PE20110116A1 - Asociacion de ivabradina y perindopril y composicion farmaceutica que la contiene - Google Patents

Asociacion de ivabradina y perindopril y composicion farmaceutica que la contiene

Info

Publication number
PE20110116A1
PE20110116A1 PE2010001026A PE2010001026A PE20110116A1 PE 20110116 A1 PE20110116 A1 PE 20110116A1 PE 2010001026 A PE2010001026 A PE 2010001026A PE 2010001026 A PE2010001026 A PE 2010001026A PE 20110116 A1 PE20110116 A1 PE 20110116A1
Authority
PE
Peru
Prior art keywords
ivabradine
perindopril
pharmaceutical composition
association
composition containing
Prior art date
Application number
PE2010001026A
Other languages
English (en)
Inventor
Vidal Benatar
Guy Lerebours-Pigeonniere
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36685870&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20110116(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Servier Lab filed Critical Servier Lab
Publication of PE20110116A1 publication Critical patent/PE20110116A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/4045Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA QUE COMPRENDE: A) UN INHIBIDOR SELECTIVO DE LA CORRIENTE SINUSAL TAL COMO IVABRADINA EN FORMA DE SAL DE HIDROCLORURO, SUS HIDRATOS O FORMAS CRISTALINAS; B)UN AGENTE INHIBIDOR DE LA ENZIMA CONVERTIDORA DE ANGIOTENSINA TAL COMO PERINDOPRIL EN FORMA DE SAL TERCBUTILAMINA O DE ARGININA Y UNO O VARIOS EXCIPIENTES FARMACEUTICAMENTE ACEPTABLES. DICHA COMPOSICION ES UTIL EN EL TRATAMIENTO DE LA HIPERTENSION ARTERIAL
PE2010001026A 2005-12-21 2006-12-18 Asociacion de ivabradina y perindopril y composicion farmaceutica que la contiene PE20110116A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0513006A FR2894825B1 (fr) 2005-12-21 2005-12-21 Nouvelle association d'un inhibiteur du courant if sinusal et d'un inhibiteur de l'enzyme de conversion et les compositions pharmaceutiques qui la contiennent

Publications (1)

Publication Number Publication Date
PE20110116A1 true PE20110116A1 (es) 2011-03-02

Family

ID=36685870

Family Applications (2)

Application Number Title Priority Date Filing Date
PE2010001026A PE20110116A1 (es) 2005-12-21 2006-12-18 Asociacion de ivabradina y perindopril y composicion farmaceutica que la contiene
PE2006001619A PE20071004A1 (es) 2005-12-21 2006-12-18 Composiciones farmaceuticas que comprenden la combinacion de ivabradina y perindropil

Family Applications After (1)

Application Number Title Priority Date Filing Date
PE2006001619A PE20071004A1 (es) 2005-12-21 2006-12-18 Composiciones farmaceuticas que comprenden la combinacion de ivabradina y perindropil

Country Status (42)

