NZ592382A - Thioamide compounds, method of making and method of using thereof - Google Patents

Thioamide compounds, method of making and method of using thereof

Info

Publication number
NZ592382A
NZ592382A NZ592382A NZ59238209A NZ592382A NZ 592382 A NZ592382 A NZ 592382A NZ 592382 A NZ592382 A NZ 592382A NZ 59238209 A NZ59238209 A NZ 59238209A NZ 592382 A NZ592382 A NZ 592382A
Authority
NZ
New Zealand
Prior art keywords
compounds
thiocarbamoyl
ethyl
methyl
making
Prior art date
Application number
NZ592382A
Other languages
English (en)
Inventor
Hir De Fallois Loic Patrick Le
Hyoung Ik Lee
Philip Reid Timmons
Original Assignee
Merial Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Ltd filed Critical Merial Ltd
Publication of NZ592382A publication Critical patent/NZ592382A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/16—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C07D249/18—Benzotriazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4192—1,2,3-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
NZ592382A 2008-10-21 2009-10-20 Thioamide compounds, method of making and method of using thereof NZ592382A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10711408P 2008-10-21 2008-10-21
PCT/US2009/061337 WO2010048191A1 (en) 2008-10-21 2009-10-20 Thioamide compounds, method of making and method of using thereof

Publications (1)

Publication Number Publication Date
NZ592382A true NZ592382A (en) 2013-03-28

Family

ID=41404569

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ592382A NZ592382A (en) 2008-10-21 2009-10-20 Thioamide compounds, method of making and method of using thereof

Country Status (15)

Country Link
US (2) US7964621B2 (enExample)
EP (1) EP2358687B9 (enExample)
JP (1) JP5614853B2 (enExample)
KR (2) KR101782311B1 (enExample)
CN (1) CN102239151B (enExample)
AU (1) AU2009307736B2 (enExample)
BR (1) BRPI0920145B8 (enExample)
CA (1) CA2741186C (enExample)
CL (1) CL2011000917A1 (enExample)
EA (1) EA026649B1 (enExample)
ES (1) ES2393965T3 (enExample)
MX (1) MX2011004217A (enExample)
NZ (1) NZ592382A (enExample)
WO (1) WO2010048191A1 (enExample)
ZA (1) ZA201103033B (enExample)

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NZ716598A (en) 2012-11-20 2017-02-24 Merial Inc Anthelmintic compounds and compositions and method of using thereof
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JP6682719B2 (ja) 2014-04-17 2020-04-15 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 寄生生物から動物を保護するためのマロノニトリル化合物の使用
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BR112019009977A2 (pt) 2016-11-16 2019-08-27 Boehringer Ingelheim Animal Health Usa Inc compostos depsipeptídicos anti-helmínticos
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MX2021000293A (es) 2018-07-09 2021-07-15 Boehringer Ingelheim Animal Health Usa Inc Compuestos heterociclicos antihelminticos.
US11773066B2 (en) 2018-11-20 2023-10-03 Boehringer Ingelheim Animal Health USA Inc. Indazolylcyanoethylamino compound, compositions of same, method of making, and methods of using thereof
KR102281492B1 (ko) * 2018-12-24 2021-07-26 동인당제약 주식회사 세벨라머 함유 경구투여용 현탁제 조성물 및 그 제조방법
KR20220002890A (ko) 2019-03-19 2022-01-07 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 아자-벤조티오펜 및 아자-벤조푸란 화합물
BR112022024156A2 (pt) 2020-05-29 2023-02-14 Boehringer Ingelheim Animal Health Usa Inc Compostos heterocílicos antelmínticos
CN111781291A (zh) * 2020-06-23 2020-10-16 广西壮族自治区水产科学研究院 一种水中13种大环内酯类抗生素的高分辨质谱检测方法
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US12258193B2 (en) 2022-02-17 2025-03-25 Boehringer Ingelheim Vetmedica Gmbh Method and system for providing a fluid product mailer
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Also Published As

Publication number Publication date
ES2393965T9 (es) 2013-07-19
KR101782308B1 (ko) 2017-09-27
EA026649B1 (ru) 2017-05-31
ES2393965T3 (es) 2013-01-03
CA2741186A1 (en) 2010-04-29
KR101782311B1 (ko) 2017-09-27
BRPI0920145A2 (pt) 2017-06-06
CL2011000917A1 (es) 2011-09-16
EP2358687B9 (en) 2013-04-17
US7964621B2 (en) 2011-06-21
EP2358687A1 (en) 2011-08-24
WO2010048191A1 (en) 2010-04-29
EA201100666A1 (ru) 2011-12-30
JP2012506441A (ja) 2012-03-15
AU2009307736B2 (en) 2015-02-05
BRPI0920145B8 (pt) 2021-05-25
US20110190231A1 (en) 2011-08-04
EP2358687B1 (en) 2012-09-19
US20100130565A1 (en) 2010-05-27
JP5614853B2 (ja) 2014-10-29
ZA201103033B (en) 2012-02-29
MX2011004217A (es) 2011-06-20
CA2741186C (en) 2016-07-19
BRPI0920145B1 (pt) 2021-03-30
AU2009307736A1 (en) 2010-04-29
US8314146B2 (en) 2012-11-20
KR20170003704A (ko) 2017-01-09
KR20110071140A (ko) 2011-06-28
CN102239151A (zh) 2011-11-09
CN102239151B (zh) 2014-07-02

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