PT3029043T - Composto de benzoxaborole tricíclico, método para a sua preparação e sua utilização - Google Patents

Composto de benzoxaborole tricíclico, método para a sua preparação e sua utilização

Info

Publication number
PT3029043T
PT3029043T PT14831789T PT14831789T PT3029043T PT 3029043 T PT3029043 T PT 3029043T PT 14831789 T PT14831789 T PT 14831789T PT 14831789 T PT14831789 T PT 14831789T PT 3029043 T PT3029043 T PT 3029043T
Authority
PT
Portugal
Prior art keywords
preparation
method therefor
benzoxaborole compound
tricyclic benzoxaborole
tricyclic
Prior art date
Application number
PT14831789T
Other languages
English (en)
Inventor
Kim Soon-Hoe
Im Weon-Bin
Ha Seung-Bum
Park Jung-Sang
Kim Mi-Yeon
Choi Sung-Hak
Sung Hyun-Jung
Original Assignee
Dong A St Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dong A St Co Ltd filed Critical Dong A St Co Ltd
Publication of PT3029043T publication Critical patent/PT3029043T/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT14831789T 2013-07-30 2014-07-28 Composto de benzoxaborole tricíclico, método para a sua preparação e sua utilização PT3029043T (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR20130090493 2013-07-30
KR1020140093765A KR101636431B1 (ko) 2013-07-30 2014-07-24 트리사이클릭 벤즈옥사보롤 화합물, 이의 제조방법 및 용도

Publications (1)

Publication Number Publication Date
PT3029043T true PT3029043T (pt) 2018-10-26

Family

ID=52571626

Family Applications (1)

Application Number Title Priority Date Filing Date
PT14831789T PT3029043T (pt) 2013-07-30 2014-07-28 Composto de benzoxaborole tricíclico, método para a sua preparação e sua utilização

Country Status (17)

Country Link
US (1) US9676796B2 (pt)
EP (1) EP3029043B1 (pt)
JP (1) JP6130600B2 (pt)
KR (1) KR101636431B1 (pt)
CN (1) CN105452259B (pt)
AU (1) AU2014297102B2 (pt)
BR (1) BR112016001876B1 (pt)
CA (1) CA2918249C (pt)
ES (1) ES2688597T3 (pt)
HK (1) HK1218120A1 (pt)
IL (1) IL243699A0 (pt)
MX (1) MX363530B (pt)
NZ (1) NZ716154A (pt)
PT (1) PT3029043T (pt)
RU (1) RU2639153C2 (pt)
SG (1) SG11201600563UA (pt)
WO (1) WO2015016558A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
PE20160752A1 (es) 2013-08-09 2016-08-17 Anacor Pharmaceuticals Inc Compuestos de benzoxaborol triciclicos y usos de los mismos
WO2016001834A1 (en) 2014-07-01 2016-01-07 Daiichi Sankyo Company, Limited Tricyclic benzoxaboroles as antibacterial agents
MA41494B1 (fr) 2015-02-12 2020-10-28 Glaxosmithkline Ip No 2 Ltd Composés benzoxaborole substitués en position 4 et utilisations associées
RS64770B1 (sr) 2016-03-07 2023-11-30 Agrofresh Inc Sinergistički postupci upotrebe jedinjenja benzoksaborola i gasova za prezerviranje kao antimikrobnih agenasa za useve
CN113214302B (zh) * 2021-04-23 2022-06-24 四川大学 一种抑制金属β-内酰胺酶和/或丝氨酸β-内酰胺酶的3-取代五元环状硼酸酯衍生物
CA3239096A1 (en) * 2022-06-23 2023-12-28 Shanghai Micurx Pharmaceutical Co., Ltd. Methods and uses of boron compounds in the treatment of nontuberculous mycobacterium infections and pharmaceutical compositions for treatment of same

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7390806B2 (en) 2002-12-18 2008-06-24 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use
RU2397986C2 (ru) 2002-12-18 2010-08-27 Анакор Фармасьютикалз, Инк. Антибиотики, содержащие комплексы бориновой кислоты, и способы их получения
EP2987796B1 (en) 2005-02-16 2018-08-08 Anacor Pharmaceuticals, Inc. Halogen-substituted boronophthalides for the treatment of infections
RU2008131324A (ru) 2005-12-30 2010-02-10 Анакор Фармасьютикалз, Инк. (Us) Борсодержащие малые молекулы
ME02188B (me) 2006-02-16 2016-02-20 Anacor Pharmaceuticals Inc Mali molekuli koji sadrže boron kao antiinflamatorni agensi
JO3396B1 (ar) * 2007-06-20 2019-10-20 Anacor Pharmaceuticals Inc جزيئات صغيرة تحتوي على البورون
KR100925333B1 (ko) 2008-03-14 2009-11-04 엘지전자 주식회사 랜덤 액세스 과정에서 상향링크 동기화를 수행하는 방법
WO2009140309A2 (en) 2008-05-12 2009-11-19 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US20110212918A1 (en) 2009-11-11 2011-09-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
SG184268A1 (en) 2010-04-07 2012-10-30 Glaxosmithkline Llc Process for preparing benzoxaboroles
EP2613788B1 (en) 2010-09-07 2017-06-21 Anacor Pharmaceuticals, Inc. Benzoxaborole derivatives for treating bacterial infections
CA2858799A1 (en) 2011-12-22 2013-06-27 Micurx Pharmaceuticals, Inc. Tricyclic boron compounds for antimicrobial therapy
PE20160752A1 (es) 2013-08-09 2016-08-17 Anacor Pharmaceuticals Inc Compuestos de benzoxaborol triciclicos y usos de los mismos

Also Published As

Publication number Publication date
ES2688597T3 (es) 2018-11-05
KR20150014858A (ko) 2015-02-09
IL243699A0 (en) 2016-04-21
CN105452259A (zh) 2016-03-30
AU2014297102A1 (en) 2016-02-04
EP3029043A4 (en) 2017-04-05
RU2016103919A (ru) 2017-08-31
CA2918249A1 (en) 2015-02-05
EP3029043B1 (en) 2018-08-29
JP6130600B2 (ja) 2017-05-17
EP3029043A1 (en) 2016-06-08
US9676796B2 (en) 2017-06-13
NZ716154A (en) 2017-08-25
BR112016001876B1 (pt) 2022-02-22
SG11201600563UA (en) 2016-02-26
BR112016001876A2 (pt) 2017-08-01
MX2016001138A (es) 2016-04-29
RU2639153C2 (ru) 2017-12-20
US20160168167A1 (en) 2016-06-16
KR101636431B1 (ko) 2016-07-05
JP2016530250A (ja) 2016-09-29
AU2014297102B2 (en) 2017-02-23
CA2918249C (en) 2018-05-08
HK1218120A1 (zh) 2017-02-03
CN105452259B (zh) 2018-01-12
MX363530B (es) 2019-03-27
WO2015016558A1 (ko) 2015-02-05

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