MX363530B - Compuesto de benzoxaborol tricíclico, método de preparación y uso del mismo. - Google Patents

Compuesto de benzoxaborol tricíclico, método de preparación y uso del mismo.

Info

Publication number
MX363530B
MX363530B MX2016001138A MX2016001138A MX363530B MX 363530 B MX363530 B MX 363530B MX 2016001138 A MX2016001138 A MX 2016001138A MX 2016001138 A MX2016001138 A MX 2016001138A MX 363530 B MX363530 B MX 363530B
Authority
MX
Mexico
Prior art keywords
preparation
method therefor
tricyclic benzoxaborole
benzoxaborole compound
tricyclic
Prior art date
Application number
MX2016001138A
Other languages
English (en)
Other versions
MX2016001138A (es
Inventor
Kim Soon-Hoe
Sang Park Jung-
Yeon Kim Mi-
Hak Choi Sung-
Jung Sung Hyun-
Bin Im Weon-
Bum Ha Seung-
Original Assignee
Dong A St Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dong A St Co Ltd filed Critical Dong A St Co Ltd
Publication of MX2016001138A publication Critical patent/MX2016001138A/es
Publication of MX363530B publication Critical patent/MX363530B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

La presente invención se relaciona con un derivado de benzoxaborol tricíclico novedoso, con un método de preparación del mismo, y con el uso de una composición farmacéutica antibiótica que incluye al mismo como un ingrediente activo.
MX2016001138A 2013-07-30 2014-07-28 Compuesto de benzoxaborol tricíclico, método de preparación y uso del mismo. MX363530B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR20130090493 2013-07-30
KR1020140093765A KR101636431B1 (ko) 2013-07-30 2014-07-24 트리사이클릭 벤즈옥사보롤 화합물, 이의 제조방법 및 용도
PCT/KR2014/006894 WO2015016558A1 (ko) 2013-07-30 2014-07-28 트리사이클릭 벤즈옥사보롤 화합물, 이의 제조방법 및 용도

Publications (2)

Publication Number Publication Date
MX2016001138A MX2016001138A (es) 2016-04-29
MX363530B true MX363530B (es) 2019-03-27

Family

ID=52571626

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016001138A MX363530B (es) 2013-07-30 2014-07-28 Compuesto de benzoxaborol tricíclico, método de preparación y uso del mismo.

Country Status (17)

Country Link
US (1) US9676796B2 (es)
EP (1) EP3029043B1 (es)
JP (1) JP6130600B2 (es)
KR (1) KR101636431B1 (es)
CN (1) CN105452259B (es)
AU (1) AU2014297102B2 (es)
BR (1) BR112016001876B1 (es)
CA (1) CA2918249C (es)
ES (1) ES2688597T3 (es)
HK (1) HK1218120A1 (es)
IL (1) IL243699A0 (es)
MX (1) MX363530B (es)
NZ (1) NZ716154A (es)
PT (1) PT3029043T (es)
RU (1) RU2639153C2 (es)
SG (1) SG11201600563UA (es)
WO (1) WO2015016558A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
CN105492388B (zh) 2013-08-09 2018-12-21 葛兰素史克知识产权第二有限公司 三环苯并氧杂硼杂环戊烯化合物及其用途
JP6605513B2 (ja) 2014-07-01 2019-11-13 第一三共株式会社 抗菌剤としての三環式ベンゾオキサボロール
MA41495A (fr) 2015-02-12 2017-12-19 Anacor Pharmaceuticals Inc Composés benzoxaborole et leurs utilisations
NZ745681A (en) 2016-03-07 2022-05-27 Agrofresh Inc Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops
CN113214302B (zh) * 2021-04-23 2022-06-24 四川大学 一种抑制金属β-内酰胺酶和/或丝氨酸β-内酰胺酶的3-取代五元环状硼酸酯衍生物
CN119233823A (zh) * 2022-06-23 2024-12-31 上海盟科药业股份有限公司 硼化合物治疗非结核分枝杆菌感染的方法和用途及用于治疗相同疾病的药物组合物

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2397986C2 (ru) 2002-12-18 2010-08-27 Анакор Фармасьютикалз, Инк. Антибиотики, содержащие комплексы бориновой кислоты, и способы их получения
US7390806B2 (en) 2002-12-18 2008-06-24 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use
JP5038912B2 (ja) 2005-02-16 2012-10-03 アナコール ファーマシューティカルズ，インコーポレイテッド ホウ素含有小分子
US7767657B2 (en) 2005-02-16 2010-08-03 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
NZ570257A (en) * 2006-02-16 2011-11-25 Anacor Pharmaceuticals Inc Boron-containing small molecules as anti-inflammatory agents
JO3396B1 (ar) * 2007-06-20 2019-10-20 Anacor Pharmaceuticals Inc جزيئات صغيرة تحتوي على البورون
KR100925333B1 (ko) 2008-03-14 2009-11-04 엘지전자 주식회사 랜덤 액세스 과정에서 상향링크 동기화를 수행하는 방법
US20100256092A1 (en) 2008-05-12 2010-10-07 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US20110212918A1 (en) 2009-11-11 2011-09-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
JP5603998B2 (ja) 2010-04-07 2014-10-08 グラクソスミスクライン エルエルシー ベンゾオキサボロールの調製方法
SG10201507032YA (en) 2010-09-07 2015-10-29 Anacor Pharmaceuticals Inc Benzoxaborole derivatives for treating bacterial infections
US8530452B2 (en) 2011-12-22 2013-09-10 Micurx Pharmaceuticals, Inc. Tricyclic boron compounds for antimicrobial therapy
CN105492388B (zh) 2013-08-09 2018-12-21 葛兰素史克知识产权第二有限公司 三环苯并氧杂硼杂环戊烯化合物及其用途

Also Published As

Publication number Publication date
WO2015016558A1 (ko) 2015-02-05
KR101636431B1 (ko) 2016-07-05
JP2016530250A (ja) 2016-09-29
EP3029043B1 (en) 2018-08-29
NZ716154A (en) 2017-08-25
EP3029043A4 (en) 2017-04-05
RU2016103919A (ru) 2017-08-31
KR20150014858A (ko) 2015-02-09
MX2016001138A (es) 2016-04-29
SG11201600563UA (en) 2016-02-26
CN105452259A (zh) 2016-03-30
JP6130600B2 (ja) 2017-05-17
AU2014297102B2 (en) 2017-02-23
AU2014297102A1 (en) 2016-02-04
BR112016001876A2 (pt) 2017-08-01
US20160168167A1 (en) 2016-06-16
CA2918249A1 (en) 2015-02-05
BR112016001876B1 (pt) 2022-02-22
CN105452259B (zh) 2018-01-12
PT3029043T (pt) 2018-10-26
EP3029043A1 (en) 2016-06-08
US9676796B2 (en) 2017-06-13
CA2918249C (en) 2018-05-08
IL243699A0 (en) 2016-04-21
RU2639153C2 (ru) 2017-12-20
HK1218120A1 (zh) 2017-02-03
ES2688597T3 (es) 2018-11-05

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