NZ548091A - Transdermal delivery system of hormones without penetration enhancers - Google Patents
Transdermal delivery system of hormones without penetration enhancersInfo
- Publication number
- NZ548091A NZ548091A NZ548091A NZ54809104A NZ548091A NZ 548091 A NZ548091 A NZ 548091A NZ 548091 A NZ548091 A NZ 548091A NZ 54809104 A NZ54809104 A NZ 54809104A NZ 548091 A NZ548091 A NZ 548091A
- Authority
- NZ
- New Zealand
- Prior art keywords
- drug
- containing layer
- gestodene
- kit
- weight
- Prior art date
Links
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Classifications
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- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
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- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
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- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
- A61K9/7061—Polyacrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7076—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising ingredients of undetermined constitution or reaction products thereof, e.g. rosin or other plant resins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
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- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Botany (AREA)
- Reproductive Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Organic Chemistry (AREA)
- Gynecology & Obstetrics (AREA)
- Inorganic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US52871803P | 2003-12-12 | 2003-12-12 | |
| EP03078881 | 2003-12-12 | ||
| PCT/IB2004/052752 WO2005058287A2 (en) | 2003-12-12 | 2004-12-10 | Transdermal delivery system of hormones without penetration enhancers |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ548091A true NZ548091A (en) | 2009-12-24 |
Family
ID=34702342
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ548091A NZ548091A (en) | 2003-12-12 | 2004-12-10 | Transdermal delivery system of hormones without penetration enhancers |
Country Status (15)
| Country | Link |
|---|---|
| JP (1) | JP4965263B2 (es) |
| KR (1) | KR101168449B1 (es) |
| CN (1) | CN1913878B (es) |
| AU (1) | AU2004298930B2 (es) |
| BR (1) | BRPI0417530B8 (es) |
| CA (1) | CA2549916C (es) |
| CU (1) | CU23868B1 (es) |
| EA (1) | EA011160B1 (es) |
| EC (1) | ECSP066694A (es) |
| IL (1) | IL176112A (es) |
| MX (1) | MXPA06006682A (es) |
| NO (1) | NO341989B1 (es) |
| NZ (1) | NZ548091A (es) |
| WO (1) | WO2005058287A2 (es) |
| ZA (1) | ZA200605713B (es) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1594483B1 (de) | 2003-02-21 | 2006-07-19 | Schering AG | Uv-stabiles transdermales pflaster |
| US8962013B2 (en) | 2005-05-02 | 2015-02-24 | Bayer Intellectual Property Gmbh | Multi-layered transdermal system with triazine UV absorber |
| DE102005050729A1 (de) * | 2005-10-19 | 2007-04-26 | Schering Ag | Verfahren zur präventiven bedarfsweisen hormonalen Kontrazeption |
| FR2900048B1 (fr) * | 2006-04-21 | 2012-11-16 | Oreal | Compositions comprenant un derive diphenyl-methane hydroxyle |
| DE102010040299A1 (de) | 2010-09-06 | 2012-03-08 | Bayer Schering Pharma Aktiengesellschaft | Transdermale therapeutische Systeme mit kristallisationsinhibierender Schutzfolie (Release Liner) |
| AU2015203180B2 (en) * | 2010-09-06 | 2016-06-30 | Bayer Intellectual Property Gmbh | Transdermal therapeutic systems with crystallization-inhibiting protective film (release liner) |
| EP2613772B1 (en) | 2010-09-06 | 2016-12-14 | Bayer Intellectual Property GmbH | Low-dose transdermal patches with high drug release |
| CA2861324A1 (en) * | 2012-01-27 | 2013-08-01 | Agile Therapeutics, Inc. | Transdermal hormone delivery |
| CN107995864A (zh) * | 2015-05-18 | 2018-05-04 | 敏捷治疗公司 | 避孕组合物及提高效能和调节副作用的方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0370220B1 (de) * | 1988-10-27 | 1996-01-10 | Schering Aktiengesellschaft | Mittel zur transdermalen Applikation enthaltend Gestoden |
