PH22338A - 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines - Google Patents

1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines

Info

Publication number
PH22338A
PH22338A PH31451A PH31451A PH22338A PH 22338 A PH22338 A PH 22338A PH 31451 A PH31451 A PH 31451A PH 31451 A PH31451 A PH 31451A PH 22338 A PH22338 A PH 22338A
Authority
PH
Philippines
Prior art keywords
imidazo
carbon atoms
group
quinolines
quinolin
Prior art date
Application number
PH31451A
Other languages
English (en)
Inventor
John F Gerster
Original Assignee
Riker Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Riker Laboratories Inc filed Critical Riker Laboratories Inc
Publication of PH22338A publication Critical patent/PH22338A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Physical Water Treatments (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Macromonomer-Based Addition Polymer (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Quinoline Compounds (AREA)
  • Alarm Systems (AREA)
  • Luminescent Compositions (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Lubricants (AREA)
PH31451A 1983-11-18 1984-11-16 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines PH22338A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55315883A 1983-11-18 1983-11-18
US55315783A 1983-11-18 1983-11-18

Publications (1)

Publication Number Publication Date
PH22338A true PH22338A (en) 1988-08-12

Family

ID=27070262

Family Applications (1)

Application Number Title Priority Date Filing Date
PH31451A PH22338A (en) 1983-11-18 1984-11-16 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines

Country Status (15)

Country Link
EP (2) EP0145340B1 (de)
JP (1) JPS60123488A (de)
KR (1) KR900005657B1 (de)
AT (2) ATE84525T1 (de)
AU (2) AU581190B2 (de)
CA (1) CA1271477A (de)
DE (3) DE3486043T2 (de)
DK (6) DK164280C (de)
ES (1) ES8603477A1 (de)
IE (1) IE57874B1 (de)
IL (2) IL84537A (de)
NL (2) NL980043I1 (de)
NO (7) NO163819C (de)
NZ (1) NZ210228A (de)
PH (1) PH22338A (de)

