PH12013500923A1 - Compositions of rotigotine, derivatives thereof, or pharmaceutically acceptable salts of rotigotine or its derivative - Google Patents
Compositions of rotigotine, derivatives thereof, or pharmaceutically acceptable salts of rotigotine or its derivativeInfo
- Publication number
- PH12013500923A1 PH12013500923A1 PH1/2013/500923A PH12013500923A PH12013500923A1 PH 12013500923 A1 PH12013500923 A1 PH 12013500923A1 PH 12013500923 A PH12013500923 A PH 12013500923A PH 12013500923 A1 PH12013500923 A1 PH 12013500923A1
- Authority
- PH
- Philippines
- Prior art keywords
- rotigotine
- composition
- pharmaceutically acceptable
- derivative
- derivatives
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 5
- KFQYTPMOWPVWEJ-INIZCTEOSA-N rotigotine Chemical group CCCN([C@@H]1CC2=CC=CC(O)=C2CC1)CCC1=CC=CS1 KFQYTPMOWPVWEJ-INIZCTEOSA-N 0.000 title abstract 3
- 229960003179 rotigotine Drugs 0.000 title abstract 3
- 150000003839 salts Chemical class 0.000 title abstract 2
- 235000014113 dietary fatty acids Nutrition 0.000 abstract 2
- 229930195729 fatty acid Natural products 0.000 abstract 2
- 239000000194 fatty acid Substances 0.000 abstract 2
- 150000004665 fatty acids Chemical class 0.000 abstract 2
- 229920001606 poly(lactic acid-co-glycolic acid) Polymers 0.000 abstract 2
- 208000018737 Parkinson disease Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Inorganic Chemistry (AREA)
- Psychology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201010576447 | 2010-11-25 | ||
| PCT/CN2011/001958 WO2012068783A1 (en) | 2010-11-25 | 2011-11-25 | Compositions of rotigotine, derivatives thereof, or pharmaceutically acceptable salts of rotigotine or its derivative |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH12013500923A1 true PH12013500923A1 (en) | 2016-02-08 |
Family
ID=46145374
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH1/2013/500923A PH12013500923A1 (en) | 2010-11-25 | 2011-11-25 | Compositions of rotigotine, derivatives thereof, or pharmaceutically acceptable salts of rotigotine or its derivative |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US9265835B2 (https=) |
| EP (1) | EP2642993B1 (https=) |
| JP (2) | JP6006225B2 (https=) |
| KR (1) | KR101481643B1 (https=) |
| CN (1) | CN103458895B (https=) |
| AU (1) | AU2011334494B2 (https=) |
| BR (1) | BR112013012726B1 (https=) |
| CA (1) | CA2816288C (https=) |
| ES (1) | ES2572948T3 (https=) |
| MY (1) | MY165003A (https=) |
| PH (1) | PH12013500923A1 (https=) |
| PL (1) | PL2642993T3 (https=) |
| RU (1) | RU2589700C2 (https=) |
| WO (1) | WO2012068783A1 (https=) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8682462B2 (en) | 2011-08-13 | 2014-03-25 | Colin M. Leonard | Systems and methods for dynamic audio processing |
| US11074031B1 (en) | 2016-09-06 | 2021-07-27 | Colin Leonard | Systems and methods for dynamic audio processing |
| EP2559435A1 (en) | 2011-08-19 | 2013-02-20 | UCB Pharma GmbH | Rotigotine in the treatment of hemispatial neglect, stroke and deficits following stroke |
| KR101558042B1 (ko) * | 2012-07-05 | 2015-10-07 | 에스케이케미칼주식회사 | 로티고틴을 함유한 경피흡수제제 |
| CA2935311C (en) | 2013-12-31 | 2018-11-27 | Pb&B Sa | Controlled release fatty acid compositions for use in body reconstruction and body-shaping |
| CN105310974B (zh) * | 2014-08-01 | 2019-08-23 | 山东绿叶制药有限公司 | 罗替戈汀及其衍生物或其药用盐的植入剂 |
| CN106474070B (zh) * | 2015-08-26 | 2020-03-17 | 四川科伦药物研究院有限公司 | 一种克服停滞期、恒速释放疏水性药物的微球及制备方法 |
| CN105963253A (zh) * | 2016-06-19 | 2016-09-28 | 朱武欣 | 一种罗替戈汀长效水性混悬型注射剂 |
| ES2855976T3 (es) * | 2016-07-21 | 2021-09-27 | Shandong luye pharmaceutical co ltd | Behenato de rotigotina y procedimiento de fabricación y aplicación del mismo |
