PT920421E - Derivados de isoxazolina uteis como agentes antimicrobianos - Google Patents

Derivados de isoxazolina uteis como agentes antimicrobianos

Info

Publication number
PT920421E
PT920421E PT97937156T PT97937156T PT920421E PT 920421 E PT920421 E PT 920421E PT 97937156 T PT97937156 T PT 97937156T PT 97937156 T PT97937156 T PT 97937156T PT 920421 E PT920421 E PT 920421E
Authority
PT
Portugal
Prior art keywords
uteis
antimicrobial agents
isoxazoline derivatives
isoxazoline
derivatives
Prior art date
Application number
PT97937156T
Other languages
English (en)
Portuguese (pt)
Inventor
Richard C Thomas
Michael R Barbachyn
Gary J Cleek
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of PT920421E publication Critical patent/PT920421E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
PT97937156T 1996-08-21 1997-08-15 Derivados de isoxazolina uteis como agentes antimicrobianos PT920421E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2428796P 1996-08-21 1996-08-21

Publications (1)

Publication Number Publication Date
PT920421E true PT920421E (pt) 2003-03-31

Family

ID=21819822

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97937156T PT920421E (pt) 1996-08-21 1997-08-15 Derivados de isoxazolina uteis como agentes antimicrobianos

Country Status (10)

Country Link
US (2) US5990136A (Direct)
EP (1) EP0920421B1 (Direct)
JP (1) JP2000516245A (Direct)
AT (1) ATE227277T1 (Direct)
AU (1) AU3973697A (Direct)
DE (1) DE69716925T2 (Direct)
DK (1) DK0920421T3 (Direct)
ES (1) ES2186916T3 (Direct)
PT (1) PT920421E (Direct)
WO (1) WO1998007708A1 (Direct)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9609919D0 (en) 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
DE69829846T2 (de) * 1997-05-30 2006-02-23 Pharmacia & Upjohn Co. Llc, Kalamazoo Antibakteriell wirksam oxazolidinone mit einer thiocarbonylfunktionalität
US6255304B1 (en) 1997-05-30 2001-07-03 Pharmacia & Upjohn Company Oxazolidinone antibacterial agents having a thiocarbonyl functionality
GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9717807D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9725244D0 (en) 1997-11-29 1998-01-28 Zeneca Ltd Chemical compounds
ES2182485T3 (es) * 1998-02-13 2003-03-01 Upjohn Co Derivados de aminofenil isosazolina sustituidos utiles como agentes antimicrobianos.
CA2318762A1 (en) * 1998-02-25 1999-09-02 Richard Charles Thomas Substituted aminomethyl isoxazoline derivatives useful as antimicrobials
KR20010052615A (ko) 1998-06-05 2001-06-25 다비드 에 질레스 옥사졸리디논 유도체, 이것의 제조 방법 및 이것을함유하는 약학 조성물
TW572757B (en) * 1998-08-24 2004-01-21 Bristol Myers Squibb Co Novel isoxazolinone antibacterial agents
US6420349B1 (en) 1998-08-24 2002-07-16 Bristol-Myers Squibb Company Isoxazolinone antibacterial agents
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
GB0009803D0 (en) 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
US6465456B2 (en) 2000-06-29 2002-10-15 Bristol-Myers Squibb Company Isoxazolinone antibacterial agents
JP2004518677A (ja) 2000-12-21 2004-06-24 ファルマシア・アンド・アップジョン・カンパニー 抗菌性キノロン誘導体および細菌感染を治療するためのその使用
KR20030077558A (ko) * 2000-12-26 2003-10-01 재단법인 이쯔우 연구소 트로폴론 유도체
WO2003035073A1 (en) * 2001-10-25 2003-05-01 Astrazeneca Ab Isoxazoline derivatives useful as antimicrobials
AR038536A1 (es) * 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
US7141588B2 (en) * 2002-02-25 2006-11-28 Pfizer, Inc. N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
JP2006516989A (ja) * 2003-02-07 2006-07-13 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー 抗菌剤として使用するための二環式環によりｎ−置換されたオキサゾリジノン誘導体
BRPI0407252A (pt) * 2003-02-07 2006-01-31 Warner Lambert Co Agentes antibacterianos.
US7304050B2 (en) * 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
WO2005082900A2 (en) * 2004-01-28 2005-09-09 Pharmacia & Upjohn Company Llc Oxazolidinone amidoximes as antibacterial agents
AU2005270951A1 (en) * 2004-08-06 2006-02-16 Pharmacia & Upjohn Company Llc Oxazolidinones containing oxindoles as antibacterial agents
EP1794167A4 (en) * 2004-09-10 2009-10-21 Syngenta Ltd SUBSTITUTED ISOXAZOLE AS FUNGICIDES
CN103270036B (zh) * 2010-08-05 2015-11-25 佐蒂斯有限责任公司 作为抗寄生物剂的异噁唑啉衍生物
JP5918264B2 (ja) 2010-12-22 2016-05-18 アッヴィ・インコーポレイテッド Ｃ型肝炎阻害剤およびその使用
GB2521558B (en) * 2012-10-03 2019-03-27 Shell Int Research Optimizing performance of a drilling assembly
WO2021000297A1 (en) * 2019-07-03 2021-01-07 Merck Sharp & Dohme Corp. Compounds and methods of use thereof as antibacterial agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL137326C (Direct) * 1967-08-26
US4283403A (en) * 1976-06-14 1981-08-11 Eli Lilly And Company Substituted isoxazolines for control of plant phytopathogens
US4948801A (en) * 1988-07-29 1990-08-14 E. I. Du Pont De Nemours And Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
DE69316240T2 (de) * 1992-12-08 1998-05-20 Upjohn Co Durch eine tropon gruppe substituierte phenyloxazolidinone-derivate als antibakterielles mittel
PT730587E (pt) * 1993-11-26 2000-05-31 Pfizer 3-aril-2-isoxazolinas como agentes anti-inflamatorios
DE4425612A1 (de) * 1994-07-20 1996-04-04 Bayer Ag 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone
DE4425613A1 (de) * 1994-07-20 1996-01-25 Bayer Ag 5-gliedrige Heteroaryl-oxazolidinone
US5710159A (en) * 1996-05-09 1998-01-20 The Dupont Merck Pharmaceutical Company Integrin receptor antagonists

