RS50138B - Derivati streptogramina, njihovo dobivanje i smeše koje ih sardže - Google Patents

Derivati streptogramina, njihovo dobivanje i smeše koje ih sardže

Info

Publication number
RS50138B
RS50138B YUP-895/01A YUP89501A RS50138B RS 50138 B RS50138 B RS 50138B YU P89501 A YUP89501 A YU P89501A RS 50138 B RS50138 B RS 50138B
Authority
RS
Serbia
Prior art keywords
denotes
preparation
compositions containing
hydrogen atom
bond
Prior art date
Application number
YUP-895/01A
Other languages
English (en)
Inventor
Yves Ribeill
Daniel Achard
Eric Bacque
Jean-Claude Barriere
Jean Bouquerel
Pascal Desmazeau
Serge Grisoni
Jean-Pierre Leconte
Baptiste Ronan
Original Assignee
Novexel,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9547496&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS50138(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novexel, filed Critical Novexel,
Publication of YU89501A publication Critical patent/YU89501A/sh
Publication of RS50138B publication Critical patent/RS50138B/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C07K5/06182—Dipeptides with the first amino acid being heterocyclic and Pristinamycin II; Derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Derivat streptogramina grupe A opšte formule u kojoj : - R1 označava atom halogena ili radikal azido ili tiocij anato, - R2 označava atom vodonika ili radikal metil ili etil, - R3 označava atom vodonika ili ostatak alifatičnog, cikloalifatičnog, aromatičnog, aralifatičnog, heterocikličnog ili heterociklilalifatičnog estra koji može biti supstituisan, i - veza = označava prostu vezu (stereohemije 27R) ili dvostruku vezu, kao i njihove soli, kada postoje. Prijava sadrži još 2 nezavisna i 12 zavisnih patentnih zahteva.
YUP-895/01A 1999-06-30 2000-07-29 Derivati streptogramina, njihovo dobivanje i smeše koje ih sardže RS50138B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9908375A FR2795733B1 (fr) 1999-06-30 1999-06-30 Derives de streptogramines, leur preparation et les compositions qui les contiennent

Publications (2)

Publication Number Publication Date
YU89501A YU89501A (sh) 2004-05-12
RS50138B true RS50138B (sr) 2009-03-25

Family

ID=9547496

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-895/01A RS50138B (sr) 1999-06-30 2000-07-29 Derivati streptogramina, njihovo dobivanje i smeše koje ih sardže

Country Status (37)

Country Link
US (2) US6569854B1 (sr)
EP (1) EP1187847B1 (sr)
JP (1) JP4585728B2 (sr)
KR (1) KR100742035B1 (sr)
CN (2) CN1961878A (sr)
AP (1) AP1392A (sr)
AR (2) AR029758A1 (sr)
AT (1) ATE255592T1 (sr)
AU (1) AU781923B2 (sr)
BG (1) BG65786B1 (sr)
BR (1) BRPI0012032B1 (sr)
CA (1) CA2376698C (sr)
CZ (1) CZ301048B6 (sr)
DE (1) DE60006958T2 (sr)
DK (1) DK1187847T3 (sr)
EA (1) EA005199B1 (sr)
EE (1) EE04683B1 (sr)
ES (1) ES2207535T3 (sr)
FR (1) FR2795733B1 (sr)
GE (1) GEP20063972B (sr)
HR (1) HRP20010937B1 (sr)
HU (1) HUP0201692A3 (sr)
IL (2) IL146185A0 (sr)
MA (1) MA26802A1 (sr)
MX (1) MXPA01012807A (sr)
NO (1) NO329456B1 (sr)
NZ (1) NZ516100A (sr)
OA (1) OA11979A (sr)
PT (1) PT1187847E (sr)
RS (1) RS50138B (sr)
SI (1) SI1187847T1 (sr)
SK (1) SK285605B6 (sr)
TN (1) TNSN00145A1 (sr)
TR (1) TR200103829T2 (sr)
UA (1) UA71619C2 (sr)
WO (1) WO2001002427A1 (sr)
ZA (1) ZA200110150B (sr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2775288B1 (fr) * 1998-02-26 2000-03-31 Rhone Poulenc Rorer Sa Derives de streptogramines, leur preparation et les compositons qui les contiennent
FR2795733B1 (fr) * 1999-06-30 2001-09-07 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
US7232799B2 (en) 2000-12-21 2007-06-19 Aventis Pharma Sa Streptogramin derivatives and compositions thereof
US6596717B2 (en) 2000-12-21 2003-07-22 Aventis Pharma S.A. Streptogramin derivatives, their preparation and compositions which contain them
WO2005066135A2 (en) 2003-12-29 2005-07-21 Sepracor Inc. Pyrrole and pyrazole daao inhibitors
US7565200B2 (en) * 2004-11-12 2009-07-21 Advanced Neuromodulation Systems, Inc. Systems and methods for selecting stimulation sites and applying treatment, including treatment of symptoms of Parkinson's disease, other movement disorders, and/or drug side effects
CN101394847B (zh) 2006-01-06 2017-05-24 塞普拉柯公司 作为单胺重摄取抑制剂的环烷基胺类
AU2006335174B2 (en) 2006-01-06 2012-09-06 Sunovion Pharmaceuticals Inc. Tetralone-based monoamine reuptake inhibitors
CN103588659A (zh) 2006-03-31 2014-02-19 赛诺维信制药公司 手性酰胺和胺的制备
US7884124B2 (en) 2006-06-30 2011-02-08 Sepracor Inc. Fluoro-substituted inhibitors of D-amino acid oxidase
US7902252B2 (en) 2007-01-18 2011-03-08 Sepracor, Inc. Inhibitors of D-amino acid oxidase
EP2154962A4 (en) 2007-05-31 2012-08-15 Sepracor Inc PHENYL-SUBSTITUTED CYCLOALKYLAMINE AS A MONOAMINE RECOVERY INHIBITOR
CN103508981A (zh) * 2012-06-18 2014-01-15 北京美倍他药物研究有限公司 新的哌嗪衍生物及其医药用途
CA3070851A1 (en) * 2017-08-01 2019-02-07 The Regents Of The University Of California Methods of making streptogramin compositions and the use thereof
KR102107659B1 (ko) 2018-12-07 2020-05-07 경상대학교 산학협력단 Mmagnu1 화합물을 유효성분으로 함유하는 결핵균 또는 비결핵 항산균 감염 질환 예방 또는 치료용 조성물
EP4157268A1 (en) 2020-05-27 2023-04-05 Università Degli Studi Di Trento New therapy for the treatment of tumors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2549065B1 (fr) * 1983-07-13 1985-10-25 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2576022B1 (fr) * 1985-01-11 1987-09-11 Rhone Poulenc Sante Nouveaux derives de la pristinamycine ii b, leur preparation et les compositions pharmaceutiques qui les contiennent
BE1001013A4 (fr) 1987-10-22 1989-06-13 Icp Internat Inst Of Cellular Derives de synergimycines de types a et b, procede pour leur preparation et utilisation de ceux-ci.
IL121821A (en) * 1993-02-17 2000-02-17 Rhone Poulenc Rorer Sa Process for purifying a group A minority component of streptogramin some such purified components and their uses
FR2766489B1 (fr) * 1997-07-28 1999-08-27 Rhone Poulenc Rorer Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
FR2795733B1 (fr) * 1999-06-30 2001-09-07 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent

