PE20171177A1 - Compuestos aminopirimidinilo inhibidores de jak - Google Patents

Compuestos aminopirimidinilo inhibidores de jak

Info

Publication number
PE20171177A1
PE20171177A1 PE2017000248A PE2017000248A PE20171177A1 PE 20171177 A1 PE20171177 A1 PE 20171177A1 PE 2017000248 A PE2017000248 A PE 2017000248A PE 2017000248 A PE2017000248 A PE 2017000248A PE 20171177 A1 PE20171177 A1 PE 20171177A1
Authority
PE
Peru
Prior art keywords
deuterium
alkyl
bond
compounds
aminopyrimidinyl
Prior art date
Application number
PE2017000248A
Other languages
English (en)
Spanish (es)
Inventor
Andrew Fensome
Ariamala Gopalsamy
Brian S Gerstenberger
Ivan Viktorovich Efremov
Zhao-Kui Wan
Betsy PIERCE
Jean-Baptiste Telliez
Jhon I Trujillo
Liying Zhang
Li Xing
Eddine Saiah
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54148580&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20171177(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of PE20171177A1 publication Critical patent/PE20171177A1/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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PE2017000248A 2014-08-21 2015-08-07 Compuestos aminopirimidinilo inhibidores de jak PE20171177A1 (es)

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US201462039969P 2014-08-21 2014-08-21

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PE20171177A1 true PE20171177A1 (es) 2017-08-22

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US (5) US9663526B2 (enExample)
EP (1) EP3183247B9 (enExample)
JP (1) JP6218260B2 (enExample)
KR (1) KR101877189B1 (enExample)
CN (1) CN107074867B (enExample)
AP (1) AP2017009748A0 (enExample)
AR (1) AR101599A1 (enExample)
AU (1) AU2015304883B2 (enExample)
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MD4800B1 (ro) 2022-03-31
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