NZ182779A - C-(2-oxazolin-2-yl or 2-thiazolin-2-yl)-aminoindazoles - Google Patents

C-(2-oxazolin-2-yl or 2-thiazolin-2-yl)-aminoindazoles

Info

Publication number
NZ182779A
NZ182779A NZ182779A NZ18277976A NZ182779A NZ 182779 A NZ182779 A NZ 182779A NZ 182779 A NZ182779 A NZ 182779A NZ 18277976 A NZ18277976 A NZ 18277976A NZ 182779 A NZ182779 A NZ 182779A
Authority
NZ
New Zealand
Prior art keywords
aminoindazoles
thiazolin
oxazolin
Prior art date
Application number
NZ182779A
Other languages
English (en)
Inventor
P Neumann
Original Assignee
Sandoz Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1571675A external-priority patent/CH605934A5/de
Priority claimed from CH1664575A external-priority patent/CH605858A5/de
Application filed by Sandoz Ltd filed Critical Sandoz Ltd
Publication of NZ182779A publication Critical patent/NZ182779A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NZ182779A 1975-12-03 1976-12-01 C-(2-oxazolin-2-yl or 2-thiazolin-2-yl)-aminoindazoles NZ182779A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH1571675A CH605934A5 (en) 1975-12-03 1975-12-03 Myotonolytic oxazolinyl- and thiazolinyl-amino-indazole derivs.
CH1664575A CH605858A5 (en) 1975-12-22 1975-12-22 Myotonolytic oxazolinyl- and thiazolinyl-amino-indazole derivs.
CH927976 1976-07-20
CH931276 1976-07-21

Publications (1)

Publication Number Publication Date
NZ182779A true NZ182779A (en) 1979-08-31

Family

ID=27429211

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ182779A NZ182779A (en) 1975-12-03 1976-12-01 C-(2-oxazolin-2-yl or 2-thiazolin-2-yl)-aminoindazoles

Country Status (20)

Country Link
US (1) US4086353A (enExample)
JP (1) JPS5268177A (enExample)
AU (1) AU510820B2 (enExample)
BE (1) BE848962A (enExample)
CA (1) CA1082714A (enExample)
DE (1) DE2653005A1 (enExample)
DK (1) DK528976A (enExample)
ES (1) ES453861A1 (enExample)
FI (1) FI763385A7 (enExample)
FR (1) FR2333504A1 (enExample)
GB (1) GB1564327A (enExample)
IE (1) IE44316B1 (enExample)
IL (1) IL51028A (enExample)
NL (1) NL7613317A (enExample)
NO (1) NO764039L (enExample)
NZ (1) NZ182779A (enExample)
PH (1) PH12642A (enExample)
PT (1) PT65918B (enExample)
SE (1) SE424553B (enExample)
YU (1) YU293876A (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4436913A (en) * 1980-09-05 1984-03-13 Siegfried Aktiengesellschaft 1H- and 2H- indazole derivatives
CZ2004359A3 (cs) * 2001-09-26 2004-09-15 Pharmacia Italia S.P.A. Aminoindazolové deriváty aktivní jako inhibitory kinázy, způsob jejich přípravy a farmaceutické prostředky obsahující tyto deriváty
SE0402763D0 (sv) * 2004-11-11 2004-11-11 Astrazeneca Ab Nitro indazole derivatives
SE0402762D0 (sv) * 2004-11-11 2004-11-11 Astrazeneca Ab Indazole sulphonamide derivatives
CA2755268C (en) * 2005-11-15 2013-12-31 Array Biopharma, Inc. Erbb inhibitors
JP2009520825A (ja) * 2005-12-20 2009-05-28 武田薬品工業株式会社 グルコキナーゼ活性剤
JP5323834B2 (ja) * 2007-08-17 2013-10-23 エルジー・ライフ・サイエンシーズ・リミテッド 細胞壊死阻害剤としてのインドール化合物
RU2460525C2 (ru) * 2008-01-04 2012-09-10 Эл Джи Лайф Сайенсиз Лтд. Производные индола и индазола, обладающие консервирующим действием по отношению к клеткам, тканям и органам
WO2013077579A1 (ko) * 2011-11-25 2013-05-30 가톨릭대학교 산학협력단 안과 질환의 예방 및 치료용 약학 조성물
WO2016115272A1 (en) 2015-01-13 2016-07-21 Vanderbilt University Benzothiazole and benzisothiazole-substituted compounds as mglur4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
US9980945B2 (en) 2015-01-13 2018-05-29 Vanderbilt University Benzoisoxazole-substituted compounds as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
US10526323B2 (en) 2015-01-30 2020-01-07 Vanderbilt University Indazole and azaindazole substituted compounds as mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3759903A (en) * 1971-07-28 1973-09-18 Squibb & Sons Inc Thiazolinyl and thiazinyl derivatives of indazoles

Also Published As

Publication number Publication date
US4086353A (en) 1978-04-25
AU510820B2 (en) 1980-07-17
IL51028A (en) 1980-06-30
IL51028A0 (en) 1977-02-28
GB1564327A (en) 1980-04-10
SE424553B (sv) 1982-07-26
IE44316L (en) 1977-06-03
PH12642A (en) 1979-07-11
AU2025276A (en) 1978-06-08
JPS5268177A (en) 1977-06-06
PT65918A (fr) 1977-01-01
NL7613317A (nl) 1977-06-07
FI763385A7 (enExample) 1977-06-04
NO764039L (enExample) 1977-06-06
IE44316B1 (en) 1981-10-21
BE848962A (fr) 1977-06-01
CA1082714A (en) 1980-07-29
YU293876A (en) 1982-05-31
FR2333504A1 (fr) 1977-07-01
ES453861A1 (es) 1978-03-01
FR2333504B1 (enExample) 1980-08-29
PT65918B (fr) 1978-07-05
DK528976A (da) 1977-06-04
SE7613195L (sv) 1977-06-04
DE2653005A1 (de) 1977-06-08

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