OA13258A - Amino acids with affinity for the alpha2delta-protein. - Google Patents

Amino acids with affinity for the alpha2delta-protein. Download PDF

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Publication number
OA13258A
OA13258A OA1200600094A OA1200600094A OA13258A OA 13258 A OA13258 A OA 13258A OA 1200600094 A OA1200600094 A OA 1200600094A OA 1200600094 A OA1200600094 A OA 1200600094A OA 13258 A OA13258 A OA 13258A
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OA
OAPI
Prior art keywords
acid
phenyl
amino
aminomethyl
methyl
Prior art date
Application number
OA1200600094A
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English (en)
Inventor
Christopher James Deur
Christine Nylund Kolz
Augustine Tobi Osuma
Mark Stephen Plummer
Jacob Bradley Schwarz
Andrew John Thorpe
David Juergen Wustrow
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Warner Lambert Co
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34396281&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA13258(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of OA13258A publication Critical patent/OA13258A/en

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    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
    • C07C229/08—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to hydrogen atoms
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • C07D263/18—Oxygen atoms
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  • Physical Education & Sports Medicine (AREA)
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OA1200600094A 2003-09-25 2004-09-13 Amino acids with affinity for the alpha2delta-protein. OA13258A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50595303P 2003-09-25 2003-09-25
US50744303P 2003-09-30 2003-09-30

Publications (1)

Publication Number Publication Date
OA13258A true OA13258A (en) 2007-01-31

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OA1200600094A OA13258A (en) 2003-09-25 2004-09-13 Amino acids with affinity for the alpha2delta-protein.

Country Status (27)

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US (3) US20050124668A1 (nl)
EP (1) EP1667957A2 (nl)
JP (2) JP4001349B2 (nl)
KR (2) KR20070039986A (nl)
AP (1) AP2006003544A0 (nl)
AR (1) AR046022A1 (nl)
AU (1) AU2004276072A1 (nl)
BR (1) BRPI0414781A (nl)
CA (1) CA2540208A1 (nl)
CO (1) CO5680413A2 (nl)
CR (1) CR8290A (nl)
EA (1) EA200600467A1 (nl)
EC (1) ECSP066450A (nl)
IL (1) IL173764A0 (nl)
IS (1) IS8308A (nl)
MA (1) MA28048A1 (nl)
MX (1) MXPA06003395A (nl)
NL (2) NL1027115C2 (nl)
NO (1) NO20061812L (nl)
OA (1) OA13258A (nl)
PA (1) PA8613101A1 (nl)
PE (1) PE20050434A1 (nl)
RS (1) RS20060210A (nl)
TN (1) TNSN06095A1 (nl)
TW (1) TW200528420A (nl)
UY (1) UY28533A1 (nl)
WO (1) WO2005030700A2 (nl)

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KR20080019732A (ko) * 2004-07-09 2008-03-04 워너-램버트 캄파니 엘엘씨 알파-2-델타 단백질에 대한 친화도를 갖는 베타-아미노산의제조 방법
BRPI0609435A2 (pt) * 2005-03-24 2010-04-06 Pharmacia & Upjohn Co Llc preparação de beta-aminoácidos opticamente puros tendo afinidade com a proteìna alfa-2-delta
JP2009516675A (ja) * 2005-11-17 2009-04-23 ファイザー・リミテッド 疼痛を治療するためのイソシステイン誘導体
BRPI0708671A2 (pt) * 2006-03-06 2011-06-07 Pfizer Prod Inc ligantes alfa-2-delta para sono não restaurador
AR061728A1 (es) * 2006-06-30 2008-09-17 Pfizer Prod Inc Composicion para tratamiento usando compuestos selectivos alfa-2-delta-1
EP1903027A1 (en) 2006-09-13 2008-03-26 Novartis AG Process for preparing biaryl substituted 4-amino-butyric acid or derivatives thereof and their use in the production of NEP inhibitors
US20110124705A1 (en) * 2009-11-24 2011-05-26 Xenoport, Inc. Prodrugs of alpha-2-delta ligands, pharmaceutical compositions and uses thereof
US20110130454A1 (en) * 2009-11-24 2011-06-02 Xenoport, Inc. Prodrugs of gamma-amino acid, alpha-2-delta ligands, pharmaceutical compositions and uses thereof
WO2014069626A1 (ja) * 2012-11-01 2014-05-08 協和発酵キリン株式会社 ピリミドジアゼピノン化合物の製造方法
CA2952934A1 (en) 2014-06-26 2015-12-30 Island Breeze Systems Ca, Llc Mdi related products and methods of use
CN114700006B (zh) * 2022-06-07 2023-03-24 北京先通国际医药科技股份有限公司 一种液体组合物的生产设备及其制备方法和用途

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