Also Published As

Publication number Publication date
US5990136A (en) 1999-11-23
EP0920421B1 (en) 2002-11-06
JP2000516245A (ja) 2000-12-05
DE69716925T2 (de) 2003-09-11
ES2186916T3 (es) 2003-05-16
DK0920421T3 (da) 2003-03-10
ATE227277T1 (de) 2002-11-15
EP0920421A1 (en) 1999-06-09
DE69716925D1 (de) 2002-12-12
WO1998007708A1 (en) 1998-02-26
US6093736A (en) 2000-07-25
AU3973697A (en) 1998-03-06

Similar Documents

Publication Publication Date Title
PT920421E (pt) Derivados de isoxazolina uteis como agentes antimicrobianos
DE69829846D1 (de) Antibakteriell wirksam oxazolidinone mit einer thiocarbonylfunktionalität
UY26551A1 (es) " agentes antibacterianos de 3-aminoquinazolin-2,4,dionas".
DE60118885D1 (de) Nitratsalze von antimikrobiellen wirkstoffen
PT942904E (pt) Derivados de 3-tiocarbamoilpirazol como pesticidas
PT1028961E (pt) Derivados de pleuromutilina como agentes antimicrobianos
PT960107E (pt) Compostos de paclitaxel 6-tio-substituidos
PT1453512E (pt) Derivados de acetileno tendo actividade antagonistica do mglur 5
DE69636791D1 (de) Derivate von glykopeptidantibiotika
DE60131138D1 (de) Antibakterielle mittel
ES2243579T3 (es) Derivados de pirazolopirideno.
ES2195397T3 (es) Quinazolin-2,4-dionas sustituidas en posicion 7 utiles como agentes antibacterianos.
BR0014775B1 (pt) misturas antimicrobianas de 1,3-bis (hidroximetil) -5,5-dimetilidantoina e 1,2-benzisotiazolin-3-ona.
DE69835536D1 (de) Zusammensetzungen zur behandlung von staphylococcus aureus infektionen
EA200500353A1 (ru) Производные линкомицина, обладающие антибактериальной активностью
UA83266C2 (en) Oxazole derivatives of tetracyclines
TR200301650T4 (tr) Ziraat ve bahçecilikte kullanım için okzim O-eter bileşikleri ve fungusitler
AR025379A1 (es) 9a-azalidas con actividad antibacteriana.
DK1073447T3 (da) N1-modificerede glycopeptider
PT1268475E (pt) Novos agentes bacterianos de benzosultam-oxazolidinona
TW200420561A (en) Antimicrobial 1-aryl dihydropyridone compounds
MXPA05009243A (es) N-aril-2-oxazolidinona-5-carboxamidas y sus derivados.
DE60014915D1 (de) Hypoxanthin- und thiohypxanthin-verbindungen
NO982879L (no) Vannlöselige antibiotika
BRPI0411537A (pt) derivados de lincomicina que possuem atividade antibacteriana