OA11438A - Novel macrolides. - Google Patents

Novel macrolides. Download PDF

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Publication number
OA11438A
OA11438A OA1200000192A OA1200000192A OA11438A OA 11438 A OA11438 A OA 11438A OA 1200000192 A OA1200000192 A OA 1200000192A OA 1200000192 A OA1200000192 A OA 1200000192A OA 11438 A OA11438 A OA 11438A
Authority
OA
OAPI
Prior art keywords
alkyl
groups
optionally
substituted
halo
Prior art date
Application number
OA1200000192A
Other languages
English (en)
Inventor
John Philip Dirlam
Hamish Alastair Irvin Mcarthur
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of OA11438A publication Critical patent/OA11438A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
OA1200000192A 1998-01-02 2000-06-30 Novel macrolides. OA11438A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7034398P 1998-01-02 1998-01-02

Publications (1)

Publication Number Publication Date
OA11438A true OA11438A (en) 2004-04-30

Family

ID=22094723

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200000192A OA11438A (en) 1998-01-02 2000-06-30 Novel macrolides.

Country Status (34)

Country Link
US (2) US6472371B1 (ja)
EP (1) EP1044207A1 (ja)
JP (1) JP2002500230A (ja)
KR (1) KR100352809B1 (ja)
CN (1) CN1284081A (ja)
AP (1) AP9801420A0 (ja)
AR (4) AR014948A1 (ja)
AU (1) AU756409B2 (ja)
BG (1) BG104644A (ja)
BR (1) BR9814601A (ja)
CA (1) CA2316919C (ja)
CO (1) CO4970821A1 (ja)
CZ (1) CZ20002458A3 (ja)
DZ (1) DZ2698A1 (ja)
EA (1) EA200000594A1 (ja)
GT (1) GT199800206A (ja)
HR (1) HRP20000442A2 (ja)
HU (1) HUP0100420A3 (ja)
IL (1) IL137024A0 (ja)
IS (1) IS5528A (ja)
MA (1) MA24729A1 (ja)
NO (1) NO20003347L (ja)
NZ (1) NZ504986A (ja)
OA (1) OA11438A (ja)
PA (1) PA8465301A1 (ja)
PE (1) PE20000049A1 (ja)
PL (1) PL341642A1 (ja)
SK (1) SK9782000A3 (ja)
TN (1) TNSN98238A1 (ja)
TW (1) TW520374B (ja)
UY (2) UY25330A1 (ja)
WO (1) WO1999035156A1 (ja)
YU (1) YU41500A (ja)
ZA (1) ZA9811939B (ja)

