PT84561B - Processo aperfeicoado para a preparacao de derivados macrolidos - Google Patents

Processo aperfeicoado para a preparacao de derivados macrolidos

Info

Publication number
PT84561B
PT84561B PT84561A PT8456187A PT84561B PT 84561 B PT84561 B PT 84561B PT 84561 A PT84561 A PT 84561A PT 8456187 A PT8456187 A PT 8456187A PT 84561 B PT84561 B PT 84561B
Authority
PT
Portugal
Prior art keywords
macrolidary
derivatives
preparation
appropriate process
appropriate
Prior art date
Application number
PT84561A
Other languages
English (en)
Other versions
PT84561A (en
Inventor
Eddie Vi-Ping Tao
Jeffrey Thomas Vicenzi
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT84561A publication Critical patent/PT84561A/pt
Publication of PT84561B publication Critical patent/PT84561B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H5/00Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
PT84561A 1986-03-31 1987-03-26 Processo aperfeicoado para a preparacao de derivados macrolidos PT84561B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/846,446 US4921947A (en) 1986-03-31 1986-03-31 Process for preparing macrolide derivatives

Publications (2)

Publication Number Publication Date
PT84561A PT84561A (en) 1987-04-01
PT84561B true PT84561B (pt) 1989-11-10

Family

ID=25297965

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84561A PT84561B (pt) 1986-03-31 1987-03-26 Processo aperfeicoado para a preparacao de derivados macrolidos

Country Status (21)

Country Link
US (1) US4921947A (pt)
EP (1) EP0240264B1 (pt)
JP (1) JPH0710876B2 (pt)
KR (1) KR900001166B1 (pt)
CN (1) CN1018647B (pt)
AR (1) AR247402A1 (pt)
AT (1) ATE66678T1 (pt)
AU (1) AU593894B2 (pt)
CA (1) CA1292737C (pt)
DE (1) DE3772423D1 (pt)
DK (1) DK172935B1 (pt)
EG (1) EG18550A (pt)
ES (1) ES2028865T3 (pt)
GR (1) GR3002764T3 (pt)
HK (1) HK82492A (pt)
HU (1) HU199864B (pt)
IE (1) IE61018B1 (pt)
IL (1) IL82005A (pt)
NZ (1) NZ219784A (pt)
PT (1) PT84561B (pt)
ZA (1) ZA872201B (pt)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2638458A1 (fr) * 1988-10-27 1990-05-04 Adir Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW226373B (pt) * 1992-07-15 1994-07-11 Pfizer
AU6019794A (en) * 1993-03-18 1994-10-11 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at c-20
WO1995002594A1 (en) * 1993-07-15 1995-01-26 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
DE102004027417A1 (de) * 2004-06-04 2005-12-22 Basf Ag Verbundelement
PL2474545T3 (pl) 2005-12-13 2017-04-28 Incyte Holdings Corporation Podstawione heteroarylem pirolo[2,3-b]pirydyny i pirolo[2,3-b]pirymidyny jako inhibitory kinazy Janusowej
JP5126685B2 (ja) * 2006-05-01 2013-01-23 大正製薬株式会社 マクロライド誘導体
NZ574193A (en) * 2006-07-28 2011-09-30 Intervet Int Bv Macrolide synthesis process
EP2019112A1 (en) * 2007-07-26 2009-01-28 Intervet International BV Macrolide solid-state forms
KR101538599B1 (ko) * 2006-07-28 2015-07-21 인터벳 인터내셔널 비.브이. 마크롤라이드 합성 방법
JP5917544B2 (ja) 2010-11-19 2016-05-18 インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation Jak阻害剤としての複素環置換ピロロピリジンおよびピロロピリミジン
EA026201B1 (ru) 2010-11-19 2017-03-31 Инсайт Холдингс Корпорейшн Циклобутилзамещенные производные пирролопиридина и пирролопиримидина как ингибиторы jak
AR086983A1 (es) 2011-06-20 2014-02-05 Incyte Corp Derivados de azetidinil fenil, piridil o pirazinil carboxamida como inhibidores de jak
CA2856708C (en) 2011-11-25 2022-01-11 Bayer Intellectual Property Gmbh Antibacterial tylosin derivatives and methods for their preparation
CN102382159B (zh) * 2011-12-07 2013-11-13 齐鲁动物保健品有限公司 一种替米考星的制备方法
AU2014225938B2 (en) 2013-03-06 2018-07-19 Incyte Holdings Corporation Processes and intermediates for making a JAK inhibitor
JP6494600B2 (ja) 2013-05-23 2019-04-03 バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Animal Health Gmbh タイロシン誘導体およびその調製方法
CN105837648B (zh) * 2015-11-02 2018-07-06 湖北龙翔药业科技股份有限公司 一种磷酸替米考星的制备方法
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法
CN111269275A (zh) * 2020-03-09 2020-06-12 浙江康牧药业有限公司 一种替米考星的制备方法
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4454314A (en) * 1982-08-02 1984-06-12 Pfizer Inc. Antibacterial mycaminosyl tylonolide and related macrolide derivatives
AU561147B2 (en) * 1982-09-13 1987-04-30 Eli Lilly And Company 20-amino macrolide antibiotics
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
US4468511A (en) * 1983-02-28 1984-08-28 Eli Lilly And Company C-20- And C-23-Modified macrolide derivatives

Also Published As

Publication number Publication date
CA1292737C (en) 1991-12-03
HUT43087A (en) 1987-09-28
DK154087D0 (da) 1987-03-26
JPS62240681A (ja) 1987-10-21
IL82005A (en) 1991-08-16
ATE66678T1 (de) 1991-09-15
HK82492A (en) 1992-10-30
AU593894B2 (en) 1990-02-22
IE870796L (en) 1987-09-30
DK172935B1 (da) 1999-10-11
IL82005A0 (en) 1987-10-20
AR247402A1 (es) 1994-12-29
NZ219784A (en) 1989-01-27
EP0240264A2 (en) 1987-10-07
EP0240264A3 (en) 1987-11-19
GR3002764T3 (en) 1993-01-25
DE3772423D1 (de) 1991-10-02
IE61018B1 (en) 1994-09-07
EP0240264B1 (en) 1991-08-28
DK154087A (da) 1987-10-01
ES2028865T3 (es) 1992-07-16
ZA872201B (en) 1988-10-26
EG18550A (en) 1993-10-30
CN1018647B (zh) 1992-10-14
PT84561A (en) 1987-04-01
JPH0710876B2 (ja) 1995-02-08
KR870008906A (ko) 1987-10-21
KR900001166B1 (ko) 1990-02-27
US4921947A (en) 1990-05-01
AU7067087A (en) 1987-10-08
HU199864B (en) 1990-03-28
CN87102397A (zh) 1987-10-07

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