PL1877403T3 - Sole mono-lizynowe związków azolowych - Google Patents

Sole mono-lizynowe związków azolowych

Info

Publication number
PL1877403T3
PL1877403T3 PL06746245T PL06746245T PL1877403T3 PL 1877403 T3 PL1877403 T3 PL 1877403T3 PL 06746245 T PL06746245 T PL 06746245T PL 06746245 T PL06746245 T PL 06746245T PL 1877403 T3 PL1877403 T3 PL 1877403T3
Authority
PL
Poland
Prior art keywords
mono
azole compounds
lysine salts
lysine
salts
Prior art date
Application number
PL06746245T
Other languages
English (en)
Inventor
Qi Gao
Chung-Pin H Chen
Michael G Fakes
Yadagiri R Pendri
Susanne Kiau
Blisse Vakkalagadda
Original Assignee
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd
Publication of PL1877403T3 publication Critical patent/PL1877403T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/26Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having more than one amino group bound to the carbon skeleton, e.g. lysine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65586Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PL06746245T 2005-05-03 2006-05-01 Sole mono-lizynowe związków azolowych PL1877403T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67693205P 2005-05-03 2005-05-03
EP06746245A EP1877403B1 (en) 2005-05-03 2006-05-01 Mono-lysine salts of azole compounds
PCT/JP2006/309435 WO2006118351A1 (en) 2005-05-03 2006-05-01 Mono-lysine salts of azole compounds

Publications (1)

Publication Number Publication Date
PL1877403T3 true PL1877403T3 (pl) 2011-08-31

Family

ID=36910951

Family Applications (1)

Application Number Title Priority Date Filing Date
PL06746245T PL1877403T3 (pl) 2005-05-03 2006-05-01 Sole mono-lizynowe związków azolowych

Country Status (34)

Country Link
US (1) US20060264406A1 (pl)
EP (1) EP1877403B1 (pl)
JP (1) JP4015691B1 (pl)
KR (1) KR100887044B1 (pl)
CN (1) CN101213193B (pl)
AR (1) AR053862A1 (pl)
AT (1) ATE503753T1 (pl)
AU (1) AU2006241694B2 (pl)
BR (1) BRPI0610423B8 (pl)
CA (1) CA2606185C (pl)
CY (1) CY1111569T1 (pl)
DE (1) DE602006020998D1 (pl)
DK (1) DK1877403T3 (pl)
EC (1) ECSP077812A (pl)
ES (1) ES2361768T3 (pl)
HK (1) HK1117502A1 (pl)
HR (1) HRP20110467T1 (pl)
IL (1) IL187059A (pl)
JO (1) JO2691B1 (pl)
MX (1) MX2007013605A (pl)
MY (1) MY138095A (pl)
NO (1) NO20075541L (pl)
NZ (1) NZ563092A (pl)
PE (1) PE20071423A1 (pl)
PL (1) PL1877403T3 (pl)
PT (1) PT1877403E (pl)
RS (1) RS51779B (pl)
RU (1) RU2399625C2 (pl)
SA (1) SA06270126B1 (pl)
SI (1) SI1877403T1 (pl)
TW (1) TWI363630B (pl)
UY (1) UY29507A1 (pl)
WO (1) WO2006118351A1 (pl)
ZA (1) ZA200709127B (pl)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2632842C (en) 2005-12-20 2013-06-25 Eisai R & D Management Co., Ltd. Process for preparation of water-soluble azole prodrugs
CN101389333A (zh) 2006-02-22 2009-03-18 卫材R&D管理有限公司 稳定化药物组合物
CN105287403A (zh) * 2014-08-02 2016-02-03 陕西合成药业股份有限公司 一种泊沙康唑前体药物的冻干组合物及其制备方法和用途
CN106432338A (zh) * 2015-08-08 2017-02-22 陕西合成药业股份有限公司 泊沙康唑衍生物、合成和在长效制剂中的用途
WO2019106571A1 (en) 2017-11-28 2019-06-06 Roivant Sciences Gmbh Dosing regimens for the treatment of fungal infections
CN110938093B (zh) * 2018-09-21 2022-08-19 华创合成制药股份有限公司 一种泊沙康唑磷酸酯单胆碱盐及其制备方法和用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI0741737T1 (en) * 1994-01-24 2000-02-29 Janssen Pharmaceutica N.V. Watersoluble azole antifungals
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
US5883097A (en) * 1998-04-16 1999-03-16 Schering Corporation Soluble azole antifungal salt
US6265584B1 (en) * 1998-05-22 2001-07-24 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
WO2000030655A1 (en) * 1998-11-20 2000-06-02 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
US6235728B1 (en) * 1999-02-19 2001-05-22 Bristol-Myers Squibb Company Water-soluble prodrugs of azole compounds
US6362172B2 (en) * 2000-01-20 2002-03-26 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
US6448401B1 (en) * 2000-11-20 2002-09-10 Bristol-Myers Squibb Company Process for water soluble azole compounds

