RO73278A - PROCESS FOR THE PREPARATION OF PIPERAZINE DERIVATIVES PROCESS FOR THE PREPARATION OF A PIPERAZINE DERIVATIVE - Google Patents

PROCESS FOR THE PREPARATION OF PIPERAZINE DERIVATIVES PROCESS FOR THE PREPARATION OF A PIPERAZINE DERIVATIVE

Info

Publication number
RO73278A
RO73278A RO7685688A RO8568876A RO73278A RO 73278 A RO73278 A RO 73278A RO 7685688 A RO7685688 A RO 7685688A RO 8568876 A RO8568876 A RO 8568876A RO 73278 A RO73278 A RO 73278A
Authority
RO
Romania
Prior art keywords
preparation
piperazine
derivative
derivatives
piperazine derivatives
Prior art date
Application number
RO7685688A
Other languages
French (fr)
Romanian (ro)
Inventor
Walfred S Saari
Jr William C Lumma
William C Lumma
Original Assignee
Merc & Co Inc,Us
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merc & Co Inc,Us filed Critical Merc & Co Inc,Us
Publication of RO73278A publication Critical patent/RO73278A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
RO7685688A 1975-04-21 1976-04-20 PROCESS FOR THE PREPARATION OF PIPERAZINE DERIVATIVES PROCESS FOR THE PREPARATION OF A PIPERAZINE DERIVATIVE RO73278A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57005275A 1975-04-21 1975-04-21

Publications (1)

Publication Number Publication Date
RO73278A true RO73278A (en) 1982-09-09

Family

ID=24277994

Family Applications (1)

Application Number Title Priority Date Filing Date
RO7685688A RO73278A (en) 1975-04-21 1976-04-20 PROCESS FOR THE PREPARATION OF PIPERAZINE DERIVATIVES PROCESS FOR THE PREPARATION OF A PIPERAZINE DERIVATIVE

Country Status (36)

Country Link
JP (1) JPS51136688A (en)
AR (1) AR210349A1 (en)
AT (1) AT353795B (en)
AU (1) AU496854B2 (en)
BE (1) BE840904A (en)
BG (1) BG34185A3 (en)
CA (1) CA1059128A (en)
CH (1) CH619462A5 (en)
CS (1) CS195726B2 (en)
CY (1) CY1090A (en)
DD (1) DD124599A5 (en)
DE (1) DE2617205C3 (en)
DK (1) DK143899C (en)
EG (1) EG12387A (en)
ES (4) ES447150A1 (en)
FI (1) FI62666C (en)
FR (1) FR2308367A1 (en)
GB (1) GB1492528A (en)
GR (1) GR59900B (en)
HK (1) HK60380A (en)
HU (1) HU172684B (en)
IE (1) IE42979B1 (en)
IL (1) IL49391A (en)
KE (1) KE3088A (en)
LU (1) LU74795A1 (en)
MY (1) MY8100225A (en)
NL (1) NL167692C (en)
NO (1) NO146599C (en)
PH (1) PH12274A (en)
PL (1) PL99664B1 (en)
PT (1) PT65027B (en)
RO (1) RO73278A (en)
SE (1) SE421695B (en)
SU (1) SU638260A3 (en)
YU (1) YU100676A (en)
ZA (1) ZA762320B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4091098A (en) * 1977-04-25 1978-05-23 Merck & Co., Inc. 3-(1-PIPERAZINYL)-1,2,4-BENZOTRIAZINES AND N-oxides
US4163849A (en) 1978-03-17 1979-08-07 Merck & Co., Inc. Piperazinylpyrazines
US4252816A (en) * 1979-12-03 1981-02-24 Merck & Co., Inc. Tetrahydro-1H-1,4-diazepino(1,7-a)benzimidazoles useful as analgesic agents
US4339579A (en) 1980-12-29 1982-07-13 American Home Products Corporation 2,6-Bis-(pyrrolopyrazinyl)pyrazines
EP0094498A3 (en) * 1982-05-06 1985-04-03 American Cyanamid Company Antiatherosclerotic 1-piperazine derivatives
US4547505A (en) * 1983-03-25 1985-10-15 Degussa Aktiengesellschaft N-Phenyl-N-'-cycloalkylalkanoylpiperazine useful as analgetics and process for its production
US4788290A (en) * 1987-12-11 1988-11-29 American Home Products Corporation Serotonergic pyrazine derivatives
EP0580465A1 (en) * 1992-06-25 1994-01-26 Sanofi New therapeutic use of heterocyclic piperazines as 5-HT3 agonists and new derivatives
SK285198B6 (en) * 1997-10-27 2006-08-03 Neurosearch A/S Homopiperazine derivative, pharmaceutical composition containing this derivative and using of it
JP2002543070A (en) 1999-04-26 2002-12-17 ニューロサーチ、アクティーゼルスカブ Heteroaryldiazacycloalkanes, their production and use
DK1255740T3 (en) * 2000-02-16 2006-02-06 Neurogen Corp Substituted arylpyrazines
US6825198B2 (en) * 2001-06-21 2004-11-30 Pfizer Inc 5-HT receptor ligands and uses thereof
SE0202287D0 (en) * 2002-07-19 2002-07-19 Biovitrum Ab New compounds
CA2492924C (en) * 2002-07-19 2011-12-20 Biovitrum Ab Novel piperazinone derivates for the treatment of 5-ht2a receptor-related disorders

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2606906A (en) * 1948-10-14 1952-08-12 American Cyanamid Co 1-(2-pyridyl) piperazine and process of preparing same

