IS6531A - Aðferðir til að búa til klaríþrómýsín og klaríþrómýsínmilliefni, í megindráttum oxímlaust klaríþrómýsín og lyfjablanda sem inniheldur það - Google Patents

Aðferðir til að búa til klaríþrómýsín og klaríþrómýsínmilliefni, í megindráttum oxímlaust klaríþrómýsín og lyfjablanda sem inniheldur það

Info

Publication number
IS6531A
IS6531A IS6531A IS6531A IS6531A IS 6531 A IS6531 A IS 6531A IS 6531 A IS6531 A IS 6531A IS 6531 A IS6531 A IS 6531A IS 6531 A IS6531 A IS 6531A
Authority
IS
Iceland
Prior art keywords
clariodorphysin
oxymorphic
clariforomycin
intermediates
essentially
Prior art date
Application number
IS6531A
Other languages
English (en)
Inventor
Avrutov Ilya
Lifshitz Igor
Lewiner Elizabeth
Original Assignee
Teva Pharmaceutical Industries Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharmaceutical Industries Ltd. filed Critical Teva Pharmaceutical Industries Ltd.
Publication of IS6531A publication Critical patent/IS6531A/is

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C07F7/1872—Preparation; Treatments not provided for in C07F7/20
    • C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IS6531A 2000-02-29 2002-08-28 Aðferðir til að búa til klaríþrómýsín og klaríþrómýsínmilliefni, í megindráttum oxímlaust klaríþrómýsín og lyfjablanda sem inniheldur það IS6531A (is)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US18588800P 2000-02-29 2000-02-29
US18912000P 2000-03-14 2000-03-14
US21323900P 2000-06-22 2000-06-22
PCT/US2000/033843 WO2001064224A1 (en) 2000-02-29 2000-12-15 Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same

Publications (1)

Publication Number Publication Date
IS6531A true IS6531A (is) 2002-08-28

Family

ID=27392028

Family Applications (1)

Application Number Title Priority Date Filing Date
IS6531A IS6531A (is) 2000-02-29 2002-08-28 Aðferðir til að búa til klaríþrómýsín og klaríþrómýsínmilliefni, í megindráttum oxímlaust klaríþrómýsín og lyfjablanda sem inniheldur það

Country Status (15)

Country Link
US (3) US6617436B2 (is)
EP (1) EP1313486A1 (is)
JP (1) JP2004509062A (is)
KR (1) KR20030047873A (is)
AU (2) AU2578701A (is)
CA (1) CA2401571A1 (is)
CZ (1) CZ20023167A3 (is)
HR (1) HRP20020709A2 (is)
HU (1) HUP0302466A2 (is)
IL (1) IL151496A0 (is)
IS (1) IS6531A (is)
PL (1) PL366021A1 (is)
SK (1) SK13722002A3 (is)
WO (1) WO2001064224A1 (is)
YU (1) YU64202A (is)

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CN102417532A (zh) * 2011-12-20 2012-04-18 浙江国邦药业有限公司 一种泰利霉素关键中间体5-德胺糖基-6-o-甲基红霉素的合成方法
CN102718821B (zh) * 2012-06-27 2014-12-03 浙江国邦药业有限公司 一种克拉霉素合成过程中甲基化反应以及甲基化试剂的回收套用方法
CN103880901A (zh) * 2012-12-23 2014-06-25 菏泽市方明制药有限公司 一种克拉霉素中间甲化物的制备方法
CN106905204B (zh) * 2017-02-24 2018-07-20 杭州新桂实业有限公司 一种克拉霉素合成过程中甲基化反应溶剂的回收套用方法
CN108117573A (zh) * 2017-12-26 2018-06-05 宁夏启元药业有限公司 4"-o-（三甲基硅）红霉素a 9-o-（1-乙氧基-1-甲基乙基）肟的合成方法

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Also Published As

Publication number Publication date
KR20030047873A (ko) 2003-06-18
EP1313486A1 (en) 2003-05-28
YU64202A (sh) 2005-03-15
SK13722002A3 (sk) 2003-08-05
PL366021A1 (en) 2005-01-24
US20060205683A1 (en) 2006-09-14
US6617436B2 (en) 2003-09-09
CZ20023167A3 (cs) 2003-10-15
AU2001225787C1 (en) 2006-09-21
CA2401571A1 (en) 2001-09-07
WO2001064224A1 (en) 2001-09-07
US7101858B2 (en) 2006-09-05
AU2578701A (en) 2001-09-12
US20010037015A1 (en) 2001-11-01
JP2004509062A (ja) 2004-03-25
IL151496A0 (en) 2003-04-10
US20030216556A1 (en) 2003-11-20
HRP20020709A2 (en) 2004-12-31
HUP0302466A2 (hu) 2003-11-28
AU2001225787B2 (en) 2005-12-08

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