Country Link
US (2) US20070142355A1 (es)
EP (2) EP1800678B1 (es)
JP (2) JP4705564B2 (es)
KR (2) KR100907583B1 (es)
CN (1) CN101015557B (es)
AP (1) AP2119A (es)
AR (1) AR058574A1 (es)
AT (1) ATE508742T1 (es)
AU (1) AU2006252210B2 (es)
BR (1) BRPI0605517A (es)
CA (1) CA2571644C (es)
CO (1) CO5790168A1 (es)
CR (1) CR8820A (es)
CY (1) CY1111575T1 (es)
DK (1) DK1800678T3 (es)
EA (1) EA011253B1 (es)
ES (1) ES2366570T3 (es)
FR (1) FR2894825B1 (es)
GE (1) GEP20094604B (es)
GT (1) GT200600522A (es)
HK (1) HK1106444A1 (es)
HR (1) HRP20110532T1 (es)
IL (1) IL180204A (es)
JO (1) JO2699B1 (es)
MA (1) MA28723B1 (es)
ME (1) ME01958B (es)
MX (1) MXPA06014885A (es)
MY (1) MY146956A (es)
NO (1) NO337640B1 (es)
NZ (1) NZ552221A (es)
PE (2) PE20110116A1 (es)
PL (1) PL1800678T3 (es)
PT (1) PT1800678E (es)
RS (1) RS51731B (es)
SA (1) SA06270480B1 (es)
SG (2) SG173243A1 (es)
SI (1) SI1800678T1 (es)
TW (1) TWI369206B (es)
UA (1) UA86417C2 (es)
UY (1) UY30023A1 (es)
WO (1) WO2007077327A1 (es)
ZA (1) ZA200610824B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2894825B1 (fr) * 2005-12-21 2010-12-03 Servier Lab Nouvelle association d'un inhibiteur du courant if sinusal et d'un inhibiteur de l'enzyme de conversion et les compositions pharmaceutiques qui la contiennent
FR2920772B1 (fr) * 2007-09-11 2009-10-23 Servier Lab Association entre un anti-atherothrombotique et un inhibiteur de l'enzyme de conversion de l'angiotensine
FR2927538B1 (fr) * 2008-02-14 2010-02-19 Servier Lab Association d'un inhibiteur du courant if sinusal et d'un beta-bloquant.
CN101564394B (zh) * 2008-04-21 2010-12-15 鲁南制药集团股份有限公司 含有伊伐布雷定和曲美他嗪的药物组合物
FR2961105B1 (fr) * 2010-06-15 2013-02-08 Servier Lab Utilisation de l'association d'un inhibiteur du courant if sinusal et d'un inhibiteur de l'enzyme de conversion de l'angiotensine pour le traitement de l'insuffisance cardiaque
WO2013116738A1 (en) * 2012-02-03 2013-08-08 Cardeus Pharmaceuticals, Inc. Drug formulations
FR3050380B1 (fr) 2016-04-20 2020-07-10 Les Laboratoires Servier Composition pharmaceutique comprenant un betabloquant, un inhibiteur de l'enzyme de conversion et un antihypertenseur ou un ains.

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4508729A (en) * 1979-12-07 1985-04-02 Adir Substituted iminodiacids, their preparation and pharmaceutical compositions containing them
DE3736866A1 (de) * 1987-10-30 1989-05-11 Thomae Gmbh Dr K Mittel zur behandlung des bluthochdrucks und der herzinsuffizienz
FR2681862B1 (fr) * 1991-09-27 1993-11-12 Adir Cie Nouvelles (benzocycloalkyl)alkylamines, leur procede de preparation, et les compositions pharmaceutiques qui les contiennent.
DE10018401A1 (de) * 2000-04-13 2001-10-25 Boehringer Ingelheim Pharma Verwendung von Bradycardica bei der Behandlung von mit Hypertrophie einhergehenden Myocarderkrankungen und neue Arzneimittelkombinationen
CA2449934A1 (en) * 2001-06-08 2002-12-19 Ortho-Mcneil Pharmaceutical, Inc. Treating pain by targeting hyperpolarization-activated, cyclic nucleotide-gated channels
AR036187A1 (es) * 2001-07-24 2004-08-18 Adir Un proceso para la preparacion de perindopril, compuestos analogos y sus sales, compuesto intermediario 2,5-dioxo-oxazolidina y proceso para preparar un intermediario
US20040242565A1 (en) * 2001-09-11 2004-12-02 Yoshinori Toshima Medicinal composition for prevention of or treatment for cerebrovascular disorder and cardiopathy
FR2834896B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible d'ivabradine
FR2838648B1 (fr) * 2002-04-18 2004-05-21 Servier Lab Nouveau sel de perindopril et les compositions pharmaceutiques qui le contiennent
DE60200160T2 (de) * 2002-07-25 2004-11-04 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verwendung von Cilobradine oder pharmazeutisch akzeptablen Salze zur Behandlung oder Prävention von Herzversagen
FR2882556B1 (fr) * 2005-02-28 2007-05-04 Servier Lab Forme cristalline gamma d du chlorhydrate de l'ivabradine, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
FR2882555B1 (fr) * 2005-02-28 2007-05-04 Servier Lab Forme cristalline gamma du chlorhydrate de l'ivabradine, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
FR2882554B1 (fr) * 2005-02-28 2007-05-04 Servier Lab Forme critalline beta d du chlorhydrate de l'ivabradine, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
FR2882553B1 (fr) * 2005-02-28 2007-05-04 Servier Lab Forme cristalline beta du chlorhydrate de l'ivabradine, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
FR2894825B1 (fr) * 2005-12-21 2010-12-03 Servier Lab Nouvelle association d'un inhibiteur du courant if sinusal et d'un inhibiteur de l'enzyme de conversion et les compositions pharmaceutiques qui la contiennent