Also Published As

Publication number Publication date
SK19302001A3 (sk) 2002-07-02
MXPA01012807A (es) 2002-07-22
NO329456B1 (no) 2010-10-25
KR100742035B1 (ko) 2007-07-23
AU6288600A (en) 2001-01-22
HRP20010937A2 (en) 2003-08-31
KR20020020763A (ko) 2002-03-15
YU89501A (sh) 2004-05-12
PL352781A1 (en) 2003-09-08
UA71619C2 (uk) 2004-12-15
AP2001002371A0 (en) 2001-12-31
NO20016247L (no) 2002-02-08
DE60006958D1 (de) 2004-01-15
ZA200110150B (en) 2003-03-10
SI1187847T1 (en) 2004-04-30
TNSN00145A1 (fr) 2002-05-30
US7166594B2 (en) 2007-01-23
HUP0201692A2 (en) 2002-09-28
CN1358194A (zh) 2002-07-10
EP1187847B1 (fr) 2003-12-03
BR0012032A (pt) 2002-03-19
EP1187847A1 (fr) 2002-03-20
CZ301048B6 (cs) 2009-10-21
EA200200108A1 (ru) 2002-06-27
NO20016247D0 (no) 2001-12-19
CN1961878A (zh) 2007-05-16
AU781923B2 (en) 2005-06-23
EA005199B1 (ru) 2004-12-30
BRPI0012032B1 (pt) 2015-06-30
AR029758A1 (es) 2003-07-16
GEP20063972B (en) 2006-11-27
ES2207535T3 (es) 2004-06-01
JP4585728B2 (ja) 2010-11-24
FR2795733A1 (fr) 2001-01-05
OA11979A (fr) 2006-04-18
US20030149004A1 (en) 2003-08-07
HUP0201692A3 (en) 2002-10-28
AR066926A2 (es) 2009-09-23
ATE255592T1 (de) 2003-12-15
EE04683B1 (et) 2006-08-15
MA26802A1 (fr) 2004-12-20
TR200103829T2 (tr) 2002-04-22
CZ20014641A3 (cs) 2002-04-17
DE60006958T2 (de) 2004-10-21
CN100543032C (zh) 2009-09-23
IL146185A0 (en) 2002-07-25
CA2376698A1 (fr) 2001-01-11
SK285605B6 (sk) 2007-04-05
BG65786B1 (bg) 2009-11-30
US6569854B1 (en) 2003-05-27
NZ516100A (en) 2004-01-30
EE200100706A (et) 2003-04-15
HRP20010937B1 (en) 2005-02-28
DK1187847T3 (da) 2004-01-05
WO2001002427A1 (fr) 2001-01-11
BG106235A (en) 2002-08-30
CA2376698C (fr) 2013-05-14
AP1392A (en) 2005-04-15
JP2003503509A (ja) 2003-01-28
PT1187847E (pt) 2004-04-30
FR2795733B1 (fr) 2001-09-07
IL146185A (en) 2007-08-19

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