OA07044A - Nouveaux dérivés solubles N2 substitués de la diamino-2,4-benzyl-5-pyrimidines, leur procédé de préparation et médicaments les contenant. - Google Patents

Nouveaux dérivés solubles N2 substitués de la diamino-2,4-benzyl-5-pyrimidines, leur procédé de préparation et médicaments les contenant.

Info

Publication number
OA07044A
OA07044A OA57639A OA57639A OA07044A OA 07044 A OA07044 A OA 07044A OA 57639 A OA57639 A OA 57639A OA 57639 A OA57639 A OA 57639A OA 07044 A OA07044 A OA 07044A
Authority
OA
OAPI
Prior art keywords
diamino
substituted derivatives
pyrimidines
benzyl
preparation process
Prior art date
Application number
OA57639A
Other languages
English (en)
French (fr)
Inventor
Claude Laruelle
Original Assignee
Panmedica Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Panmedica Sa filed Critical Panmedica Sa
Publication of OA07044A publication Critical patent/OA07044A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
OA57639A 1981-03-20 1982-03-19 Nouveaux dérivés solubles N2 substitués de la diamino-2,4-benzyl-5-pyrimidines, leur procédé de préparation et médicaments les contenant. OA07044A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8105592A FR2502152A1 (fr) 1981-03-20 1981-03-20 Nouveaux derives solubles n2 substitues de la diamino-2,4-benzyl-5-pyrimidines, leur procede de preparation et medicaments les contenant

Publications (1)

Publication Number Publication Date
OA07044A true OA07044A (fr) 1983-12-31

Family

ID=9256463

Family Applications (1)

Application Number Title Priority Date Filing Date
OA57639A OA07044A (fr) 1981-03-20 1982-03-19 Nouveaux dérivés solubles N2 substitués de la diamino-2,4-benzyl-5-pyrimidines, leur procédé de préparation et médicaments les contenant.

Country Status (13)

Country Link
US (1) US4415574A (xx)
EP (1) EP0061397B1 (xx)
JP (1) JPS57169472A (xx)
AT (1) ATE17483T1 (xx)
AU (1) AU555274B2 (xx)
CA (1) CA1180015A (xx)
DE (2) DE61397T1 (xx)
ES (1) ES510618A0 (xx)
FR (1) FR2502152A1 (xx)
GR (1) GR75938B (xx)
MA (1) MA19413A1 (xx)
OA (1) OA07044A (xx)
ZA (1) ZA821785B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5707996A (en) * 1995-11-06 1998-01-13 Macleod Pharmaceuticals, Inc. Pharmaceutical solution and methods for preparation thereof
EP1438053B1 (de) * 2001-10-17 2008-09-10 Boehringer Ingelheim Pharma GmbH & Co.KG Pyrimidinderivate, arzneimittel enthaltend diese verbindungen, deren verwendung und verfahren zu ihrer herstellung
CN1930135B (zh) * 2004-03-05 2011-12-28 弗·哈夫曼-拉罗切有限公司 作为p2x3和p2x2/3拮抗剂的二氨基嘧啶
JP4850913B2 (ja) * 2005-09-01 2012-01-11 エフ.ホフマン−ラ ロシュ アーゲー P2x3及びp2x2/3調節因子としてのジアミノピリジン
BRPI0615613A2 (pt) * 2005-09-01 2009-05-19 Hoffmann La Roche diaminopirimidinas como moduladores de p2x3 e p3x2/3
JP4850911B2 (ja) * 2005-09-01 2012-01-11 エフ.ホフマン−ラ ロシュ アーゲー P2x3およびp2x2/3モジュレーターとしてのジアミノピリミジン
JP6788524B2 (ja) * 2017-02-28 2020-11-25 ダイコク電機株式会社 遊技用装置及び遊技場システム

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1407971A (en) * 1971-04-16 1975-10-01 Wellcome Found 2,4-diamino -4-3,4,5-triethoxybenzyl pyrimidine and methods of preparation therefor
FR2358148A1 (fr) * 1976-07-12 1978-02-10 Dick Pr Derives de 2,4-diaminopyrimidines et leur mise en solution en association avec des sulfamides
FR2397407A2 (fr) * 1977-07-11 1979-02-09 Dick Pierre Derives de 2,4-diamino pyrimidines et leur mise en solution en association avec des sulfamides

Also Published As

Publication number Publication date
GR75938B (xx) 1984-08-02
EP0061397A1 (fr) 1982-09-29
FR2502152B1 (xx) 1984-01-20
ES8302669A1 (es) 1983-02-01
ES510618A0 (es) 1983-02-01
ATE17483T1 (de) 1986-02-15
JPS57169472A (en) 1982-10-19
EP0061397B1 (fr) 1986-01-15
CA1180015A (en) 1984-12-27
AU8172882A (en) 1982-09-23
FR2502152A1 (fr) 1982-09-24
DE61397T1 (de) 1983-10-13
JPH0340026B2 (xx) 1991-06-17
AU555274B2 (en) 1986-09-18
US4415574A (en) 1983-11-15
DE3268481D1 (en) 1986-02-27
MA19413A1 (fr) 1982-10-01
ZA821785B (en) 1983-02-23

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