RU2002126272A - Производные азолов в качестве терапевтических агентов против грибковых инфекций - Google Patents
Производные азолов в качестве терапевтических агентов против грибковых инфекций Download PDFInfo
- Publication number
- RU2002126272A RU2002126272A RU2002126272/04A RU2002126272A RU2002126272A RU 2002126272 A RU2002126272 A RU 2002126272A RU 2002126272/04 A RU2002126272/04 A RU 2002126272/04A RU 2002126272 A RU2002126272 A RU 2002126272A RU 2002126272 A RU2002126272 A RU 2002126272A
- Authority
- RU
- Russia
- Prior art keywords
- group
- hydroxy
- amino
- alkoxy
- compound
- Prior art date
Links
- 0 Cc1c(*)c(*)c(*)c(*)c1N1C*(*)CN(*N(C(*)=NN2C(C(*N3)C4C=CC(*)=C[C@@]4C3=NC=N)C=*)C2=O)CC1 Chemical compound Cc1c(*)c(*)c(*)c(*)c1N1C*(*)CN(*N(C(*)=NN2C(C(*N3)C4C=CC(*)=C[C@@]4C3=NC=N)C=*)C2=O)CC1 0.000 description 2
- VMLFEGKGYIEHLK-UHFFFAOYSA-N CC(C(c(c(F)c1)ccc1F)=O)Oc(cc1)ccc1N(CC1)CCN1C(C)=O Chemical compound CC(C(c(c(F)c1)ccc1F)=O)Oc(cc1)ccc1N(CC1)CCN1C(C)=O VMLFEGKGYIEHLK-UHFFFAOYSA-N 0.000 description 1
- YKLLQPPSMNHDKT-UHFFFAOYSA-N CN(CC(CN/C=N\C=N)(c(c(F)c1)ccc1F)O)c(cc1)ccc1[N+]([O-])=O Chemical compound CN(CC(CN/C=N\C=N)(c(c(F)c1)ccc1F)O)c(cc1)ccc1[N+]([O-])=O YKLLQPPSMNHDKT-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Virology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN198/DEL/2000 | 2000-03-07 | ||
| IN198DE2000 IN191188B (fr) | 2000-03-07 | 2000-03-07 | |
| US09/575,578 | 2000-05-22 | ||
| US09/575,578 US6670363B1 (en) | 2000-03-07 | 2000-05-22 | Azole compounds as therapeutic agents for fungal infections |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RU2002126272A true RU2002126272A (ru) | 2004-08-10 |
Family
ID=26324879
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2002126272/04A RU2002126272A (ru) | 2000-03-07 | 2001-03-01 | Производные азолов в качестве терапевтических агентов против грибковых инфекций |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP1278755A2 (fr) |
| JP (1) | JP2004501867A (fr) |
| AU (1) | AU3402301A (fr) |
| CA (1) | CA2402345A1 (fr) |
| NZ (1) | NZ521241A (fr) |
| PL (1) | PL365072A1 (fr) |
| RU (1) | RU2002126272A (fr) |
| WO (1) | WO2001066551A2 (fr) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2002218505A1 (en) * | 2000-11-30 | 2002-06-11 | Senju Pharmaceutical Co. Ltd. | Pancreatitis remedies and medicines for prevention and therapy of reflux esophagitis |
| US6710049B2 (en) | 2000-12-26 | 2004-03-23 | Ranbaxy Laboratories Limited | Azole compounds as anti-fungal agents |
| DE60234812D1 (de) | 2001-01-29 | 2010-02-04 | Shionogi & Co | Arzneipräparat, das als wirkstoff 5-methyl-1-phenyl-2-(1h)-pyridon enthält |
| HUP0303249A3 (en) | 2001-02-22 | 2007-03-28 | Sankyo Co | Water-soluble triazole fungicide compounds and pharmaceutical compositions containing them |
| IN192526B (fr) * | 2001-09-25 | 2004-04-24 | Ranbaxy Lab | |