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EP0361489A3 (de) * 1988-09-30 1991-06-12 Chugai Seiyaku Kabushiki Kaisha 3,4-Diaminochinolin- und Pyridinverbindungen
EP0385630B1 (de) * 1989-02-27 1996-11-27 Riker Laboratories, Inc. 4-Amino-1H-Imidazo(4,5-c)chinoline als antivirale Mittel
CA2011504C (en) * 1989-03-07 1998-06-02 Kenji Ohmori Imidazoquinolone derivatives
US4929624A (en) * 1989-03-23 1990-05-29 Minnesota Mining And Manufacturing Company Olefinic 1H-imidazo(4,5-c)quinolin-4-amines
CA2021338C (en) * 1989-07-18 1996-07-16 Fumio Suzuki Imidazoquinolone derivatives
US4988815A (en) * 1989-10-26 1991-01-29 Riker Laboratories, Inc. 3-Amino or 3-nitro quinoline compounds which are intermediates in preparing 1H-imidazo[4,5-c]quinolines
FR2654021B1 (fr) * 1989-11-07 1992-02-28 Simond Jacques Procede de vitrification de cendres volantes et dispositif pour sa mise en óoeuvre.
GB8928281D0 (en) * 1989-12-14 1990-02-21 Smith Kline French Lab Compounds
ES2094772T3 (es) * 1990-06-01 1997-02-01 Kyowa Hakko Kogyo Kk Derivados de imidazonaftiridinas.
DE69229114T2 (de) * 1991-03-01 1999-11-04 Minnesota Mining And Mfg. Co., Saint Paul 1,2-substituierte 1h-imidazo[4,5-c]chinolin-4-amine
US5266575A (en) * 1991-11-06 1993-11-30 Minnesota Mining And Manufacturing Company 2-ethyl 1H-imidazo[4,5-ciquinolin-4-amines
IL105325A (en) * 1992-04-16 1996-11-14 Minnesota Mining & Mfg Immunogen/vaccine adjuvant composition
US5395937A (en) * 1993-01-29 1995-03-07 Minnesota Mining And Manufacturing Company Process for preparing quinoline amines
US5693811A (en) * 1996-06-21 1997-12-02 Minnesota Mining And Manufacturing Company Process for preparing tetrahdroimidazoquinolinamines
US6069149A (en) * 1997-01-09 2000-05-30 Terumo Kabushiki Kaisha Amide derivatives and intermediates for the synthesis thereof
JPH10298181A (ja) * 1997-04-25 1998-11-10 Sumitomo Pharmaceut Co Ltd タイプ２ヘルパーｔ細胞選択的免疫応答抑制剤
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WO2003035626A2 (en) * 2001-10-23 2003-05-01 Applied Research Systems Ars Holding N.V. Azole derivatives and pharmaceutical compositions containing them
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SI1539752T1 (sl) 2002-07-26 2007-08-31 Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag Priprava 1H-imidazo(4,5-c)kinolin-4-aminov preko novih imidazo(4,5-c)kinolin-4-ciano in 1H-imidazo(4,5-c)kinolin-4- karboksamidnih intermediatov
WO2005018556A2 (en) 2003-08-12 2005-03-03 3M Innovative Properties Company Hydroxylamine substituted imidazo-containing compounds
ES2406730T3 (es) 2003-08-27 2013-06-07 3M Innovative Properties Company Imidazoquinolinas sustituidas con ariloxi y arilalquilenoxi
AU2004270201A1 (en) 2003-09-05 2005-03-17 3M Innovative Properties Company Treatment for CD5+ B cell lymphoma
CA2536530A1 (en) 2003-10-01 2005-04-14 Taro Pharmaceuticals U.S.A., Inc. Method of preparing 4-amino-1h-imidazo(4,5-c)quinolines and acid addition salts thereof
CA2540541C (en) 2003-10-03 2012-03-27 3M Innovative Properties Company Alkoxy substituted imidazoquinolines
US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
ITMI20032121A1 (it) * 2003-11-04 2005-05-05 Dinamite Dipharma Spa In Forma Abbr Eviata Dipharm Procedimento per la preparazione di imiquimod e suoi intermedi
EP1685129A4 (de) 2003-11-14 2008-10-22 3M Innovative Properties Co Oximsubstituierte imidazoringverbindungen
WO2005048945A2 (en) 2003-11-14 2005-06-02 3M Innovative Properties Company Hydroxylamine substituted imidazo ring compounds
JP4891088B2 (ja) 2003-11-25 2012-03-07 スリーエム イノベイティブ プロパティズ カンパニー 置換されたイミダゾ環系および方法
JP2007517035A (ja) 2003-12-29 2007-06-28 スリーエム イノベイティブ プロパティズ カンパニー アリールアルケニルおよびアリールアルキニル置換されたイミダゾキノリン
CA2551399A1 (en) 2003-12-30 2005-07-21 3M Innovative Properties Company Imidazoquinolinyl, imidazopyridinyl, and imidazonaphthyridinyl sulfonamides
CA2559863A1 (en) 2004-03-24 2005-10-13 3M Innovative Properties Company Amide substituted imidazopyridines, imidazoquinolines, and imidazonaphthyridines
US8017779B2 (en) 2004-06-15 2011-09-13 3M Innovative Properties Company Nitrogen containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
US7915281B2 (en) 2004-06-18 2011-03-29 3M Innovative Properties Company Isoxazole, dihydroisoxazole, and oxadiazole substituted imidazo ring compounds and method
US8026366B2 (en) 2004-06-18 2011-09-27 3M Innovative Properties Company Aryloxy and arylalkyleneoxy substituted thiazoloquinolines and thiazolonaphthyridines
WO2006038923A2 (en) 2004-06-18 2006-04-13 3M Innovative Properties Company Aryl substituted imidazonaphthyridines
AU2005322898B2 (en) 2004-12-30 2011-11-24 3M Innovative Properties Company Chiral fused (1,2)imidazo(4,5-c) ring compounds
AU2005326708C1 (en) 2004-12-30 2012-08-30 3M Innovative Properties Company Substituted chiral fused [1,2]imidazo[4,5-c] ring compounds
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JP2009504803A (ja) 2005-08-22 2009-02-05 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア Ｔｌｒアゴニスト
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EP2009002A1 (de) * 2007-06-21 2008-12-31 Institut National De La Sante Et De La Recherche Medicale (Inserm) Neues Verfahren zur Herstellung von 1H-imidazo [4,5-c]-chinolin-Ringsystemen
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HUE033901T2 (en) * 2010-08-17 2018-01-29 3M Innovative Properties Co Formulations and formulations for lipidized immune response modifying compounds and related processes
US8728486B2 (en) 2011-05-18 2014-05-20 University Of Kansas Toll-like receptor-7 and -8 modulatory 1H imidazoquinoline derived compounds
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CN118515666A (zh) 2017-04-27 2024-08-20 博笛生物科技有限公司 2-氨基-喹啉衍生物
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Also Published As

