PH23813A - Pyridazodiazepine derivatives - Google Patents
Pyridazodiazepine derivativesInfo
- Publication number
- PH23813A PH23813A PH36217A PH36217A PH23813A PH 23813 A PH23813 A PH 23813A PH 36217 A PH36217 A PH 36217A PH 36217 A PH36217 A PH 36217A PH 23813 A PH23813 A PH 23813A
- Authority
- PH
- Philippines
- Prior art keywords
- pyridazodiazepine
- derivatives
- pyridazodiazepine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Pharmacology & Pharmacy (AREA)
- Cardiology (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB868629875A GB8629875D0 (en) | 1986-12-15 | 1986-12-15 | Pyridazodiazepine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
PH23813A true PH23813A (en) | 1989-11-23 |
Family
ID=10609005
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PH36217A PH23813A (en) | 1986-12-15 | 1987-12-14 | Pyridazodiazepine derivatives |
Country Status (17)
Country | Link |
---|---|
US (2) | US4757069A (fi) |
EP (1) | EP0271795A3 (fi) |
JP (1) | JPS63162693A (fi) |
KR (1) | KR880007538A (fi) |
AU (1) | AU602546B2 (fi) |
CA (1) | CA1291478C (fi) |
DK (1) | DK628087A (fi) |
FI (1) | FI85482C (fi) |
GB (1) | GB8629875D0 (fi) |
HU (1) | HU198492B (fi) |
IL (1) | IL84765A (fi) |
MC (1) | MC1879A1 (fi) |
NO (1) | NO166083C (fi) |
NZ (1) | NZ222825A (fi) |
PH (1) | PH23813A (fi) |
PT (1) | PT86365B (fi) |
ZA (1) | ZA879229B (fi) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5430145A (en) * | 1990-10-18 | 1995-07-04 | Merrell Dow Pharmaceuticals Inc. | Mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace |
US5308841A (en) * | 1990-12-21 | 1994-05-03 | Merrell Dow Pharmaceuticals Inc. | Amino and nitro containing tricyclic compounds useful as inhibitors of ACE |
US5455242A (en) * | 1991-09-27 | 1995-10-03 | Merrell Dow Pharmaceuticals Inc. | Carboxyalkyl tricyclic derivatives useful as inhibitors of enkephalinase and ace |
DK0534363T3 (da) * | 1991-09-27 | 1997-09-22 | Merrell Pharma Inc | 2-substituerede indan-2-mercaptoacetylamid-forbindelse med inhiberende virkning på enkephalinase og ACE. |
US5457196A (en) * | 1991-09-27 | 1995-10-10 | Merrell Dow Pharmaceuticals Inc. | 2-substituted indane-2-carboxyalkyl derivatives useful as inhibitors of enkephalinase and ACE |
CA2130116C (en) * | 1992-02-14 | 1998-04-07 | Gary A. Flynn | Aminoacetylmercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace |
ATE182892T1 (de) * | 1992-05-15 | 1999-08-15 | Merrell Pharma Inc | Mercaptoacetylamide von pyridazo(1,2-a>(1,2>- diazepin -derivaten als eukephalinase und ace- inhibitoren |
US5420271A (en) * | 1992-08-24 | 1995-05-30 | Merrell Dow Pharmaceuticals, Inc. | 2-substituted indane-2-mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase |
CA2146238C (en) * | 1992-10-30 | 2001-03-13 | Gary A. Flynn | Novel mercaptoacetylamide bicyclic lactam derivatives useful as inhibitors of enkephalinase and ace |
CN1142831A (zh) * | 1994-02-14 | 1997-02-12 | 默里尔药物公司 | 用作脑啡肽酶和ace抑制剂的新的2-取代的1,2-二氢化茚-2-巯基乙酰胺二硫化物衍生物 |
ATE177098T1 (de) * | 1994-02-14 | 1999-03-15 | Merrell Pharma Inc | Mercaptoacetylamid disulfidderivate als enkephalinase und ace inhibitoren |
WO1995021840A1 (en) * | 1994-02-14 | 1995-08-17 | Merrell Pharmaceuticals Inc. | Novel indane-2-mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase |
US5530013A (en) * | 1994-02-14 | 1996-06-25 | American Home Products Corporation | Venlafaxine in the inducement of cognition enhancement |
PT750631E (pt) * | 1994-02-14 | 2000-07-31 | Merrell Pharma Inc | Novos derivados de dissulfureto de mercapto-aacetilamido-1,3,4,5-tetra-hidro-benzo¬c)azepin-3-ona uteis como inibidores de encefalinase e ace |
US5484783A (en) * | 1994-03-24 | 1996-01-16 | Merrell Dow Pharmaceuticals Inc. | Hypocholesterolemic, antiatherosclerotic and hypotriglyceridemic mercaptoacetylamide and benzazapine derivatives |