| AU2002328176A1 (en) * | 2002-08-26 | 2004-03-11 | Ranbaxy Laboratories Limited | Azole derivatives as antifungal agents |
| EP1413301A1 (fr) * | 2002-10-24 | 2004-04-28 | Bayer CropScience SA | Médicaments antifongiques à base de dérivés d'arylamidine |
| WO2007020888A1 (fr) | 2005-08-12 | 2007-02-22 | Takeda Pharmaceutical Company Limited | Agent protegeant des cellules du cerveau/neuronales et agent therapeutique pour des troubles du sommeil |
| EP2709609B1 (fr) | 2011-05-17 | 2017-10-04 | Shionogi & Co., Ltd. | Composés hétérocycliques |
| US9907812B2 (en) | 2011-06-22 | 2018-03-06 | Vyome Biosciences Pvt. Ltd. | Conjugate-based antifungal and antibacterial prodrugs |
| CN102617494B (zh) * | 2012-03-15 | 2014-10-29 | 南京工业大学 | 一种含有烯醚结构的三唑类化合物及其制备方法和用途 |
| NZ714817A (en) | 2013-06-04 | 2017-07-28 | Vyome Biosciences Pvt Ltd | Coated particles and compositions comprising same |
| MY188541A (en) | 2014-01-29 | 2021-12-21 | Vyome Therapeutics Ltd | Besifloxacin for the treatment of resistant acne |
| CA2937365C (fr) | 2016-03-29 | 2018-09-18 | F. Hoffmann-La Roche Ag | Formulation en granules de 5-methyl-1-phenyl-2-(1h)-pyridone et methode de fabrication associee |
| AR109545A1 (es) | 2016-09-29 | 2018-12-19 | Bayer Cropscience Ag | Derivados de triazol |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW218017B (fr) * | 1992-04-28 | 1993-12-21 | Takeda Pharm Industry Co Ltd | |
| CA2134417A1 (fr) * | 1993-12-22 | 1995-06-23 | Katsumi Itoh | Derives azotes optiquement actifs leur production et leur utilisation |
| US5639754A (en) * | 1994-07-12 | 1997-06-17 | Janssen Pharmaceutica N.V. | Urea and thiourea derivatives of azolones |
| EP0957101A1 (fr) * | 1998-05-14 | 1999-11-17 | Janssen Pharmaceutica N.V. | Azoles solubles dans l'eau, antifongiques à large spectre |
-
2001
- 2001-03-01 NZ NZ521241A patent/NZ521241A/en unknown
- 2001-03-01 PL PL01365072A patent/PL365072A1/xx not_active Application Discontinuation
- 2001-03-01 WO PCT/IB2001/000300 patent/WO2001066551A2/fr not_active Application Discontinuation
- 2001-03-01 RU RU2002126272/04A patent/RU2002126272A/ru not_active Application Discontinuation
- 2001-03-01 EP EP01906061A patent/EP1278755A2/fr not_active Withdrawn
- 2001-03-01 JP JP2001565367A patent/JP2004501867A/ja active Pending
- 2001-03-01 AU AU34023/01A patent/AU3402301A/en not_active Abandoned
- 2001-03-01 CA CA002402345A patent/CA2402345A1/fr not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2402345A1 (fr) | 2001-09-13 |
| AU3402301A (en) | 2001-09-17 |
| WO2001066551A8 (fr) | 2003-06-26 |
| NZ521241A (en) | 2004-02-27 |
| WO2001066551A2 (fr) | 2001-09-13 |
| PL365072A1 (en) | 2004-12-27 |
| JP2004501867A (ja) | 2004-01-22 |
| EP1278755A2 (fr) | 2003-01-29 |
| WO2001066551A3 (fr) | 2002-03-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA92 | Acknowledgement of application withdrawn (lack of supplementary materials submitted) |
Effective date: 20051115 |