PL363679A1 - Nowe zastosowanie 2-fenylo-podstawionych imidazotriazynonów - Google Patents

Nowe zastosowanie 2-fenylo-podstawionych imidazotriazynonów

Info

Publication number
PL363679A1
PL363679A1 PL02363679A PL36367902A PL363679A1 PL 363679 A1 PL363679 A1 PL 363679A1 PL 02363679 A PL02363679 A PL 02363679A PL 36367902 A PL36367902 A PL 36367902A PL 363679 A1 PL363679 A1 PL 363679A1
Authority
PL
Poland
Prior art keywords
power
phenyl
novel use
substituted imidazotriazinones
perception
Prior art date
Application number
PL02363679A
Other languages
English (en)
Inventor
Ulrich Niewohner
Erwin Bischoff
Helmut Haning
Afssaneh Rahbar
Tiemo-Joerg Bandel
Wolfgang Barth
Der Staay Franz-Josef Van
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10126198A external-priority patent/DE10126198A1/de
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of PL363679A1 publication Critical patent/PL363679A1/pl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Organic Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PL02363679A 2001-05-09 2002-05-07 Nowe zastosowanie 2-fenylo-podstawionych imidazotriazynonów PL363679A1 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10122576 2001-05-09
DE10126198A DE10126198A1 (de) 2001-05-09 2001-05-30 Neue Verwendung von 2-Phenyl-substituierten Imidazotriazinonen
PCT/EP2002/005002 WO2002089808A1 (de) 2001-05-09 2002-05-07 Neue verwendung von 2-phenyl-substituierten imidazotriazinonen

Publications (1)

Publication Number Publication Date
PL363679A1 true PL363679A1 (pl) 2004-11-29

Family

ID=26009261

Family Applications (1)

Application Number Title Priority Date Filing Date
PL02363679A PL363679A1 (pl) 2001-05-09 2002-05-07 Nowe zastosowanie 2-fenylo-podstawionych imidazotriazynonów

Country Status (15)

Country Link
US (1) US20040152700A1 (pl)
EP (1) EP1392314B1 (pl)
JP (1) JP4540295B2 (pl)
CN (1) CN1633298A (pl)
AT (1) ATE348618T1 (pl)
AU (1) AU2002314044B2 (pl)
BR (1) BR0209541A (pl)
CA (1) CA2449163C (pl)
DE (1) DE50209015D1 (pl)
DK (1) DK1392314T3 (pl)
ES (1) ES2278927T3 (pl)
IL (1) IL158738A0 (pl)
MX (1) MXPA03010119A (pl)
PL (1) PL363679A1 (pl)
WO (1) WO2002089808A1 (pl)

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US6362178B1 (en) * 1997-11-12 2002-03-26 Bayer Aktiengesellschaft 2-phenyl substituted imidazotriazinones as phosphodiesterase inhibitors
DE10135815A1 (de) * 2001-07-23 2003-02-06 Bayer Ag Verwendung von 2-Alkoxyphenyl-substituierten Imidazotriazinonen
DE10232113A1 (de) * 2002-07-16 2004-01-29 Bayer Ag Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel
CA2557792C (en) 2004-03-05 2012-12-18 Altana Pharma Ag Novel use for pde5 inhibitors
DE102004023069A1 (de) 2004-05-11 2005-12-08 Bayer Healthcare Ag Neue Darreichungsformen des PDE 5-Inhibitors Vardenafil
DE102004038328A1 (de) * 2004-08-06 2006-03-16 Bayer Healthcare Ag Neue Verwendungen von 2-Phenyl-substituierten Imidazotriazinon-Derivaten
DE102005001989A1 (de) * 2005-01-15 2006-07-20 Bayer Healthcare Ag Intravenöse Formulierungen von PDE-Inhibitoren
DE102005009241A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit kontrollierter Bioverfügbarkeit
DE102005009240A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften
US20090186896A1 (en) * 2005-09-29 2009-07-23 Bayer Healthcare Ag PDE Inhibitors and Combinations Thereof for the Treatment of Urological Disorders
US8841300B2 (en) 2006-10-02 2014-09-23 Jerry M. Held Treatment for Parkinson's disease—combination high dose serotonergic synaptic reuptake inhibitor with phosphodiesterase inhibitor
CA2687679A1 (en) * 2007-05-18 2008-11-27 Vivus, Inc. Novel compositions comprising a phosphodiesterase-5 inhibitor and their use in methods of treatment
EP2167057A1 (en) * 2007-06-13 2010-03-31 Bayer HealthCare AG Pde inhibitors for the treatment of hearing impairment
WO2009030095A1 (fr) * 2007-09-06 2009-03-12 Topharman Shanghai Co., Ltd. Procédé de préparation de vardénafil et de ses intermédiaires
US9750743B2 (en) * 2012-12-04 2017-09-05 Aribio Inc. Composition comprising phosphodiesterase type 5 inhibitor for inhibiting apoptosis of nerve cells
WO2020109354A1 (en) 2018-11-28 2020-06-04 Topadur Pharma Ag Novel dual mode of action soluble guanylate cyclase activators and phosphodiesterase inhibitors and uses thereof
CN113493459B (zh) * 2020-04-07 2022-12-13 广州白云山医药集团股份有限公司白云山制药总厂 Pde5抑制剂化合物及其制备方法和应用

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DE102004023069A1 (de) * 2004-05-11 2005-12-08 Bayer Healthcare Ag Neue Darreichungsformen des PDE 5-Inhibitors Vardenafil

Also Published As

Publication number Publication date
EP1392314B1 (de) 2006-12-20
JP4540295B2 (ja) 2010-09-08
CA2449163C (en) 2010-07-13
EP1392314A1 (de) 2004-03-03
WO2002089808A1 (de) 2002-11-14
AU2002314044B2 (en) 2006-09-21
IL158738A0 (en) 2004-05-12
CN1633298A (zh) 2005-06-29
ES2278927T3 (es) 2007-08-16
DE50209015D1 (de) 2007-02-01
DK1392314T3 (da) 2007-03-12
US20040152700A1 (en) 2004-08-05
JP2004528363A (ja) 2004-09-16
BR0209541A (pt) 2004-04-20
MXPA03010119A (es) 2005-03-07
ATE348618T1 (de) 2007-01-15
CA2449163A1 (en) 2002-11-14

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Legal Events

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