JPH10503468A (ja) * | 1994-03-24 | 1998-03-31 | メリル・フアーマシユウテイカルズ・インコーポレイテツド | 低コレステロール血性、抗アテローム性動脈硬化性および低トリグリセライド血性のメルカプトアセチルアミドジスルフィド誘導体 |
DE69514912T2 (de) * | 1994-03-24 | 2000-10-05 | Merrell Pharmaceuticals Inc., Cincinnati | Hypocholesterolemische, antiatherosklerotische und hypotriglyceridemische verwendung von aminoacetylmercapto derivaten |
WO2001060879A1 (fr) * | 2000-02-17 | 2001-08-23 | China Petroleum & Chemical Corporation | Copolymere multisequence et son procede de preparation |
GB0119305D0 (en) | 2001-04-12 | 2001-10-03 | Aventis Pharma Gmbh | Mercaptoacetylamide derivatives,a process for their preparation and their use |
IE20070935A1 (en) * | 2007-12-21 | 2009-06-24 | Trinity College Dublin | Guanidine based compounds and their use in the treatment of mental and neurological disorders. |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4092438A (en) * | 1977-04-29 | 1978-05-30 | Carnation Company | Non-dairy coffee whitener containing acetate salt |
GB2128984B (en) * | 1982-05-12 | 1985-05-22 | Hoffmann La Roche | Diaza-bicyclic compounds |
GB8320764D0 (en) * | 1983-08-02 | 1983-09-01 | Rhodes Joseph Ltd | Bending machines |
US4692438A (en) * | 1984-08-24 | 1987-09-08 | Hoffmann-La Roche Inc. | Pyridazo-diazepines, diazocines, and -triazepines having anti-hypertensive activity |
EP0187037A3 (en) * | 1984-12-21 | 1988-03-23 | Takeda Chemical Industries, Ltd. | Piperidine derivatives, their production and use |
-
1986
- 1986-12-15 GB GB868629875A patent/GB8629875D0/en active Pending
-
1987
- 1987-11-24 US US07/124,749 patent/US4757069A/en not_active Expired - Fee Related
- 1987-11-30 DK DK628087A patent/DK628087A/da not_active Application Discontinuation
- 1987-12-07 EP EP87118047A patent/EP0271795A3/de not_active Ceased
- 1987-12-07 NZ NZ222825A patent/NZ222825A/en unknown
- 1987-12-08 ZA ZA879229A patent/ZA879229B/xx unknown
- 1987-12-08 CA CA000553720A patent/CA1291478C/en not_active Expired - Fee Related
- 1987-12-09 AU AU82254/87A patent/AU602546B2/en not_active Ceased
- 1987-12-09 IL IL84765A patent/IL84765A/xx unknown
- 1987-12-10 MC MC871934A patent/MC1879A1/xx unknown
- 1987-12-11 HU HU875592A patent/HU198492B/hu unknown
- 1987-12-14 KR KR870014258A patent/KR880007538A/ko not_active Application Discontinuation
- 1987-12-14 FI FI875483A patent/FI85482C/fi not_active IP Right Cessation
- 1987-12-14 PH PH36217A patent/PH23813A/en unknown
- 1987-12-14 NO NO875200A patent/NO166083C/no unknown
- 1987-12-14 JP JP62314308A patent/JPS63162693A/ja active Pending
- 1987-12-15 PT PT86365A patent/PT86365B/pt not_active IP Right Cessation
-
1988
- 1988-03-17 US US07/169,266 patent/US4782149A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
MC1879A1 (fr) | 1989-01-24 |
US4757069A (en) | 1988-07-12 |
FI875483A (fi) | 1988-06-16 |
IL84765A0 (en) | 1988-05-31 |
AU8225487A (en) | 1988-06-16 |
JPS63162693A (ja) | 1988-07-06 |
ZA879229B (en) | 1988-06-15 |
NO875200L (no) | 1988-06-16 |
NZ222825A (en) | 1990-11-27 |
NO166083B (no) | 1991-02-18 |
DK628087A (da) | 1988-06-16 |
PT86365A (en) | 1988-01-01 |
GB8629875D0 (en) | 1987-01-28 |
FI85482C (fi) | 1992-04-27 |
CA1291478C (en) | 1991-10-29 |
NO166083C (no) | 1991-05-29 |
FI85482B (fi) | 1992-01-15 |
HUT47279A (en) | 1989-02-28 |
DK628087D0 (da) | 1987-11-30 |
AU602546B2 (en) | 1990-10-18 |
PT86365B (pt) | 1990-11-20 |
US4782149A (en) | 1988-11-01 |
EP0271795A2 (de) | 1988-06-22 |
KR880007538A (ko) | 1988-08-27 |
HU198492B (en) | 1989-10-30 |
IL84765A (en) | 1991-06-30 |
FI875483A0 (fi) | 1987-12-14 |
EP0271795A3 (de) | 1989-08-09 |
NO875200D0 (no) | 1987-12-14 |
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