PT1385850E - Novo processo para a preparacao de oxabispidinas - Google Patents

Novo processo para a preparacao de oxabispidinas

Info

Publication number
PT1385850E
PT1385850E PT02718766T PT02718766T PT1385850E PT 1385850 E PT1385850 E PT 1385850E PT 02718766 T PT02718766 T PT 02718766T PT 02718766 T PT02718766 T PT 02718766T PT 1385850 E PT1385850 E PT 1385850E
Authority
PT
Portugal
Prior art keywords
sup
formula
compound
preparation
oxabispidins
Prior art date
Application number
PT02718766T
Other languages
English (en)
Inventor
David Cladingboel
Cheema Lal
Sinclair Rhona
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of PT1385850E publication Critical patent/PT1385850E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT02718766T 2001-04-12 2002-04-12 Novo processo para a preparacao de oxabispidinas PT1385850E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0101324A SE0101324D0 (sv) 2001-04-12 2001-04-12 New process

Publications (1)

Publication Number Publication Date
PT1385850E true PT1385850E (pt) 2005-03-31

Family

ID=20283781

Family Applications (1)

Application Number Title Priority Date Filing Date
PT02718766T PT1385850E (pt) 2001-04-12 2002-04-12 Novo processo para a preparacao de oxabispidinas

Country Status (20)

Country Link
US (2) US7169921B2 (pt)
EP (1) EP1385850B1 (pt)
JP (1) JP4248880B2 (pt)
KR (1) KR100848613B1 (pt)
CN (1) CN1267435C (pt)
AT (1) ATE284405T1 (pt)
AU (1) AU2002249748B2 (pt)
BR (1) BR0208861A (pt)
CA (1) CA2443475A1 (pt)
DE (1) DE60202203T2 (pt)
ES (1) ES2233809T3 (pt)
HK (1) HK1060886A1 (pt)
IL (2) IL158249A0 (pt)
MX (1) MXPA03009211A (pt)
NO (1) NO20034526L (pt)
NZ (1) NZ528515A (pt)
PT (1) PT1385850E (pt)
SE (1) SE0101324D0 (pt)
WO (1) WO2002083690A1 (pt)
ZA (1) ZA200307676B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0101324D0 (sv) * 2001-04-12 2001-04-12 Astrazeneca Ab New process
GB0223712D0 (en) 2002-10-14 2002-11-20 Astrazeneca Ab Chemical intermediate
US20040192738A1 (en) * 2003-03-18 2004-09-30 Aventis Pharma Deutschland Gmbh 2-(Butyl-1-sulfonylamino)-N-[1(R)-(6-methoxypyridin-3-yl)propyl] benzamide, its use as a medicament, and pharmaceutical preparations comprising it
SE0401539D0 (sv) * 2004-06-15 2004-06-15 Astrazeneca Ab New compounds
SE0401540D0 (sv) * 2004-06-15 2004-06-15 Astrazeneca Ab New compounds
CA2609938A1 (en) * 2005-06-13 2006-12-21 Astrazeneca Ab New oxabispidine compounds for the treatment of cardiac arrhythmias
RU2008101665A (ru) * 2005-06-16 2009-07-27 Гириндус Аг (De) Синтез производных гидрохинона
AR057364A1 (es) * 2005-06-20 2007-11-28 Astrazeneca Ab Proceso para el aislamiento de 4-(oxiranilmetoxi) -benzonitrilos
AR053901A1 (es) * 2005-06-20 2007-05-23 Astrazeneca Ab Formas fisicas de oxabispidinas n,n'- disustituidas
WO2006137770A1 (en) * 2005-06-20 2006-12-28 Astrazeneca Ab Process for the preparation of n,n´- disubstituted oxabispidines
BRPI0611842A2 (pt) * 2005-06-20 2016-08-30 Astrazeneca Ab "processo para a preparação de um composto"
MX2007016492A (es) * 2005-06-20 2008-03-07 Astrazeneca Ab Proceso para la preparacion de sales de acido sulfonico de oxabispidinas.
WO2006137774A1 (en) * 2005-06-20 2006-12-28 Astrazeneca Ab Process for the production of (alkoxycarbonylamino)alkyl sulfonates
ES2852054T3 (es) 2013-03-15 2021-09-10 Global Blood Therapeutics Inc Compuestos y usos de los mismos para la modulación de hemoglobina
EA202092627A1 (ru) 2013-11-18 2021-09-30 Глобал Блад Терапьютикс, Инк. Соединения и их применения для модуляции гемоглобина

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3196154A (en) * 1962-05-17 1965-07-20 Sterling Drug Inc 3-substituted-9-methyl-3, 9-diazabicyclo [3.3.1] nonanes
US5110933A (en) * 1989-11-13 1992-05-05 Board Of Regents Of Oklahoma State University Salts of 3-azabicyclo[3.3.1]nonanes as antiarrhythmic agents, and precursors thereof
SE9704709D0 (sv) * 1997-12-17 1997-12-17 Astra Ab Pharmaceutically active compounds
SE9903759D0 (sv) 1999-10-18 1999-10-18 Astra Ab Pharmaceutically active compounds
SE0101324D0 (sv) * 2001-04-12 2001-04-12 Astrazeneca Ab New process

Also Published As

Publication number Publication date
DE60202203T2 (de) 2005-12-15
JP4248880B2 (ja) 2009-04-02
US20070197519A1 (en) 2007-08-23
SE0101324D0 (sv) 2001-04-12
CN1267435C (zh) 2006-08-02
WO2002083690A1 (en) 2002-10-24
HK1060886A1 (en) 2004-08-27
CA2443475A1 (en) 2002-10-24
EP1385850A1 (en) 2004-02-04
NO20034526D0 (no) 2003-10-09
ZA200307676B (en) 2004-07-13
KR100848613B1 (ko) 2008-07-28
IL158249A0 (en) 2004-05-12
ATE284405T1 (de) 2004-12-15
JP2004533432A (ja) 2004-11-04
DE60202203D1 (de) 2005-01-13
KR20030087065A (ko) 2003-11-12
US7169921B2 (en) 2007-01-30
BR0208861A (pt) 2004-10-19
NZ528515A (en) 2005-06-24
ES2233809T3 (es) 2005-06-16
CN1520417A (zh) 2004-08-11
EP1385850B1 (en) 2004-12-08
AU2002249748B2 (en) 2008-02-28
US20040181060A1 (en) 2004-09-16
IL158249A (en) 2009-09-01
NO20034526L (no) 2003-10-31
MXPA03009211A (es) 2004-01-29

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