Publication number Publication date
DK135891A (da) 1991-07-16
JPS60123488A (ja) 1985-07-02
NO890822D0 (no) 1989-02-27
KR900005657B1 (ko) 1990-08-03
NO890825D0 (no) 1989-02-27
DK165921C (da) 1993-06-28
DK135891D0 (da) 1991-07-16
DE3486043D1 (de) 1993-02-25
DK164451C (da) 1992-11-09
DK164280C (da) 1992-11-30
DK164452C (da) 1992-11-09
DK164455C (da) 1992-11-16
DE19975027I2 (de) 2000-09-21
DK135991D0 (da) 1991-07-16
DK169179B1 (da) 1994-09-05
NO890823L (no) 1985-05-20
NO165146C (no) 1991-01-02
ATE84525T1 (de) 1993-01-15
DK136091A (da) 1991-07-16
DK135791D0 (da) 1991-07-16
ES537677A0 (es) 1985-12-16
NL980043I1 (nl) 1999-02-01
NO890824D0 (no) 1989-02-27
NO165146B (no) 1990-09-24
NO890826D0 (no) 1989-02-27
DK135991A (da) 1991-07-16
KR850003890A (ko) 1985-06-29
NO165145B (no) 1990-09-24
DK164451B (da) 1992-06-29
NO890824L (no) 1985-05-20
NO890825L (no) 1985-05-20
EP0145340A3 (en) 1986-06-11
DK164280B (da) 1992-06-01
DK542684D0 (da) 1984-11-15
IL84537A (en) 1990-12-23
IE57874B1 (en) 1993-05-05
CA1271477A (en) 1990-07-10
NO168705B (no) 1991-12-16
DK542684A (da) 1985-05-19
NO169437B (no) 1992-03-16
JPH0586391B2 (de) 1993-12-10
AU611997B2 (en) 1991-06-27
IE842952L (en) 1985-05-18
NO169437C (no) 1992-06-24
ATE49763T1 (de) 1990-02-15
DE3486043T2 (de) 1993-06-03
NL980041I1 (nl) 1999-02-01
AU2991189A (en) 1989-06-15
NO163819C (no) 1990-08-01
ES8603477A1 (es) 1985-12-16
DK165921B (da) 1993-02-08
NO1999015I1 (no) 1999-07-08
NO844565L (no) 1985-05-20
NO890823D0 (no) 1989-02-27
NO168705C (no) 1992-03-25
DK164455B (da) 1992-06-29
NO165147C (no) 1991-01-02
DK136091D0 (da) 1991-07-16
DK164452B (da) 1992-06-29
EP0310950B1 (de) 1993-01-13
NO890822L (no) 1985-05-20
DK135791A (da) 1991-07-16
DK136191D0 (da) 1991-07-16
DK136191A (da) 1991-07-16
IL84537A0 (en) 1988-04-29
DE3481124D1 (de) 1990-03-01
NO890826L (no) 1985-05-20
EP0145340A2 (de) 1985-06-19
NL980041I2 (nl) 1999-07-01
NO163819B (no) 1990-04-17
NO165145C (no) 1991-01-02
EP0145340B1 (de) 1990-01-24
EP0310950A1 (de) 1989-04-12
AU3540284A (en) 1985-05-23
AU581190B2 (en) 1989-02-16
NZ210228A (en) 1989-01-27
NO165147B (no) 1990-09-24

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PH22338A (en) 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines