PT1456218E - Derivados de avermectina b1 possuindo um substituinte aminossulfoniloxi na posição 4 - Google Patents

Derivados de avermectina b1 possuindo um substituinte aminossulfoniloxi na posição 4 Download PDF

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Publication number
PT1456218E
PT1456218E PT02796710T PT02796710T PT1456218E PT 1456218 E PT1456218 E PT 1456218E PT 02796710 T PT02796710 T PT 02796710T PT 02796710 T PT02796710 T PT 02796710T PT 1456218 E PT1456218 E PT 1456218E
Authority
PT
Portugal
Prior art keywords
aminosulfonyloxy
avermectin
substituent
derivatives
aminosulfonyloxy substituent
Prior art date
Application number
PT02796710T
Other languages
English (en)
Portuguese (pt)
Inventor
Jerome Cassayre
Original Assignee
Merial Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Ltd filed Critical Merial Ltd
Publication of PT1456218E publication Critical patent/PT1456218E/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/10Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
PT02796710T 2001-12-21 2002-12-20 Derivados de avermectina b1 possuindo um substituinte aminossulfoniloxi na posição 4 PT1456218E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH23632001 2001-12-21
CH11902002 2002-07-05

Publications (1)

Publication Number Publication Date
PT1456218E true PT1456218E (pt) 2008-08-06

Family

ID=25738950

Family Applications (1)

Application Number Title Priority Date Filing Date
PT02796710T PT1456218E (pt) 2001-12-21 2002-12-20 Derivados de avermectina b1 possuindo um substituinte aminossulfoniloxi na posição 4

Country Status (26)

Country Link
US (1) US6933260B2 (enExample)
EP (1) EP1456218B1 (enExample)
JP (1) JP2005513137A (enExample)
KR (1) KR20040068335A (enExample)
CN (1) CN1608075A (enExample)
AR (1) AR037938A1 (enExample)
AT (1) ATE397007T1 (enExample)
AU (1) AU2002361197A1 (enExample)
BR (1) BR0215170A (enExample)
CA (1) CA2469905A1 (enExample)
CO (1) CO5590963A2 (enExample)
CY (1) CY1108269T1 (enExample)
DE (1) DE60226895D1 (enExample)
DK (1) DK1456218T3 (enExample)
ES (1) ES2307823T3 (enExample)
HU (1) HUP0402290A2 (enExample)
IL (1) IL162452A0 (enExample)
MA (1) MA26300A1 (enExample)
MX (1) MXPA04006121A (enExample)
NZ (1) NZ533584A (enExample)
PL (1) PL370835A1 (enExample)
PT (1) PT1456218E (enExample)
RU (1) RU2004122622A (enExample)
SI (1) SI1456218T1 (enExample)
TW (1) TW200301079A (enExample)
WO (1) WO2003053988A2 (enExample)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EG23124A (en) * 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
TW200407330A (en) * 2002-05-07 2004-05-16 Syngenta Participations Ag 4"-Deoxy-4"-(S)-amido avermectin derivatives
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302310D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
FR2854071B1 (fr) * 2003-04-25 2009-01-30 Ethypharm Sa Procede de dispersion de substances hydrosolubles ou hydrophiles dans un fluide a pression supercritique
GB0313937D0 (en) * 2003-06-16 2003-07-23 Syngenta Participations Ag Avermectin B1 monosaccharide derivatives having an aminosulfonyloxy substituentin the 4'-position
GB0320176D0 (en) * 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
EP1849363A1 (en) * 2006-03-09 2007-10-31 Cheminova A/S Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin
DK2568980T3 (en) 2010-05-12 2015-11-30 Merial Inc INJECTABLE PARASITICIDE FORMULATIONS OF LEVAMISOL AND MACROCYCLIC LACTONS
WO2012078605A1 (en) 2010-12-07 2012-06-14 Merial Limited Topical combination formulations of macrocyclic lactones with synthetic pyrethroids
CN103936755B (zh) * 2014-04-08 2016-03-23 甘肃省农业科学院植物保护研究所 一种米尔贝霉素类似物及其制备方法和在农药中的应用
RU2554350C1 (ru) * 2014-04-18 2015-06-27 Игорь Викторович Заварзин Инсектицидный агент
RU2554074C1 (ru) * 2014-04-18 2015-06-27 Игорь Викторович Заварзин Антипаразитарный агент
HRP20220479T1 (hr) 2016-06-01 2022-05-27 Athira Pharma, Inc. Spojevi
CN108690108B (zh) * 2018-07-27 2022-03-11 河北威远生物化工有限公司 一种磺酰胺基取代的阿维菌素B2a/B2b衍生物及其制备方法与应用
US11351149B2 (en) 2020-09-03 2022-06-07 Pfizer Inc. Nitrile-containing antiviral compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4427663A (en) * 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof

Also Published As

Publication number Publication date
IL162452A0 (en) 2005-11-20
DK1456218T3 (da) 2008-08-04
PL370835A1 (en) 2005-05-30
WO2003053988A3 (en) 2003-12-11
SI1456218T1 (sl) 2008-10-31
TW200301079A (en) 2003-07-01
HUP0402290A2 (hu) 2005-02-28
CY1108269T1 (el) 2014-02-12
CN1608075A (zh) 2005-04-20
JP2005513137A (ja) 2005-05-12
EP1456218A2 (en) 2004-09-15
KR20040068335A (ko) 2004-07-30
BR0215170A (pt) 2004-10-19
RU2004122622A (ru) 2006-01-20
MA26300A1 (fr) 2004-09-01
US6933260B2 (en) 2005-08-23
US20050032717A1 (en) 2005-02-10
CA2469905A1 (en) 2003-07-03
NZ533584A (en) 2005-12-23
DE60226895D1 (de) 2008-07-10
CO5590963A2 (es) 2005-12-30
ES2307823T3 (es) 2008-12-01
AR037938A1 (es) 2004-12-22
MXPA04006121A (es) 2004-10-29
AU2002361197A1 (en) 2003-07-09
WO2003053988A2 (en) 2003-07-03
EP1456218B1 (en) 2008-05-28
ATE397007T1 (de) 2008-06-15

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