PH18930A - 2-phenyl-pyrimidones - Google Patents
2-phenyl-pyrimidonesInfo
- Publication number
- PH18930A PH18930A PH26759A PH26759A PH18930A PH 18930 A PH18930 A PH 18930A PH 26759 A PH26759 A PH 26759A PH 26759 A PH26759 A PH 26759A PH 18930 A PH18930 A PH 18930A
- Authority
- PH
- Philippines
- Prior art keywords
- pyrimidones
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/20—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 4
- C07D265/22—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19803046871 DE3046871A1 (de) | 1980-12-12 | 1980-12-12 | Neue chinazolinone, ihre herstellung und ihre verwendung als arzneimittel |
| DE19813115447 DE3115447A1 (de) | 1981-04-16 | 1981-04-16 | Neue pyrimidinone, ihre herstellung und ihre verwendung als arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH18930A true PH18930A (en) | 1985-11-11 |
Family
ID=25789685
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH26759A PH18930A (en) | 1980-12-12 | 1981-12-11 | 2-phenyl-pyrimidones |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US4379788A (es) |
| EP (1) | EP0054132B1 (es) |
| AR (1) | AR227567A1 (es) |
| AU (1) | AU543568B2 (es) |
| CA (1) | CA1217767A (es) |
| CS (1) | CS227024B2 (es) |
| DD (1) | DD208151A5 (es) |
| DE (1) | DE3166627D1 (es) |
| DK (1) | DK525481A (es) |
| ES (2) | ES507761A0 (es) |
| FI (1) | FI813971L (es) |
| GB (1) | GB2090249B (es) |
| GR (1) | GR76952B (es) |
| HU (1) | HU187384B (es) |
| IL (1) | IL64504A (es) |
| MY (1) | MY8700562A (es) |
| NO (1) | NO814239L (es) |
| NZ (1) | NZ199254A (es) |
| PH (1) | PH18930A (es) |
| PL (1) | PL135330B1 (es) |
| PT (1) | PT74116B (es) |
| SU (1) | SU1056900A3 (es) |
Families Citing this family (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4460589A (en) * | 1980-10-03 | 1984-07-17 | The Upjohn Company | Process for treating hypertension |
| US4379778A (en) * | 1980-10-10 | 1983-04-12 | Air Products And Chemicals, Inc. | Hydrogen peroxide synthesis |
| DE3428476A1 (de) * | 1984-08-02 | 1986-02-13 | Basf Ag, 6700 Ludwigshafen | 4h-pyrido(2,3-d)(1,3)oxazin-4-on-derivate, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung unerwuenschten pflanzenwuchses |
| DE3631294A1 (de) * | 1986-09-13 | 1988-03-24 | Thomae Gmbh Dr K | Neue synergistische kombination bestehend aus einem phosphodiesterase-hemmer und einem thromboxan-a(pfeil abwaerts)2(pfeil abwaerts)-antagonisten und deren verwendung bzw. herstellung |
| US5037980A (en) * | 1988-04-18 | 1991-08-06 | American Cyanamid Company | Phenyl imidazo[1,2-a]pyrimidines |
| GB8928346D0 (en) * | 1989-12-15 | 1990-02-21 | Smith Kline French Lab | Chemical compounds |
| GB9126260D0 (en) * | 1991-12-11 | 1992-02-12 | Pfizer Ltd | Therapeutic agents |
| GB9404485D0 (en) * | 1994-03-09 | 1994-04-20 | Cancer Res Campaign Tech | Benzamide analogues |
| CN100430396C (zh) | 1997-11-12 | 2008-11-05 | 拜耳医药保健股份公司 | 用作磷酸二酯酶抑制剂的2-苯基取代的咪唑并三嗪酮 |
| AU2645299A (en) * | 1998-11-18 | 2000-06-05 | Elena Alexandrovna Izaxon | 6-(3-carboxymethylphenyl)-aminouracyl having a biological activity |
| US20040102324A1 (en) | 2002-02-28 | 2004-05-27 | Annis Gary David | Heterocyclic diamide invertebrate pest control agents |
| US6642244B2 (en) | 2001-03-16 | 2003-11-04 | Bristol-Myers Squibb Co. | Pyrazolopyridopyrimidine inhibitors of cGMP phosphodiesterase |
| CN1518447A (zh) * | 2001-04-23 | 2004-08-04 | �������Ǵ�ѧר������� | 作为抗血管生成剂的新的苯邻二甲酰亚胺模拟物的合成和评估 |
| DE50209015D1 (de) * | 2001-05-09 | 2007-02-01 | Bayer Healthcare Ag | NEUE VERWENDUNG VON 2-Ä2-Ethoxy-5-(4-methyl-piperazin-1-sulfonyl)-phenylÜ-5-methyl-7-propyl-3H-imidazoÄ5,1-fÜÄ1,2,4Ütriazin-4-on |
| DE10232113A1 (de) * | 2002-07-16 | 2004-01-29 | Bayer Ag | Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel |
| EP1696927A4 (en) * | 2003-12-19 | 2007-10-31 | Merck & Co Inc | MITOTIC INHIBITORS OF KINESIN |
| SE0401342D0 (sv) * | 2004-05-25 | 2004-05-25 | Astrazeneca Ab | Therapeutic compounds |
| SE0401345D0 (sv) * | 2004-05-25 | 2004-05-25 | Astrazeneca Ab | Therapeutic compounds: Pyridine as scaffold |
| JPWO2005115993A1 (ja) * | 2004-05-31 | 2008-03-27 | 萬有製薬株式会社 | キナゾリン誘導体 |
