MX363530B - Compuesto de benzoxaborol tricíclico, método de preparación y uso del mismo. - Google Patents
Compuesto de benzoxaborol tricíclico, método de preparación y uso del mismo.Info
- Publication number
- MX363530B MX363530B MX2016001138A MX2016001138A MX363530B MX 363530 B MX363530 B MX 363530B MX 2016001138 A MX2016001138 A MX 2016001138A MX 2016001138 A MX2016001138 A MX 2016001138A MX 363530 B MX363530 B MX 363530B
- Authority
- MX
- Mexico
- Prior art keywords
- preparation
- method therefor
- tricyclic benzoxaborole
- benzoxaborole compound
- tricyclic
- Prior art date
Links
- 238000002360 preparation method Methods 0.000 title abstract 2
- -1 benzoxaborole compound Chemical class 0.000 title 1
- GDMJXXLVTYSBBE-UHFFFAOYSA-N 1,2-benzoxaborole Chemical class C1=CC=C2OB=CC2=C1 GDMJXXLVTYSBBE-UHFFFAOYSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La presente invención se relaciona con un derivado de benzoxaborol tricíclico novedoso, con un método de preparación del mismo, y con el uso de una composición farmacéutica antibiótica que incluye al mismo como un ingrediente activo.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20130090493 | 2013-07-30 | ||
| KR1020140093765A KR101636431B1 (ko) | 2013-07-30 | 2014-07-24 | 트리사이클릭 벤즈옥사보롤 화합물, 이의 제조방법 및 용도 |
| PCT/KR2014/006894 WO2015016558A1 (ko) | 2013-07-30 | 2014-07-28 | 트리사이클릭 벤즈옥사보롤 화합물, 이의 제조방법 및 용도 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX2016001138A MX2016001138A (es) | 2016-04-29 |
| MX363530B true MX363530B (es) | 2019-03-27 |
Family
ID=52571626
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2016001138A MX363530B (es) | 2013-07-30 | 2014-07-28 | Compuesto de benzoxaborol tricíclico, método de preparación y uso del mismo. |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US9676796B2 (es) |
| EP (1) | EP3029043B1 (es) |
| JP (1) | JP6130600B2 (es) |
| KR (1) | KR101636431B1 (es) |
| CN (1) | CN105452259B (es) |
| AU (1) | AU2014297102B2 (es) |
| BR (1) | BR112016001876B1 (es) |
| CA (1) | CA2918249C (es) |
| ES (1) | ES2688597T3 (es) |
| HK (1) | HK1218120A1 (es) |
| IL (1) | IL243699A0 (es) |
| MX (1) | MX363530B (es) |
| NZ (1) | NZ716154A (es) |
| PT (1) | PT3029043T (es) |
| RU (1) | RU2639153C2 (es) |
| SG (1) | SG11201600563UA (es) |
| WO (1) | WO2015016558A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| EP3030519B1 (en) | 2013-08-09 | 2022-01-05 | Glaxosmithkline Intellectual Property (No. 2) Limited | Tricyclic benzoxaborole compounds and uses thereof |
| EP3164404B1 (en) | 2014-07-01 | 2019-04-03 | Daiichi Sankyo Company, Limited | Tricyclic benzoxaboroles as antibacterial agents |
| MA41494B1 (fr) | 2015-02-12 | 2020-10-28 | Glaxosmithkline Ip No 2 Ltd | Composés benzoxaborole substitués en position 4 et utilisations associées |
| EP3426029B1 (en) | 2016-03-07 | 2023-08-30 | AgroFresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
| CN113214302B (zh) * | 2021-04-23 | 2022-06-24 | 四川大学 | 一种抑制金属β-内酰胺酶和/或丝氨酸β-内酰胺酶的3-取代五元环状硼酸酯衍生物 |
| JP2025520237A (ja) * | 2022-06-23 | 2025-07-03 | ミクウルク ファーマシューティカルズ， インコーポレイテッド | ホウ素化合物を用いて非結核性マイコバクテリア感染症を治療する方法及びその用途、並びに同じ疾患を治療するための医薬組成物 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7390806B2 (en) | 2002-12-18 | 2008-06-24 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
| RU2397986C2 (ru) * | 2002-12-18 | 2010-08-27 | Анакор Фармасьютикалз, Инк. | Антибиотики, содержащие комплексы бориновой кислоты, и способы их получения |
