PT2874602T - Solução injetável sobressaturada de acetaminifeno para administração espinal - Google Patents

Solução injetável sobressaturada de acetaminifeno para administração espinal

Info

Publication number
PT2874602T
PT2874602T PT137654505T PT13765450T PT2874602T PT 2874602 T PT2874602 T PT 2874602T PT 137654505 T PT137654505 T PT 137654505T PT 13765450 T PT13765450 T PT 13765450T PT 2874602 T PT2874602 T PT 2874602T
Authority
PT
Portugal
Prior art keywords
spinal administration
acetaminophen solution
injectable
supersaturated acetaminophen
injectable supersaturated
Prior art date
Application number
PT137654505T
Other languages
English (en)
Inventor
Donati Elisabetta
Mitidieri Augusto
Caronzolo Nicola
Original Assignee
Sintetica S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46690603&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2874602(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sintetica S A filed Critical Sintetica S A
Publication of PT2874602T publication Critical patent/PT2874602T/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A61K31/24Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
    • A61K31/245Amino benzoic acid types, e.g. procaine, novocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0085Brain, e.g. brain implants; Spinal cord
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • A61P23/02Local anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Emergency Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Anesthesiology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PT137654505T 2012-06-29 2013-06-27 Solução injetável sobressaturada de acetaminifeno para administração espinal PT2874602T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT001154A ITMI20121154A1 (it) 2012-06-29 2012-06-29 Soluzione iniettabile di acetaminofene per la somministrazione spinale

Publications (1)

Publication Number Publication Date
PT2874602T true PT2874602T (pt) 2016-07-13

Family

ID=46690603

Family Applications (1)

Application Number Title Priority Date Filing Date
PT137654505T PT2874602T (pt) 2012-06-29 2013-06-27 Solução injetável sobressaturada de acetaminifeno para administração espinal

Country Status (44)

Country Link
US (2) US11344517B2 (pt)
EP (1) EP2874602B1 (pt)
JP (1) JP5876620B2 (pt)
KR (1) KR102118227B1 (pt)
CN (1) CN104487051B (pt)
AP (1) AP2014008152A0 (pt)
AR (1) AR091633A1 (pt)
AU (1) AU2013282753B2 (pt)
BR (1) BR112014032818B1 (pt)
CA (1) CA2876801C (pt)
CL (1) CL2014003536A1 (pt)
CO (1) CO7240357A2 (pt)
CR (1) CR20150036A (pt)
CU (1) CU20140150A7 (pt)
CY (1) CY1117691T1 (pt)
DK (1) DK2874602T3 (pt)
DO (1) DOP2014000302A (pt)
EA (1) EA028909B1 (pt)
EC (1) ECSP15000500A (pt)
ES (1) ES2578012T3 (pt)
GE (1) GEP201706689B (pt)
HR (1) HRP20160706T1 (pt)
HU (1) HUE029431T2 (pt)
IL (1) IL236423A (pt)
IT (1) ITMI20121154A1 (pt)
MA (1) MA37811B1 (pt)
MD (1) MD4537C1 (pt)
ME (1) ME02431B (pt)
MX (1) MX369264B (pt)
MY (1) MY169251A (pt)
NI (1) NI201400147A (pt)
NZ (1) NZ703829A (pt)
PE (1) PE20150331A1 (pt)
PH (1) PH12015500178A1 (pt)
PL (1) PL2874602T3 (pt)
PT (1) PT2874602T (pt)
RS (1) RS54844B1 (pt)
SG (2) SG10201704482YA (pt)
SI (1) SI2874602T1 (pt)
SM (1) SMT201600248B (pt)
TN (1) TN2014000526A1 (pt)
UA (1) UA117101C2 (pt)
WO (1) WO2014002042A1 (pt)
ZA (1) ZA201409478B (pt)