Also Published As

Publication number Publication date
RU2007140788A (ru) 2009-06-10
BRPI0610423B1 (pt) 2020-11-10
MX2007013605A (es) 2008-01-24
NO20075541L (no) 2007-11-28
HRP20110467T1 (hr) 2011-07-31
DK1877403T3 (da) 2011-05-09
BRPI0610423B8 (pt) 2021-05-25
HK1117502A1 (en) 2009-01-16
RS51779B (en) 2011-12-31
AU2006241694A1 (en) 2006-11-09
TWI363630B (en) 2012-05-11
JP4015691B1 (ja) 2007-11-28
EP1877403A1 (en) 2008-01-16
NZ563092A (en) 2010-06-25
IL187059A (en) 2012-08-30
TW200722093A (en) 2007-06-16
BRPI0610423A2 (pt) 2010-06-22
ECSP077812A (es) 2008-01-23
SA06270126B1 (ar) 2009-09-02
JO2691B1 (en) 2013-03-03
AU2006241694B2 (en) 2011-10-20
CN101213193B (zh) 2011-02-02
KR100887044B1 (ko) 2009-03-04
SI1877403T1 (sl) 2011-05-31
PT1877403E (pt) 2011-05-31
MY138095A (en) 2009-04-30
KR20070088460A (ko) 2007-08-29
AR053862A1 (es) 2007-05-23
WO2006118351A1 (en) 2006-11-09
ZA200709127B (en) 2008-07-30
US20060264406A1 (en) 2006-11-23
PE20071423A1 (es) 2006-12-17
IL187059A0 (en) 2008-02-09
ES2361768T3 (es) 2011-06-22
CA2606185A1 (en) 2006-11-09
CA2606185C (en) 2012-08-28
JP2008544948A (ja) 2008-12-11
RU2399625C2 (ru) 2010-09-20
EP1877403B1 (en) 2011-03-30
CN101213193A (zh) 2008-07-02
CY1111569T1 (el) 2015-10-07
DE602006020998D1 (de) 2011-05-12
UY29507A1 (es) 2006-11-30
ATE503753T1 (de) 2011-04-15

Similar Documents

Publication Publication Date Title
HUS1900033I1 (hu) Szubsztituált enaminokarbonil vegyületek
ZA200904108B (en) Pyrido-pyrazine derivatives useful as herbicidal compounds
SI1919907T1 (sl) Heterocikliäśna spojina
ZA200709051B (en) Heterocyclic compound
ZA200709994B (en) Neurotherapeutic Azole Compounds
AP2008004580A0 (en) Herbicidal isoyazoline compounds
GB0614471D0 (en) Herbicidal Compounds
IL190450A0 (en) Substituted pyrazole compounds
HK1133641A1 (zh) 激酶抑製劑化合物
EP1953151A4 (en) SALTS FROM A CYNNAMIDE COMPOUND OR SOLVATE THEREOF
HK1123038A1 (en) Heterocyclic compounds
IL195158A0 (en) Novel heterocyclic compounds
ZA200803636B (en) Triazole compounds as lipoxygenase inhibitors
IL187279A0 (en) Hydantoin compounds
PL1870409T3 (pl) Związki benzimidazolowe
HK1117502A1 (en) Mono-lysine salts of azole compounds
ZA200800142B (en) Heterocyclic compound
ZA200802786B (en) Substituted pyrazole compounds
ZA200803017B (en) Heterocyclic compounds
EP2042499A4 (en) SALTS OF MORPHOLINE COMPOUND
ZA200901570B (en) Substituted azolin-2-YL-amino compounds
GB0619308D0 (en) Heterocyclic compounds
EP1940411A4 (en) MACROHETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS
GB0512626D0 (en) Inhibitor compounds
GB0517677D0 (en) Inhibitor compounds II