NZ545884A - Treating and/or preventing urinary incontinence using prodrugs of GABA analogs - Google Patents

Treating and/or preventing urinary incontinence using prodrugs of GABA analogs

Info

Publication number
NZ545884A
NZ545884A NZ545884A NZ54588404A NZ545884A NZ 545884 A NZ545884 A NZ 545884A NZ 545884 A NZ545884 A NZ 545884A NZ 54588404 A NZ54588404 A NZ 54588404A NZ 545884 A NZ545884 A NZ 545884A
Authority
NZ
New Zealand
Prior art keywords
substituted
butyl
phenethyl
dioxan
dioxolan
Prior art date
Application number
NZ545884A
Other languages
English (en)
Inventor
Ronald W Barrett
Original Assignee
Xenoport Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Xenoport Inc filed Critical Xenoport Inc
Publication of NZ545884A publication Critical patent/NZ545884A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NZ545884A 2003-09-11 2004-09-13 Treating and/or preventing urinary incontinence using prodrugs of GABA analogs NZ545884A (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US50258503P 2003-09-11 2003-09-11
US50521003P 2003-09-22 2003-09-22
US51228803P 2003-10-17 2003-10-17
US53874804P 2004-01-22 2004-01-22
PCT/US2004/029944 WO2005025562A1 (en) 2003-09-11 2004-09-13 Treating and/or preventing urinary incontinence using prodrugs of gaba analogs

Publications (1)

Publication Number Publication Date
NZ545884A true NZ545884A (en) 2010-01-29

Family

ID=34317683

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ545884A NZ545884A (en) 2003-09-11 2004-09-13 Treating and/or preventing urinary incontinence using prodrugs of GABA analogs

Country Status (11)

Country Link
US (2) US7700652B2 (enExample)
EP (1) EP1670451A4 (enExample)
JP (1) JP2007505149A (enExample)
KR (1) KR20060119971A (enExample)
AU (1) AU2004272111A1 (enExample)
CA (1) CA2537837A1 (enExample)
IL (1) IL174409A0 (enExample)
MX (1) MXPA06002731A (enExample)
NO (1) NO20061625L (enExample)
NZ (1) NZ545884A (enExample)
WO (1) WO2005025562A1 (enExample)

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Also Published As

Publication number Publication date
NO20061625L (no) 2006-06-12
AU2004272111A1 (en) 2005-03-24
CA2537837A1 (en) 2005-03-24
EP1670451A1 (en) 2006-06-21
JP2007505149A (ja) 2007-03-08
MXPA06002731A (es) 2006-06-05
WO2005025562A1 (en) 2005-03-24
KR20060119971A (ko) 2006-11-24
IL174409A0 (en) 2011-08-01
US7700652B2 (en) 2010-04-20
EP1670451A4 (en) 2009-10-21
US20050090550A1 (en) 2005-04-28
US20100166825A1 (en) 2010-07-01

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