuation
- 2001-03-01 EP EP01906061A patent/EP1278755A2/fr not_active Withdrawn
- 2001-03-01 JP JP2001565367A patent/JP2004501867A/ja active Pending
- 2001-03-01 AU AU34023/01A patent/AU3402301A/en not_active Abandoned
- 2001-03-01 CA CA002402345A patent/CA2402345A1/fr not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CA2402345A1 (fr) | 2001-09-13 |
AU3402301A (en) | 2001-09-17 |
WO2001066551A8 (fr) | 2003-06-26 |
NZ521241A (en) | 2004-02-27 |
WO2001066551A2 (fr) | 2001-09-13 |
PL365072A1 (en) | 2004-12-27 |
JP2004501867A (ja) | 2004-01-22 |
EP1278755A2 (fr) | 2003-01-29 |
WO2001066551A3 (fr) | 2002-03-07 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
RU2002126272A (ru) | Производные азолов в качестве терапевтических агентов против грибковых инфекций | |
EP0006712B1 (fr) | Dérivés de (4-aryloxyméthyl-1.3-dioxolan-2-yl)-méthyl-1H-imidazoles et -1H-1.2.4-triazoles hétérocycliques, leur préparation et ces dérives pour utilisation comme fongicides et bactéricides | |
KR970705560A (ko) | 항진균 활성을 갖는 신규한 카르복사미드(new carboxamides with antifungal activity) | |
US6432947B1 (en) | N-heterocyclic derivatives as NOS inhibitors | |
KR890006593A (ko) | 아르마타제 억제4(5)- 이미다졸 | |
HU211474A9 (en) | Azole compounds, their production and use | |
RU2006100298A (ru) | Замещенные производные 3-алкил-и 3-алкенилазетидинов | |
JPH05246999A (ja) | 置換フエニル誘導体 | |
RU2007141892A (ru) | 5-метил-1-(замещенный фенил)-2-(1н)-пиридон для производства медикаментов для лечения фиброза в органах и тканях | |
RU2007108859A (ru) | 1, 5-дифенилпиразолы | |
AU600107B2 (en) | 4-(4-(4-((2-(2,4-difluorophenyl)-2-(1h-azolylmethyl)-1,3- dioxolan-4-yl)methoxy)phenyl)-1-piperazinyl)phenyl) triazolones | |
HU192942B (en) | Process for preparing new subsituted phenyl-ethers | |
WO2009019472A4 (fr) | Nouveaux modulateurs sérotonergiques | |
Rani et al. | Imidazole and Derivatives Drugs Synthesis: A Review | |
RU97116580A (ru) | Триазоловое соединение и его фармакологически приемлемая соль и противогрибковая композиция | |
US9512087B2 (en) | Hybrid molecules containing pharmacophores of fluconazole as antifungal agents and their preparation | |
US4408049A (en) | Substituted piperazinyl-1,2,4-triazoles | |
JP2003516975A5 (fr) | ||
JP2965532B2 (ja) | N−ベンジルアゾリウム誘導体 | |
NZ210727A (en) | 1,3-dioxolanyl derivatives and pharmaceutical compositions | |
RU2002120468A (ru) | Замещенные пирольные основания манниха для борьбы с болыми и аллергическими реакциями | |
RU2006136523A (ru) | Производные простых эфиров, их получение и применение в качестве фармацевтических агентов | |
RU2008150465A (ru) | Ингибиторы калиевых каналов подтипа kv1.5 | |
KR880011115A (ko) | 1-(1-아릴-2- 하이드록시에틸)- 이미다졸 및 그의 염, 이의 제조방법, 이 화합물을 함유한 약제 및 이의 용도 | |
KR940000456A (ko) | 트리아졸 유도체 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA92 | Acknowledgement of application withdrawn (lack of supplementary materials submitted) |
Effective date: 20051115 |