PL366021A1 - Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same - Google Patents

Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same

Info

Publication number
PL366021A1
PL366021A1 PL00366021A PL36602100A PL366021A1 PL 366021 A1 PL366021 A1 PL 366021A1 PL 00366021 A PL00366021 A PL 00366021A PL 36602100 A PL36602100 A PL 36602100A PL 366021 A1 PL366021 A1 PL 366021A1
Authority
PL
Poland
Prior art keywords
clarithromycin
processes
pharmaceutical composition
same
free
Prior art date
Application number
PL00366021A
Other languages
English (en)
Polish (pl)
Inventor
Ilya Avrutov
Igor Lifshitz
Elizabeth Lewiner
Original Assignee
Teva Pharmaceutical Industries Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharmaceutical Industries Ltd. filed Critical Teva Pharmaceutical Industries Ltd.
Publication of PL366021A1 publication Critical patent/PL366021A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C07F7/1872—Preparation; Treatments not provided for in C07F7/20
    • C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biochemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL00366021A 2000-02-29 2000-12-15 Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same PL366021A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18588800P 2000-02-29 2000-02-29
US18912000P 2000-03-14 2000-03-14
US21323900P 2000-06-22 2000-06-22

Publications (1)

Publication Number Publication Date
PL366021A1 true PL366021A1 (en) 2005-01-24

Family

ID=27392028

Family Applications (1)

Application Number Title Priority Date Filing Date
PL00366021A PL366021A1 (en) 2000-02-29 2000-12-15 Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same

Country Status (15)

Country Link
US (3) US6617436B2 (enExample)
EP (1) EP1313486A1 (enExample)
JP (1) JP2004509062A (enExample)
KR (1) KR20030047873A (enExample)
AU (2) AU2001225787C1 (enExample)
CA (1) CA2401571A1 (enExample)
CZ (1) CZ20023167A3 (enExample)
HR (1) HRP20020709A2 (enExample)
HU (1) HUP0302466A2 (enExample)
IL (1) IL151496A0 (enExample)
IS (1) IS6531A (enExample)
PL (1) PL366021A1 (enExample)
SK (1) SK13722002A3 (enExample)
WO (1) WO2001064224A1 (enExample)
YU (1) YU64202A (enExample)

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CN102417532A (zh) * 2011-12-20 2012-04-18 浙江国邦药业有限公司 一种泰利霉素关键中间体5-德胺糖基-6-o-甲基红霉素的合成方法
CN102718821B (zh) * 2012-06-27 2014-12-03 浙江国邦药业有限公司 一种克拉霉素合成过程中甲基化反应以及甲基化试剂的回收套用方法
CN103880901A (zh) * 2012-12-23 2014-06-25 菏泽市方明制药有限公司 一种克拉霉素中间甲化物的制备方法
CN106905204B (zh) * 2017-02-24 2018-07-20 杭州新桂实业有限公司 一种克拉霉素合成过程中甲基化反应溶剂的回收套用方法
CN108117573A (zh) * 2017-12-26 2018-06-05 宁夏启元药业有限公司 4"-o-（三甲基硅）红霉素a 9-o-（1-乙氧基-1-甲基乙基）肟的合成方法

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Also Published As

Publication number Publication date
HUP0302466A2 (hu) 2003-11-28
SK13722002A3 (sk) 2003-08-05
JP2004509062A (ja) 2004-03-25
CA2401571A1 (en) 2001-09-07
AU2001225787C1 (en) 2006-09-21
AU2001225787B2 (en) 2005-12-08
US20060205683A1 (en) 2006-09-14
AU2578701A (en) 2001-09-12
EP1313486A1 (en) 2003-05-28
IL151496A0 (en) 2003-04-10
CZ20023167A3 (cs) 2003-10-15
US20030216556A1 (en) 2003-11-20
US6617436B2 (en) 2003-09-09
US20010037015A1 (en) 2001-11-01
IS6531A (is) 2002-08-28
KR20030047873A (ko) 2003-06-18
HRP20020709A2 (en) 2004-12-31
YU64202A (sh) 2005-03-15
US7101858B2 (en) 2006-09-05
WO2001064224A1 (en) 2001-09-07

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