PE20070431A1 - Compuestos y composiciones de carboxamidas sustituidas como moduladores de receptores cannabinoides - Google Patents
Compuestos y composiciones de carboxamidas sustituidas como moduladores de receptores cannabinoidesInfo
- Publication number
- PE20070431A1 PE20070431A1 PE2006000600A PE2006000600A PE20070431A1 PE 20070431 A1 PE20070431 A1 PE 20070431A1 PE 2006000600 A PE2006000600 A PE 2006000600A PE 2006000600 A PE2006000600 A PE 2006000600A PE 20070431 A1 PE20070431 A1 PE 20070431A1
- Authority
- PE
- Peru
- Prior art keywords
- independently
- compounds
- modulators
- compositions
- carboxamide
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
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Abstract
SE REFIERE A COMPUESTOS DE FORMULA (I) EN DONDE U y V SON INDEPENDIENTEMENTE C O N; W, X E Y SON INDEPENDIENTEMENTE C, N, O, S o C(O) SIEMPRE QUE AL MENOS DOS U, V, W, X, O Y SE SELECCIONEN INDEPENDIENTENTE DE N, O, C(O) O S; R, R1, R2 SON INDEPENDIENTEMENTE H, NITRO, ALQUILO, ARILO, CICLOALQUILO, HETEROARILO, NR3R4, ENTRE OTROS OPCIONALMENTE SUSTITUIDOS; B ES O, S o NR3; p Y m SON INDEPENDIENTEMENTE 0, 1 O 2; A ES UN GRUPO TRICICLO[5.2.2.0]UNDECAN, TETRACICLO[7.3.1.1]TETRADECAN, BICICLO[2.2.1]HEPTAN, ENTRE OTROS, OPCIONALMENTE SUSTITUIDOS CON R5, R6, R7, R8, R9, R10, R11, R12, R13 Y R14 LOS CUALES SON INDEPENDIENTEMENTE H, NITRO, CIANO, ACETILO, ENTRE OTROS. SON PREFERIDOS: N(7)-PIPERIDIN-5-(2-BROMOFENIL)-5,6-DIAZATETRACICLO[7.3.1.1(3.11).0(4.8)]TETRADECA-4(8),6-DIEN-7-CARBOXAMIDA, N(3)-BENCIL-1-FENIL-4,5,6,7-TETRAHIDRO-1H-4,7-METAN-INDAZOL-3-CARBOXAMIDA, ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA Y UN PROCEDIMIENTO DE PREPARACION. ESTOS COMPUESTOS SON MODULADORES DEL RECEPTOR CANNABINOIDE 1 (CB1) O DEL RECEPTOR CANNABINOIDE 2 (CB2) Y SON UTILES PARA EL TRATAMIENTO DEL DOLOR, TRASTORNOS DEGENERATIVOS, ALIMENTICIOS, PERDIDA O CONTROL DE PESO, Y OBESIDAD
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN659MU2005 | 2005-06-02 | ||
US69643305P | 2005-07-01 | 2005-07-01 | |
IN1370MU2005 | 2005-10-31 | ||
IN344MU2006 | 2006-03-09 | ||
US74407106P | 2006-03-31 | 2006-03-31 | |
IN689MU2006 | 2006-05-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20070431A1 true PE20070431A1 (es) | 2007-06-27 |
Family
ID=37056437
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2006000600A PE20070431A1 (es) | 2005-06-02 | 2006-06-02 | Compuestos y composiciones de carboxamidas sustituidas como moduladores de receptores cannabinoides |
Country Status (12)
Country | Link |
---|---|
US (1) | US8420689B2 (es) |
EP (1) | EP1902034B1 (es) |
JP (1) | JP2008545739A (es) |
AR (1) | AR055199A1 (es) |
AU (1) | AU2006253842A1 (es) |
CA (1) | CA2613678A1 (es) |
HK (1) | HK1118806A1 (es) |
MY (1) | MY142409A (es) |
PE (1) | PE20070431A1 (es) |
PL (1) | PL1902034T3 (es) |
TW (1) | TW200716560A (es) |
WO (1) | WO2006129178A1 (es) |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7923465B2 (en) | 2005-06-02 | 2011-04-12 | Glenmark Pharmaceuticals S.A. | Cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation |
JP2010509201A (ja) * | 2006-11-03 | 2010-03-25 | グレンマーク・ファーマシューティカルズ・エスエー | 新規なカンナビノイド受容体リガンド、およびこれらを含む薬剤組成物、およびこれらの調製方法 |
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- 2006-06-01 WO PCT/IB2006/001437 patent/WO2006129178A1/en active Application Filing
- 2006-06-01 PL PL06755930T patent/PL1902034T3/pl unknown
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- 2006-06-02 PE PE2006000600A patent/PE20070431A1/es not_active Application Discontinuation
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CA2613678A1 (en) | 2006-12-07 |
WO2006129178A1 (en) | 2006-12-07 |
AR055199A1 (es) | 2007-08-08 |
HK1118806A1 (en) | 2009-02-20 |
US8420689B2 (en) | 2013-04-16 |
JP2008545739A (ja) | 2008-12-18 |
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