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0646400B1 (en) * 1993-04-14 2001-07-18 Nippon Sanso Corporation Dissolved oxygen reducing apparatus
US6171298B1 (en) * 1996-05-03 2001-01-09 Situs Corporation Intravesical infuser
FR2751875B1 (fr) 1996-08-05 1998-12-24 Scr Newpharm Nouvelles formulations liquides stables a base de paracetamol et leur mode de preparation
FR2809619B1 (fr) 2000-06-06 2004-09-24 Pharmatop Nouvelles formulations aqueuses de principes actifs sensibles a l'oxydation et leur procede d'obtention
DE10112325A1 (de) * 2001-03-13 2002-10-02 Fresenius Kabi De Gmbh Lagerstabile Fertiginfusionslösungen des Paracetamols
SK2822004A3 (sk) * 2001-12-18 2005-01-03 Uni-Pharma Kleon Tsetis Pharmaceutical Laboratories S.A. Parenterálny prípravok obsahujúci paracetamol
FR2851164B1 (fr) 2003-02-14 2005-04-22 Xuan Tho Nguyen Formulation liquide injectable de paracetamol
DE102005037653A1 (de) * 2005-08-05 2007-02-15 Theraselect Gmbh Stabile, flüssige Formulierung von Paracetamol
US9943479B2 (en) * 2006-07-18 2018-04-17 Genfarma Laboratorio S.L. Injectable liquid paracetamol formulation
CN101015542A (zh) * 2007-02-13 2007-08-15 天津生机集团有限公司 家畜用复方对乙酰氨基酚注射液及其制备方法
MD3528G2 (ro) * 2007-09-28 2008-11-30 Сергей ШАНДРУ Metodă de anestezie spinală continuă la pacienţii în etate
US9399012B2 (en) * 2007-11-13 2016-07-26 Mallinckrodt Ip Reduced dose intravenous acetaminophen
WO2009098716A2 (en) 2008-01-17 2009-08-13 Aptuit Laurus Private Limited Stable pharmaceutical aqueous compositions
WO2009143558A1 (en) 2008-05-26 2009-12-03 Silphion Pty Limited Injectable formulations
EP2243477A1 (de) 2009-04-22 2010-10-27 Fresenius Kabi Deutschland GmbH Paracetamol zur parenteralen Verabreichung
JP2013006770A (ja) 2009-10-09 2013-01-10 Ssp Co Ltd アセトアミノフェン含有経口液剤
CA2802303C (en) * 2010-06-30 2016-06-14 Troikaa Pharmaceuticals Limited Pharmaceutical compositions comprising paracetamol and process for preparing the same

Also Published As

Publication number Publication date
MA37811A1 (fr) 2016-10-31
KR102118227B1 (ko) 2020-06-03
ECSP15000500A (es) 2015-11-30
MX2014015402A (es) 2015-06-17
EA028909B1 (ru) 2018-01-31
CR20150036A (es) 2015-03-13
CN104487051B (zh) 2017-12-12
MA37811B1 (fr) 2017-07-31
MD4537C1 (ro) 2018-07-31
IL236423A (en) 2017-07-31
PE20150331A1 (es) 2015-03-07
CA2876801C (en) 2020-11-03
CU20140150A7 (es) 2015-10-27
US20150148379A1 (en) 2015-05-28
RS54844B1 (sr) 2016-10-31
BR112014032818A2 (pt) 2017-06-27
JP2015522004A (ja) 2015-08-03
PH12015500178B1 (en) 2015-04-06
MD4537B1 (ro) 2017-12-31
GEP201706689B (en) 2017-06-26
UA117101C2 (uk) 2018-06-25
BR112014032818B1 (pt) 2022-06-14
AU2013282753B2 (en) 2017-03-02
ME02431B (me) 2016-09-20
ES2578012T3 (es) 2016-07-20
JP5876620B2 (ja) 2016-03-02
EP2874602B1 (en) 2016-03-30
AR091633A1 (es) 2015-02-18
HRP20160706T1 (hr) 2016-08-12
PL2874602T3 (pl) 2016-10-31
US20160128955A1 (en) 2016-05-12
MY169251A (en) 2019-03-19
DOP2014000302A (es) 2015-03-15
ZA201409478B (en) 2016-01-27
CA2876801A1 (en) 2014-01-03
CL2014003536A1 (es) 2015-05-08
ITMI20121154A1 (it) 2013-12-30
SMT201600248B (it) 2016-08-31
EP2874602A1 (en) 2015-05-27
DK2874602T3 (en) 2016-07-04
NI201400147A (es) 2015-04-13
CY1117691T1 (el) 2017-05-17
CN104487051A (zh) 2015-04-01
US11344517B2 (en) 2022-05-31
IL236423A0 (en) 2015-02-26
PH12015500178A1 (en) 2015-04-06
EA201500065A1 (ru) 2015-10-30
HUE029431T2 (en) 2017-03-28
MD20140138A2 (ro) 2015-06-30
TN2014000526A1 (en) 2016-03-30
AU2013282753A1 (en) 2015-02-05
KR20150027160A (ko) 2015-03-11
SG11201408479WA (en) 2015-01-29
NZ703829A (en) 2016-06-24
SI2874602T1 (sl) 2016-09-30
AP2014008152A0 (en) 2014-12-31
WO2014002042A1 (en) 2014-01-03
CO7240357A2 (es) 2015-04-17
SG10201704482YA (en) 2017-07-28
MX369264B (es) 2019-11-04

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