Also Published As

Publication number Publication date
KR100907583B1 (ko) 2009-07-14
JO2699B1 (en) 2013-03-03
ATE508742T1 (de) 2011-05-15
NO20065905L (no) 2007-06-22
SI1800678T1 (sl) 2011-08-31
PT1800678E (pt) 2011-07-12
SA06270480B1 (ar) 2011-02-23
IL180204A (en) 2014-02-27
ES2366570T3 (es) 2011-10-21
EA200602155A1 (ru) 2007-08-31
EP1800678B1 (fr) 2011-05-11
CN101015557B (zh) 2010-12-08
HK1106444A1 (en) 2008-03-14
AP2119A (en) 2010-04-21
JP2007169283A (ja) 2007-07-05
HRP20110532T1 (hr) 2011-08-31
ZA200610824B (en) 2008-06-25
PE20071004A1 (es) 2007-11-17
ME01958B (me) 2011-10-31
TWI369206B (en) 2012-08-01
AU2006252210A1 (en) 2007-07-05
EA011253B1 (ru) 2009-02-27
KR20090047424A (ko) 2009-05-12
KR20070066921A (ko) 2007-06-27
MA28723B1 (fr) 2007-07-02
CN101015557A (zh) 2007-08-15
DK1800678T3 (da) 2011-08-15
GT200600522A (es) 2007-07-25
CR8820A (es) 2007-08-28
GEP20094604B (en) 2009-02-10
AU2006252210B2 (en) 2012-04-26
EP1800678A1 (fr) 2007-06-27
PL1800678T3 (pl) 2011-08-31
CY1111575T1 (el) 2015-10-07
IL180204A0 (en) 2008-01-20
NO337640B1 (no) 2016-05-23
CO5790168A1 (es) 2007-08-31
CA2571644A1 (fr) 2007-06-21
US20120196850A1 (en) 2012-08-02
CA2571644C (fr) 2011-03-08
MXPA06014885A (es) 2009-02-11
FR2894825B1 (fr) 2010-12-03
SG173243A1 (en) 2011-08-29
BRPI0605517A (pt) 2007-10-16
UA86417C2 (ru) 2009-04-27
RS51731B (en) 2011-10-31
NZ552221A (en) 2008-05-30
JP2011079854A (ja) 2011-04-21
TW200744608A (en) 2007-12-16
AR058574A1 (es) 2008-02-13
UY30023A1 (es) 2007-01-31
WO2007077327A1 (fr) 2007-07-12
JP4705564B2 (ja) 2011-06-22
MY146956A (en) 2012-10-15
FR2894825A1 (fr) 2007-06-22
EP2298297A1 (fr) 2011-03-23
SG133545A1 (en) 2007-07-30
US20070142355A1 (en) 2007-06-21
AP2006003859A0 (en) 2006-12-31

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