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AP9801420A0 (en) 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
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EP1437360A3 (en) * 1998-08-19 2005-04-06 Pfizer Products Inc. C11 Carbamates of macrolide antibacterials
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US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
AU4354900A (en) 1999-04-16 2000-11-02 Kosan Biosciences, Inc. Ketolide antibacterials
WO2000071557A1 (en) 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
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BRPI0515917A (pt) 2004-09-23 2008-08-12 Schering Plough Ltd controle de parasitas em animais pelo uso de novos derivados de éter de oxima de trifluorometanossulfonanilida
MX2007006072A (es) * 2004-11-19 2007-07-11 Schering Plough Ltd Control de parasitos en animales mediante el uso de derivados del parasiticida 2-fenil-3-(1h-pirrol-2-il)acrilonitrilo.
EP1836211B1 (en) * 2004-12-21 2010-03-03 Pfizer Products Inc. Macrolides
EP1890547A2 (en) * 2005-06-09 2008-02-27 Schering-Plough Ltd. Control of parasites in animals by n-[(phenyloxy)phenyl]-1,1,1-trifluoromethanesulfonamide and n-[(phenylsulfanyl)phenyl]-1,1,1-trifluoromethanesulfonamide derivatives
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
CA2672795A1 (en) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
US8084643B2 (en) * 2006-12-13 2011-12-27 Intervet Inc. Water-soluble prodrugs of florfenicol and its analogs
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
HUE037127T2 (hu) 2007-06-27 2018-08-28 Du Pont Állati károkozó irtására szolgáló eljárás
WO2009064953A1 (en) * 2007-11-15 2009-05-22 Enanta Pharmaceuticals, Inc. Use of bridged macrolides or tylosin derivatives in treating inflammatory bowel diseases
TWI401023B (zh) 2008-02-06 2013-07-11 Du Pont 中離子農藥
CA2732017A1 (en) * 2008-07-30 2010-02-04 Intervet International B.V. Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
EP2461684A2 (en) 2009-08-05 2012-06-13 E. I. du Pont de Nemours and Company Mesoionic pesticides
IN2012DN00838A (ja) 2009-08-05 2015-06-26 Du Pont
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
MA34247B1 (fr) 2010-05-27 2013-05-02 Du Pont Forme cristalline du 4-[5-[3-chloro-5-(trifluorométhyl) phényl] -4,5-dihydro-5-(trifluorométhyl)-3-isoxazolyl]-n-[2-oxo-2-[(2, 2,2-trifluoroéthyl) amino] éthyl]-1-naphtalènecarboxamide
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
AU2012211760A1 (en) * 2011-01-31 2013-08-15 Meiji Seika Pharma Co., Ltd. Novel macrolide derivative
JP2014520151A (ja) 2011-06-20 2014-08-21 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 蠕虫感染を処置するためのヘテロ環式化合物
CN102260306B (zh) * 2011-07-22 2012-07-18 山东鲁抗舍里乐药业有限公司 一种制备泰拉霉素的方法
KR20140094026A (ko) 2011-11-28 2014-07-29 이 아이 듀폰 디 네모아 앤드 캄파니 N-(4-퀴놀리닐메틸) 설폰아미드 유도체 및 구충제로서의 이의 용도
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests
WO2014099837A1 (en) 2012-12-18 2014-06-26 E. I. Du Pont De Nemours And Company Sulfonamide anthelmintics
CN105669798B (zh) * 2013-08-23 2019-07-26 普莱柯生物工程股份有限公司 一种大环内酯类化合物
CN103965273B (zh) * 2013-08-23 2016-05-25 普莱柯生物工程股份有限公司 一种大环内酯类化合物

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Also Published As

Publication number Publication date
CA2316919C (en) 2004-10-26
AU756409B2 (en) 2003-01-09
AR014948A1 (es) 2001-04-11
EA200000594A1 (ru) 2001-04-23
HUP0100420A2 (hu) 2001-07-30
AP9801420A0 (en) 1998-12-31
HRP20000442A2 (en) 2001-04-30
NZ504986A (en) 2003-03-28
GT199800206A (es) 2000-06-21
DZ2698A1 (fr) 2003-03-29
TW520374B (en) 2003-02-11
NO20003347D0 (no) 2000-06-27
MA24729A1 (fr) 1999-07-01
IS5528A (is) 2000-06-09
AR020551A2 (es) 2002-05-15
WO1999035156B1 (en) 1999-10-21
US20040092459A1 (en) 2004-05-13
JP2002500230A (ja) 2002-01-08
AU1444799A (en) 1999-07-26
WO1999035156A1 (en) 1999-07-15
BR9814601A (pt) 2000-10-17
US7015203B2 (en) 2006-03-21
YU41500A (sh) 2003-02-28
EP1044207A1 (en) 2000-10-18
AR020851A2 (es) 2002-05-29
ZA9811939B (en) 2000-06-30
BG104644A (en) 2001-01-31
SK9782000A3 (en) 2001-12-03
IL137024A0 (en) 2001-06-14
PE20000049A1 (es) 2000-02-07
KR100352809B1 (ko) 2002-11-01
CZ20002458A3 (cs) 2001-10-17
PA8465301A1 (es) 2000-09-29
HUP0100420A3 (en) 2003-07-28
AR019787A2 (es) 2002-03-13
CN1284081A (zh) 2001-02-14
CO4970821A1 (es) 2000-11-07
PL341642A1 (en) 2001-04-23
NO20003347L (no) 2000-08-28
UY25330A1 (es) 2000-12-29
US6472371B1 (en) 2002-10-29
UY25574A1 (es) 1999-09-27
KR20010024818A (ko) 2001-03-26
CA2316919A1 (en) 1999-07-15
TNSN98238A1 (fr) 2005-03-15

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