Also Published As

Publication number Publication date
ES459405A1 (en) 1978-08-16
AT353795B (en) 1979-12-10
FI62666B (en) 1982-10-29
ES447150A1 (en) 1977-09-16
GB1492528A (en) 1977-11-23
PT65027B (en) 1978-04-03
EG12387A (en) 1978-12-31
DE2617205B2 (en) 1980-05-08
MY8100225A (en) 1981-12-31
PH12274A (en) 1978-12-12
ATA288376A (en) 1979-05-15
CA1059128A (en) 1979-07-24
SU638260A3 (en) 1978-12-15
NO146599C (en) 1982-11-03
IL49391A0 (en) 1976-06-30
NL167692C (en) 1982-01-18
AU1296676A (en) 1977-10-20
DE2617205A1 (en) 1976-10-28
DK164476A (en) 1976-10-22
ZA762320B (en) 1977-11-30
AR210349A1 (en) 1977-07-29
CH619462A5 (en) 1980-09-30
DK143899C (en) 1982-04-13
JPS51136688A (en) 1976-11-26
HU172684B (en) 1978-11-28
FR2308367A1 (en) 1976-11-19
CS195726B2 (en) 1980-02-29
HK60380A (en) 1980-11-07
LU74795A1 (en) 1977-02-07
SE7604093L (en) 1976-10-22
FI760978A (en) 1976-10-22
JPS5522475B2 (en) 1980-06-17
NO146599B (en) 1982-07-26
NO761207L (en) 1976-10-22
PL99664B1 (en) 1978-07-31
DD124599A5 (en) 1977-03-02
AU496854B2 (en) 1978-11-02
DE2617205C3 (en) 1981-01-29
ES459406A1 (en) 1978-08-16
NL7603800A (en) 1976-10-25
BE840904A (en) 1976-08-16
YU100676A (en) 1982-08-31
ES459407A1 (en) 1978-08-16
IE42979L (en) 1976-10-21
PT65027A (en) 1976-05-01
DK143899B (en) 1981-10-26
GR59900B (en) 1978-03-16
FR2308367B1 (en) 1979-09-21
FI62666C (en) 1983-02-10
IE42979B1 (en) 1980-11-19
IL49391A (en) 1979-09-30
CY1090A (en) 1980-12-27
NL167692B (en) 1981-08-17
SE421695B (en) 1982-01-25
KE3088A (en) 1980-11-07
BG34185A3 (en) 1983-07-15

Similar Documents

Publication Publication Date Title
RO70769A (en) PROCESS FOR THE PREPARATION OF 2-PHENYL-3-ACYLBENZOTHIOPHENE DERIVATIVES
RO68441A (en) PROCESS FOR THE PREPARATION OF ERYTHROMYCYLAMINE DERIVATIVES
RO70897A (en) PROCESS FOR THE PREPARATION OF PHENOXY-BENZYLOXYCARBONYLESUBSTITUS DERIVATIVES
RO80036A (en) PROCESS FOR OBTAINING N-THIOLCARBONYL-N-PHOSPHONOMETHYLGLYCIN DERIVATIVES
RO70768A (en) PROCESS FOR THE PREPARATION OF 2-ARYL-5-PHENYLBENZOTHIOPHENE DERIVATIVES
RO70162A (en) PROCESS FOR OBTAINING 7-ALCOXY-5-METHYL-ISOFLAVONE DERIVATIVES
RO73517A (en) PROCESS FOR THE PREPARATION OF AMINOGLYCOSIDIC DERIVATIVES
PT64912B (en) PROCESS FOR THE PREPARATION OF SALICILANILIDE DERIVATIVES
RO73278A (en) PROCESS FOR THE PREPARATION OF PIPERAZINE DERIVATIVES PROCESS FOR THE PREPARATION OF A PIPERAZINE DERIVATIVE
RO72349A (en) PROCESS FOR THE PREPARATION OF IMIDAZOLE DERIVATIVES WITH PHARMACOLOGICAL ACTION
RO75109A (en) PROCESS FOR THE PREPARATION OF DIPHENYLEAMINE DERIVATIVES
RO79969A (en) PROCESS FOR THE PREPARATION OF KANAMICINE DERIVATIVES
RO79048A (en) PROCESS FOR THE PREPARATION OF 5,11-DIHYDRO-6H-PYRIDO- (2,3B) - (1,4) -BENZODIAZEPIN-6-ONE DERIVATIVES
PT66781B (en) PROCESS FOR THE PREPARATION OF PHENOXY-HYDROXYPROPYLAMINE DERIVATIVES
BE841260A (en) PROCESS FOR THE PREPARATION OF OXAZOLE DERIVATIVES
PT66154B (en) PROCESS FOR THE PREPARATION OF NEW PIPERAZINE DERIVATIVES
RO78658A (en) PROCESS FOR THE PREPARATION OF ANTRAQUINONSULFONAMIDE DERIVATIVES
RO76588A (en) PROCESS FOR THE PREPARATION OF 1,3,4-TRIDIAZOLE DERIVATIVES
PT70007A (en) PROCESS FOR THE PREPARATION OF PHENYL-1 PIPERAZINE DERIVATIVES
RO72848A (en) PROCESS FOR THE PREPARATION OF 204 I ANTIBIOTIC DERIVATIVES
RO75387A (en) PROCESS FOR THE PREPARATION OF 4 "-AMINOOLEANDOMICYNE DERIVATIVES
RO73274A (en) PROCESS FOR THE PREPARATION OF AZETIDINE-4-ONE DERIVATIVES
RO79687A7 (en) PROCESS FOR THE PREPARATION OF 4 '' - DESOXY - 4 '' - AMINOERYTHROMYCIN A DERIVATIVES
RO71394A (en) PROCESS FOR OBTAINING PIPERAZINE DERIVATIVES
RO76124A (en) PROCESS FOR THE PREPARATION OF 3-HYDROXYMETHYLENE-4-CHROMANONE DERIVATIVES