| EP0555360A1 (en) * | 1990-10-29 | 1993-08-18 | Alza Corporation | Transdermal contraceptive formulations, methods and devices |
| US5512292A (en) * | 1990-10-29 | 1996-04-30 | Alza Corporation | Transdermal contraceptive formulations methods and devices |
| DE4329242A1 (de) * | 1993-08-26 | 1995-03-02 | Schering Ag | Mittel zur transdermalen Applikation enthaltend Gestodenester |
| DE4405898A1 (de) * | 1994-02-18 | 1995-08-24 | Schering Ag | Transdermale therapeutische Systeme enthaltend Sexualsteroide |
| WO1996015776A1 (fr) * | 1994-11-18 | 1996-05-30 | Hisamitsu Pharmaceutical Co., Inc. | Timbre absorbable par voie percutanee |
| CA2222133C (en) * | 1995-06-07 | 2002-12-24 | Cygnus, Inc. | Transdermal patch and method for administering 17-deacetyl norgestimate alone or in combination with an estrogen |
| JP4346696B2 (ja) * | 1996-05-28 | 2009-10-21 | 久光製薬株式会社 | 経皮治療用装置 |
| JP4167750B2 (ja) * | 1997-04-16 | 2008-10-22 | 久光製薬株式会社 | 経皮吸収用基剤及び該基剤を含有する経皮吸収製剤 |
| JP4399044B2 (ja) * | 1998-10-14 | 2010-01-13 | 久光製薬株式会社 | 吸収促進剤及び該吸収促進剤を有してなる経皮吸収製剤 |
| DE19906152B4 (de) * | 1999-02-10 | 2005-02-10 | Jenapharm Gmbh & Co. Kg | Wirkstoffhaltige Laminate für Transdermalsysteme |
| EP1197212A4 (en) * | 1999-07-01 | 2004-06-02 | Hisamitsu Pharmaceutical Co | ADHESIVE COMPOSITION FOR PERCUTANE ABSORPTION |
| DE10053375C1 (de) * | 2000-10-27 | 2002-01-24 | Lohmann Therapie Syst Lts | Transdermale therapeutische Systeme mit lichtempfindlichen Wirkstoffen |
| US20020106402A1 (en) * | 2000-12-05 | 2002-08-08 | Hartwig Rod Lawson | Crystallization inhibition of drugs in transdermal drug delivery systems and methods of use |
-
2004
- 2004-12-10 MX MXPA06006682A patent/MXPA06006682A/es active IP Right Grant
- 2004-12-10 AU AU2004298930A patent/AU2004298930B2/en not_active Ceased
- 2004-12-10 KR KR1020067013923A patent/KR101168449B1/ko active IP Right Grant
- 2004-12-10 BR BRPI0417530A patent/BRPI0417530B8/pt not_active IP Right Cessation
- 2004-12-10 JP JP2006543709A patent/JP4965263B2/ja active Active
- 2004-12-10 CA CA2549916A patent/CA2549916C/en not_active Expired - Fee Related
- 2004-12-10 WO PCT/IB2004/052752 patent/WO2005058287A2/en active Application Filing
- 2004-12-10 NZ NZ548091A patent/NZ548091A/en not_active IP Right Cessation
- 2004-12-10 CN CN2004800413210A patent/CN1913878B/zh active Active
- 2004-12-10 EA EA200601089A patent/EA011160B1/ru not_active IP Right Cessation
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2006
- 2006-06-05 IL IL176112A patent/IL176112A/en active IP Right Grant
- 2006-06-06 NO NO20062594A patent/NO341989B1/no not_active IP Right Cessation
- 2006-07-11 EC EC2006006694A patent/ECSP066694A/es unknown
- 2006-07-11 ZA ZA2006/05713A patent/ZA200605713B/en unknown
-
2010
- 2010-07-05 CU CU20100143A patent/CU23868B1/es active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| EA200601089A1 (ru) | 2006-12-29 |
| MXPA06006682A (es) | 2006-08-11 |
| WO2005058287A3 (en) | 2006-03-02 |
| JP2007513938A (ja) | 2007-05-31 |
| BRPI0417530B8 (pt) | 2021-05-25 |
| ZA200605713B (en) | 2008-01-08 |
| ECSP066694A (es) | 2006-10-31 |
| BRPI0417530A (pt) | 2007-03-13 |
| NO20062594L (no) | 2006-07-10 |
| IL176112A (en) | 2011-02-28 |
| CU23868B1 (es) | 2013-03-27 |
| CU20100143A7 (es) | 2011-10-31 |
| AU2004298930A1 (en) | 2005-06-30 |
| AU2004298930B2 (en) | 2009-11-26 |
| WO2005058287A2 (en) | 2005-06-30 |
| JP4965263B2 (ja) | 2012-07-04 |
| EA011160B1 (ru) | 2009-02-27 |
| CA2549916A1 (en) | 2005-06-30 |
| IL176112A0 (en) | 2006-10-05 |
| BRPI0417530B1 (pt) | 2018-01-23 |
| CA2549916C (en) | 2013-09-17 |
| CN1913878B (zh) | 2010-05-26 |
| NO341989B1 (no) | 2018-03-12 |
| KR20060128910A (ko) | 2006-12-14 |
| CN1913878A (zh) | 2007-02-14 |
| KR101168449B1 (ko) | 2012-07-25 |
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