| DE102005001989A1 (de) * | 2005-01-15 | 2006-07-20 | Bayer Healthcare Ag | Intravenöse Formulierungen von PDE-Inhibitoren |
| DE102005009241A1 (de) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit kontrollierter Bioverfügbarkeit |
| DE102005009240A1 (de) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften |
| EP1931797A2 (en) * | 2005-09-29 | 2008-06-18 | Bayer HealthCare AG | Pde inhibitors and combinations thereof for the treatment of urological disorders |
| CA2663436A1 (en) * | 2006-10-04 | 2008-04-10 | Pfizer Products Inc. | Pyrido[4,3-d]pyrimidin-4(3h)-one derivatives as calcium receptor antagonists |
| CN101711153A (zh) * | 2007-06-13 | 2010-05-19 | 拜耳先灵制药股份公司 | 用于治疗听觉损伤的pde抑制剂 |
| CN101531638B (zh) * | 2008-03-13 | 2011-12-28 | 中国科学院广州生物医药与健康研究院 | 用作雌激素相关受体调节剂的化合物及其应用 |
| CN102098918A (zh) * | 2008-05-13 | 2011-06-15 | 帕纳德制药公司 | 用于治疗癌症和神经退行性疾病的生物活性化合物 |
| CN101628913B (zh) | 2008-07-18 | 2013-01-23 | 中国科学院广州生物医药与健康研究院 | 用作雌激素相关受体调节剂的化合物及其应用 |
| KR102200628B1 (ko) * | 2012-09-26 | 2021-01-08 | 메르크 파텐트 게엠베하 | Ｐａｒｐ 억제제로서의 퀴나졸리논 유도체 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3265697A (en) * | 1964-09-04 | 1966-08-09 | Shulton Inc | 2-p-dialkylaminoalkoxyphenyl-2, 3-dihydro-4 (1h)-quinazolinones and their derivatives |
| DE1939109A1 (de) * | 1968-08-31 | 1970-03-05 | Troponwerke Dinklage & Co | 2-Methyl-3-[2-(2-diaethylaminoaethoxy)-phenyl]-chinazolinon-(4) und Verfahren zu seiner Herstellung |
| US3862191A (en) * | 1972-09-27 | 1975-01-21 | Pfizer | Pyrido{8 2,3-d{9 pyrimidin-4(3H)-one |
-
1981
- 1981-10-21 EP EP81108623A patent/EP0054132B1/de not_active Expired
- 1981-10-21 DE DE8181108623T patent/DE3166627D1/de not_active Expired
- 1981-11-18 SU SU813354550A patent/SU1056900A3/ru active
- 1981-11-26 DK DK525481A patent/DK525481A/da not_active Application Discontinuation
- 1981-12-04 US US06/327,348 patent/US4379788A/en not_active Expired - Fee Related
- 1981-12-07 ES ES507761A patent/ES507761A0/es active Granted
- 1981-12-07 DD DD81235494A patent/DD208151A5/de unknown
- 1981-12-10 GR GR66768A patent/GR76952B/el unknown
- 1981-12-10 FI FI813971A patent/FI813971L/fi not_active Application Discontinuation
- 1981-12-10 PL PL1981234175A patent/PL135330B1/pl unknown
- 1981-12-10 CS CS819180A patent/CS227024B2/cs unknown
- 1981-12-10 IL IL64504A patent/IL64504A/xx unknown
- 1981-12-11 NO NO814239A patent/NO814239L/no unknown
- 1981-12-11 GB GB8137458A patent/GB2090249B/en not_active Expired
- 1981-12-11 PT PT74116A patent/PT74116B/pt unknown
- 1981-12-11 PH PH26759A patent/PH18930A/en unknown
- 1981-12-11 CA CA000392067A patent/CA1217767A/en not_active Expired
- 1981-12-11 NZ NZ199254A patent/NZ199254A/en unknown
- 1981-12-11 AR AR287776A patent/AR227567A1/es active
- 1981-12-11 AU AU78473/81A patent/AU543568B2/en not_active Ceased
- 1981-12-11 HU HU813747A patent/HU187384B/hu unknown
-
1982
- 1982-04-30 ES ES82511835A patent/ES511835A0/es active Granted
-
1987
- 1987-12-30 MY MY562/87A patent/MY8700562A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DD208151A5 (de) | 1984-03-28 |
| NZ199254A (en) | 1985-02-28 |
| FI813971L (fi) | 1982-06-13 |
| IL64504A (en) | 1985-02-28 |
| CA1217767A (en) | 1987-02-10 |
| DE3166627D1 (en) | 1984-11-15 |
| AU543568B2 (en) | 1985-04-26 |
| SU1056900A3 (ru) | 1983-11-23 |
| GR76952B (es) | 1984-09-04 |
| US4379788A (en) | 1983-04-12 |
| ES8207156A1 (es) | 1982-09-01 |
| CS227024B2 (en) | 1984-04-16 |
| GB2090249A (en) | 1982-07-07 |
| AU7847381A (en) | 1982-06-17 |
| ES8304096A1 (es) | 1983-02-16 |
| EP0054132A1 (de) | 1982-06-23 |
| MY8700562A (en) | 1987-12-31 |
| AR227567A1 (es) | 1982-11-15 |
| PL234175A1 (es) | 1982-08-16 |
| IL64504A0 (en) | 1982-03-31 |
| PL135330B1 (en) | 1985-10-31 |
| DK525481A (da) | 1982-06-13 |
| NO814239L (no) | 1982-06-14 |
| PT74116A (de) | 1982-01-01 |
| PT74116B (de) | 1983-12-19 |
| ES511835A0 (es) | 1983-02-16 |
| GB2090249B (en) | 1984-08-22 |
| ES507761A0 (es) | 1982-09-01 |
| HU187384B (en) | 1985-12-28 |
| EP0054132B1 (de) | 1984-10-10 |
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