PT1237889E - Oxazolidinonas derivadas de sultama e de sultona como antibioticos - Google Patents

Oxazolidinonas derivadas de sultama e de sultona como antibioticos

Info

Publication number
PT1237889E
PT1237889E PT00973660T PT00973660T PT1237889E PT 1237889 E PT1237889 E PT 1237889E PT 00973660 T PT00973660 T PT 00973660T PT 00973660 T PT00973660 T PT 00973660T PT 1237889 E PT1237889 E PT 1237889E
Authority
PT
Portugal
Prior art keywords
sultona
sultama
antibiotics
oxazolidinones
derived
Prior art date
Application number
PT00973660T
Other languages
English (en)
Inventor
David John Anderson
Jackson B Hester Jr
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of PT1237889E publication Critical patent/PT1237889E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/4211,3-Oxazoles, e.g. pemoline, trimethadione
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT00973660T 1999-11-04 2000-10-30 Oxazolidinonas derivadas de sultama e de sultona como antibioticos PT1237889E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16353799P 1999-11-04 1999-11-04
PCT/US2000/028864 WO2001032657A1 (en) 1999-11-04 2000-10-30 Antibiotic sultam and sultone derived oxazolidinones

Publications (1)

Publication Number Publication Date
PT1237889E true PT1237889E (pt) 2004-12-31

Family

ID=22590470

Family Applications (1)

Application Number Title Priority Date Filing Date
PT00973660T PT1237889E (pt) 1999-11-04 2000-10-30 Oxazolidinonas derivadas de sultama e de sultona como antibioticos

Country Status (19)

Country Link
US (2) US6348459B1 (pt)
EP (1) EP1237889B1 (pt)
JP (1) JP2003513096A (pt)
KR (1) KR20020047328A (pt)
CN (1) CN1146564C (pt)
AR (1) AR029405A1 (pt)
AT (1) ATE275147T1 (pt)
AU (1) AU771655B2 (pt)
BR (1) BR0014303A (pt)
CA (1) CA2383992A1 (pt)
CO (1) CO5261568A1 (pt)
DE (1) DE60013481T2 (pt)
ES (1) ES2226937T3 (pt)
HK (1) HK1049833B (pt)
MY (1) MY120189A (pt)
PE (1) PE20011007A1 (pt)
PT (1) PT1237889E (pt)
WO (1) WO2001032657A1 (pt)
ZA (1) ZA200202605B (pt)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3506435A1 (de) 1985-02-23 1986-08-28 Hoechst Ag, 6230 Frankfurt Neue ketosultame und verfahren zu ihrer herstellung
NZ315469A (en) * 1995-09-01 2000-01-28 Upjohn Co Phenyloxazolidinones having a c-c bond to 4-8 membered heterocyclic rings
GB9702213D0 (en) * 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
WO1998054161A1 (en) * 1997-05-30 1998-12-03 Pharmacia & Upjohn Company Oxazolidinone antibacterial agents having a thiocarbonyl functionality
GB9717807D0 (en) * 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
US6083967A (en) * 1997-12-05 2000-07-04 Pharmacia & Upjohn Company S-oxide and S,S-dioxide tetrahydrothiopyran phenyloxazolidinones

Also Published As

Publication number Publication date
AR029405A1 (es) 2003-06-25
JP2003513096A (ja) 2003-04-08
ATE275147T1 (de) 2004-09-15
EP1237889B1 (en) 2004-09-01
KR20020047328A (ko) 2002-06-21
US6420360B1 (en) 2002-07-16
HK1049833B (zh) 2005-02-18
AU1214901A (en) 2001-05-14
CO5261568A1 (es) 2003-03-31
CN1378546A (zh) 2002-11-06
DE60013481T2 (de) 2005-09-01
CN1146564C (zh) 2004-04-21
EP1237889A1 (en) 2002-09-11
PE20011007A1 (es) 2001-09-14
MY120189A (en) 2005-09-30
CA2383992A1 (en) 2001-05-10
US20020055505A1 (en) 2002-05-09
DE60013481D1 (de) 2004-10-07
US6348459B1 (en) 2002-02-19
ES2226937T3 (es) 2005-04-01
BR0014303A (pt) 2002-05-21
AU771655B2 (en) 2004-04-01
HK1049833A1 (en) 2003-05-30
WO2001032657A1 (en) 2001-05-10
ZA200202605B (en) 2003-07-03

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