| HUE026021T2 (en) | 2005-02-16 | 2016-05-30 | Anacor Pharmaceuticals Inc | Biocidal boron phthalide (boronophthalide) compounds |
| CN106008583A (zh) | 2005-12-30 | 2016-10-12 | 安纳考尔医药公司 | 含硼的小分子 |
| BRPI0708051A2 (pt) | 2006-02-16 | 2011-05-17 | Anacor Pharmaceuticals Inc | moléculas pequenas contendo boro como agentes antiflamatórios |
| JO3396B1 (ar) | 2007-06-20 | 2019-10-20 | Anacor Pharmaceuticals Inc | جزيئات صغيرة تحتوي على البورون |
| KR100925333B1 (ko) | 2008-03-14 | 2009-11-04 | 엘지전자 주식회사 | 랜덤 액세스 과정에서 상향링크 동기화를 수행하는 방법 |
| WO2009140309A2 (en) | 2008-05-12 | 2009-11-19 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2011060196A1 (en) | 2009-11-11 | 2011-05-19 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2011127143A1 (en) | 2010-04-07 | 2011-10-13 | Glaxosmithkline Llc | Process for preparing benzoxaboroles |
| HRP20211762T1 (hr) | 2010-09-07 | 2022-02-18 | Anacor Pharmaceuticals, Inc. | Derivati benzoksaborola za liječenje bakterijskih infekcija |
| KR20140114380A (ko) | 2011-12-22 | 2014-09-26 | 미큐알엑스 파마슈티칼스, 인크. | 항미생물 요법용 트리시클릭 붕소 화합물 |
| EP3030519B1 (en) | 2013-08-09 | 2022-01-05 | Glaxosmithkline Intellectual Property (No. 2) Limited | Tricyclic benzoxaborole compounds and uses thereof |
-
2014
- 2014-07-24 KR KR1020140093765A patent/KR101636431B1/ko active Active
- 2014-07-28 CA CA2918249A patent/CA2918249C/en active Active
- 2014-07-28 SG SG11201600563UA patent/SG11201600563UA/en unknown
- 2014-07-28 CN CN201480043221.5A patent/CN105452259B/zh active Active
- 2014-07-28 US US14/908,006 patent/US9676796B2/en active Active
- 2014-07-28 PT PT14831789T patent/PT3029043T/pt unknown
- 2014-07-28 WO PCT/KR2014/006894 patent/WO2015016558A1/ko not_active Ceased
- 2014-07-28 MX MX2016001138A patent/MX363530B/es unknown
- 2014-07-28 BR BR112016001876-1A patent/BR112016001876B1/pt active IP Right Grant
- 2014-07-28 AU AU2014297102A patent/AU2014297102B2/en active Active
- 2014-07-28 RU RU2016103919A patent/RU2639153C2/ru active
- 2014-07-28 ES ES14831789.4T patent/ES2688597T3/es active Active
- 2014-07-28 HK HK16106048.1A patent/HK1218120A1/zh unknown
- 2014-07-28 EP EP14831789.4A patent/EP3029043B1/en active Active
- 2014-07-28 NZ NZ716154A patent/NZ716154A/en unknown
- 2014-07-28 JP JP2016531520A patent/JP6130600B2/ja active Active
-
2016
- 2016-01-20 IL IL243699A patent/IL243699A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR101636431B1 (ko) | 2016-07-05 |
| EP3029043B1 (en) | 2018-08-29 |
| AU2014297102A1 (en) | 2016-02-04 |
| RU2639153C2 (ru) | 2017-12-20 |
| PT3029043T (pt) | 2018-10-26 |
| ES2688597T3 (es) | 2018-11-05 |
| US9676796B2 (en) | 2017-06-13 |
| NZ716154A (en) | 2017-08-25 |
| CA2918249C (en) | 2018-05-08 |
| CN105452259B (zh) | 2018-01-12 |
| JP6130600B2 (ja) | 2017-05-17 |
| KR20150014858A (ko) | 2015-02-09 |
| US20160168167A1 (en) | 2016-06-16 |
| BR112016001876B1 (pt) | 2022-02-22 |
| BR112016001876A2 (pt) | 2017-08-01 |
| AU2014297102B2 (en) | 2017-02-23 |
| WO2015016558A1 (ko) | 2015-02-05 |
| IL243699A0 (en) | 2016-04-21 |
| CN105452259A (zh) | 2016-03-30 |
| JP2016530250A (ja) | 2016-09-29 |
| EP3029043A1 (en) | 2016-06-08 |
| MX2016001138A (es) | 2016-04-29 |
| EP3029043A4 (en) | 2017-04-05 |
| HK1218120A1 (zh) | 2017-02-03 |
| RU2016103919A (ru) | 2017-08-31 |
| SG11201600563UA (en) | 2016-02-26 |
| CA2918249A1 (en) | 2015-02-05 |
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