NO974233L - Aminofenolderivater - Google Patents
AminofenolderivaterInfo
- Publication number
- NO974233L NO974233L NO974233A NO974233A NO974233L NO 974233 L NO974233 L NO 974233L NO 974233 A NO974233 A NO 974233A NO 974233 A NO974233 A NO 974233A NO 974233 L NO974233 L NO 974233L
- Authority
- NO
- Norway
- Prior art keywords
- receptor
- cck
- salts
- gastrin receptor
- gastrin
- Prior art date
Links
- 108010089448 Cholecystokinin B Receptor Proteins 0.000 abstract 3
- 102000052874 Gastrin receptors Human genes 0.000 abstract 3
- 108010089335 Cholecystokinin A Receptor Proteins 0.000 abstract 2
- 102100034927 Cholecystokinin receptor type A Human genes 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- CDAWCLOXVUBKRW-UHFFFAOYSA-N 2-aminophenol Chemical class NC1=CC=CC=C1O CDAWCLOXVUBKRW-UHFFFAOYSA-N 0.000 abstract 1
- 208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
- 208000008469 Peptic Ulcer Diseases 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 125000005242 carbamoyl alkyl group Chemical group 0.000 abstract 1
- 208000015114 central nervous system disease Diseases 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 230000003287 optical effect Effects 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 239000002464 receptor antagonist Substances 0.000 abstract 1
- 229940044551 receptor antagonist Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01K—ANIMAL HUSBANDRY; AVICULTURE; APICULTURE; PISCICULTURE; FISHING; REARING OR BREEDING ANIMALS, NOT OTHERWISE PROVIDED FOR; NEW BREEDS OF ANIMALS
- A01K31/00—Housing birds
- A01K31/14—Nest-boxes, e.g. for singing birds or the like
- A01K31/16—Laying nests for poultry; Egg collecting
- A01K31/17—Laying batteries including auxiliary features, e.g. feeding, watering, demanuring, heating, ventilation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/04—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms
- C07C275/06—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton
- C07C275/16—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton being further substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/01—Sulfonic acids
- C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
- C07C309/19—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Environmental Sciences (AREA)
- Birds (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Zoology (AREA)
- Animal Husbandry (AREA)
- Biodiversity & Conservation Biology (AREA)
- Biomedical Technology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
Abstract
Aminofenolderivater som er representert ved følgende formel (1): R2 R^¿S-CO-C-.'iHCONl!-R' I X-.A-CO-R^ (1) hvor X er 0 eller S, A er alkylen. R' er fenyl, etc, R^ og R^ er H eller alkyl, R" er substituert karbamoylalkyl, etc, R^ er substituert amino etc, deres salter, og optiske isomerer av derivatene og saltene. Det er også beskrevet gastrinreseptor- antagonister, cholecystokininreseptor-antagonister, og medisiner for fordøyelses- sykdommer. Forbindelsene har sterk bindingsinhibering mot gastrinreseptor eller CCK-A-reseptor, og de har også høyere selektivitet overfor en hvilken som helst av gruppene av CCK-A-reseptor eller gastrinreseptor, og derfor er forbindelsene nyttige til å forebygge og behandle gastrointestinale sykdommer, innbefattende peptiske sår, såvel som sykdommer i sentralnervesystemet.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP5475295 | 1995-03-14 | ||
| JP1763496 | 1996-02-02 | ||
| PCT/JP1996/000611 WO1996028416A1 (fr) | 1995-03-14 | 1996-03-12 | Derives d'aminophenol |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO974233D0 NO974233D0 (no) | 1997-09-12 |
| NO974233L true NO974233L (no) | 1997-11-12 |
Family
ID=26354192
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO974233A NO974233L (no) | 1995-03-14 | 1997-09-12 | Aminofenolderivater |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US5919824A (no) |
| EP (1) | EP0985660A1 (no) |
| JP (1) | JP3688714B2 (no) |
| KR (1) | KR19980702952A (no) |
| AU (1) | AU4891396A (no) |
| CA (1) | CA2214569A1 (no) |
| NO (1) | NO974233L (no) |
| WO (1) | WO1996028416A1 (no) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2445477A1 (en) * | 2001-05-11 | 2002-11-21 | Yamanouchi Pharmaceutical Co., Ltd. | Antitumor agents |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2533210A1 (fr) * | 1982-09-17 | 1984-03-23 | Lyon I Universite Claude | Edulcorants de synthese |
| EP0514442B1 (fr) * | 1990-02-09 | 1994-04-27 | Aventis Pharma S.A. | N-phenyl n-acetamido glycinamides, leur preparation et les medicaments les contenant |
| FR2695643B1 (fr) * | 1992-09-11 | 1994-11-25 | Rhone Poulenc Rorer Sa | Dérivés d'uréido-acétamide, leur préparation et les médicaments les contenant. |
-
1996
- 1996-03-12 AU AU48913/96A patent/AU4891396A/en not_active Abandoned
- 1996-03-12 CA CA002214569A patent/CA2214569A1/en not_active Abandoned
- 1996-03-12 KR KR1019970706360A patent/KR19980702952A/ko not_active Application Discontinuation
- 1996-03-12 EP EP96905068A patent/EP0985660A1/en not_active Withdrawn
- 1996-03-12 US US08/894,799 patent/US5919824A/en not_active Expired - Fee Related
- 1996-03-12 JP JP52746696A patent/JP3688714B2/ja not_active Expired - Fee Related
- 1996-03-12 WO PCT/JP1996/000611 patent/WO1996028416A1/ja not_active Application Discontinuation
-
1997
- 1997-09-12 NO NO974233A patent/NO974233L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO1996028416A1 (fr) | 1996-09-19 |
| JP3688714B2 (ja) | 2005-08-31 |
| CA2214569A1 (en) | 1996-09-19 |
| KR19980702952A (ko) | 1998-09-05 |
| EP0985660A1 (en) | 2000-03-15 |
| US5919824A (en) | 1999-07-06 |
| NO974233D0 (no) | 1997-09-12 |
| AU4891396A (en) | 1996-10-02 |
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