| WO2018045000A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Picolinamides as fungicides |
| WO2018096560A1 (en) | 2016-11-23 | 2018-05-31 | Cipla Limited | Long acting depot formulation for the continuous dopaminergic stimulation |
| KR102089737B1 (ko) * | 2017-11-01 | 2020-03-16 | 한국화학연구원 | 에씨탈로프람을 함유한 미립구형 서방출 주사제 및 그의 제조방법 |
| KR102181231B1 (ko) * | 2018-11-22 | 2020-11-20 | 주식회사 메디포럼제약 | 로티고틴 함유 고분자 미립자의 제조방법 |
| EP4104820A4 (en) * | 2020-02-14 | 2024-04-17 | G2GBIO, Inc. | Pharmaceutical composition comprising sustained-release microspheres including glp-1 analogue or pharmaceutically acceptable salt thereof |
| WO2025243901A1 (ja) * | 2024-05-21 | 2025-11-27 | 株式会社 SENTAN Pharma | 注射製剤 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9718986D0 (en) * | 1997-09-09 | 1997-11-12 | Danbiosyst Uk | Controlled release microsphere delivery system |
| DE10234673B4 (de) * | 2002-07-30 | 2007-08-16 | Schwarz Pharma Ag | Heißschmelz-TTS zur Verabreichung von Rotigotin und Verfahren zu seiner Herstellung sowie Verwendung von Rotigotin bei der Herstellung eines TTS im Heißschmelzverfahren |
| JP4927729B2 (ja) | 2004-07-16 | 2012-05-09 | オークウッド ラボラトリーズ，エル．エル．シー． | 性腺刺激ホルモン放出ホルモンアンタゴニスト |
| CN1762495B (zh) | 2004-09-21 | 2011-04-06 | 山东绿叶制药有限公司 | 含有多巴胺受体激动剂类药物的长效缓释制剂及其制备工艺 |
| KR20070059161A (ko) | 2004-09-21 | 2007-06-11 | 산동 루예 파마슈티칼 컴파니 리미티드 | 도파민 수용체 효능제를 함유하는 장시간 작용 서방성 제제및 그 제조방법 |
| JP5222550B2 (ja) | 2007-12-27 | 2013-06-26 | 財團法人工業技術研究院 | 徐放性組成物およびその製造方法 |
-
2011
- 2011-11-25 RU RU2013128430/15A patent/RU2589700C2/ru active
- 2011-11-25 EP EP11843219.4A patent/EP2642993B1/en active Active
- 2011-11-25 JP JP2013540214A patent/JP6006225B2/ja active Active
- 2011-11-25 CA CA2816288A patent/CA2816288C/en active Active
- 2011-11-25 BR BR112013012726-0A patent/BR112013012726B1/pt active IP Right Grant
- 2011-11-25 US US13/989,550 patent/US9265835B2/en active Active
- 2011-11-25 AU AU2011334494A patent/AU2011334494B2/en active Active
- 2011-11-25 CN CN201180049447.2A patent/CN103458895B/zh active Active
- 2011-11-25 WO PCT/CN2011/001958 patent/WO2012068783A1/en not_active Ceased
- 2011-11-25 MY MYPI2013001807A patent/MY165003A/en unknown
- 2011-11-25 PH PH1/2013/500923A patent/PH12013500923A1/en unknown
- 2011-11-25 ES ES11843219.4T patent/ES2572948T3/es active Active
- 2011-11-25 KR KR20137013119A patent/KR101481643B1/ko active Active
- 2011-11-25 PL PL11843219.4T patent/PL2642993T3/pl unknown
-
2015
- 2015-08-21 JP JP2015163527A patent/JP6067803B2/ja active Active
Also Published As
| Publication number | Publication date |
|---|---|
| AU2011334494B2 (en) | 2015-11-05 |
| CN103458895B (zh) | 2014-07-09 |
| WO2012068783A1 (en) | 2012-05-31 |
| JP6067803B2 (ja) | 2017-01-25 |
| EP2642993A4 (en) | 2014-05-14 |
| RU2589700C2 (ru) | 2016-07-10 |
| CA2816288C (en) | 2016-01-26 |
| RU2013128430A (ru) | 2014-12-27 |
| JP6006225B2 (ja) | 2016-10-12 |
| US20130309314A1 (en) | 2013-11-21 |
| US9265835B2 (en) | 2016-02-23 |
| KR101481643B1 (ko) | 2015-01-12 |
| PL2642993T3 (pl) | 2016-09-30 |
| JP2013543874A (ja) | 2013-12-09 |
| BR112013012726B1 (pt) | 2022-03-29 |
| CN103458895A (zh) | 2013-12-18 |
| CA2816288A1 (en) | 2012-05-31 |
| EP2642993A1 (en) | 2013-10-02 |
| MY165003A (en) | 2018-02-28 |
| KR20130130727A (ko) | 2013-12-02 |
| HK1186978A1 (en) | 2014-03-28 |
| AU2011334494A1 (en) | 2013-07-11 |
| ES2572948T3 (es) | 2016-06-03 |
| JP2016028043A (ja) | 2016-02-25 |
| US20140377369A2 (en) | 2014-12-25 |
| BR112013012726A2 (https=) | 2017-04-04 |
| EP2642993B1 (en) | 2016-03-02 |
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