NO974125L - N-benzylazoliumderivater - Google Patents

N-benzylazoliumderivater

Info

Publication number
NO974125L
NO974125L NO974125A NO974125A NO974125L NO 974125 L NO974125 L NO 974125L NO 974125 A NO974125 A NO 974125A NO 974125 A NO974125 A NO 974125A NO 974125 L NO974125 L NO 974125L
Authority
NO
Norway
Prior art keywords
general formula
group
hydrogen
formula
independently
Prior art date
Application number
NO974125A
Other languages
English (en)
Norwegian (no)
Other versions
NO974125D0 (no
Inventor
Ichihara Shigeyasu
Sawada Daisuke
Murasaki Chikako
Shimma Nobou
Ohga Noriko
Shirai Michio
Ohwasa Jun
Umeda Isao
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO974125D0 publication Critical patent/NO974125D0/no
Publication of NO974125L publication Critical patent/NO974125L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/08—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing alicyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO974125A 1996-09-09 1997-09-08 N-benzylazoliumderivater NO974125L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP96114390 1996-09-09
EP97114246 1997-08-18

Publications (2)

Publication Number Publication Date
NO974125D0 NO974125D0 (no) 1997-09-08
NO974125L true NO974125L (no) 1998-03-10

Family

ID=26142161

Family Applications (1)

Application Number Title Priority Date Filing Date
NO974125A NO974125L (no) 1996-09-09 1997-09-08 N-benzylazoliumderivater

Country Status (12)

Country Link
US (2) US5900486A (ja)
JP (1) JP2965532B2 (ja)
KR (1) KR100252433B1 (ja)
CN (1) CN1182739A (ja)
AU (1) AU3685097A (ja)
CA (1) CA2214669A1 (ja)
CZ (1) CZ282897A3 (ja)
HU (1) HUP9701479A3 (ja)
IL (1) IL121691A0 (ja)
MA (1) MA26440A1 (ja)
NO (1) NO974125L (ja)
NZ (1) NZ328607A (ja)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2931399A (en) 1998-03-06 1999-09-20 F. Hoffmann-La Roche Ag 3-(4-(4-cyanophenyl)thiazol-2-y))-1-(1h-1,2,4-triazol-1-yl) -butan-2-ol derivatives having antifungal activity
WO2000030655A1 (en) * 1998-11-20 2000-06-02 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
US6319933B1 (en) 2000-04-17 2001-11-20 Basilea Pharmaceutica Ag Azole derivatives
AU2002351388A1 (en) * 2001-12-14 2003-06-30 The University Of Wyoming Methods and compositions for controlled release of drugs
TW200606129A (en) * 2004-07-26 2006-02-16 Chugai Pharmaceutical Co Ltd Novel cyclohexane derivative, its prodrug, its salt and diabetic therapeutic agent containing the same
CN101391985B (zh) * 2007-09-18 2013-09-11 西南大学 具抗微生物活性的三唑鎓类化合物及制备方法和医药用途
AU2012272804B2 (en) * 2011-06-22 2017-07-06 Vyome Therapeutics Limited Conjugate-based antifungal and antibacterial prodrugs
CN104974143A (zh) * 2015-05-12 2015-10-14 深圳致君制药有限公司 一种季铵盐类化合物、其制备方法以及用途

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH468788A (de) * 1966-04-29 1969-02-28 Basf Ag Mischung zur Bekämpfung von Algen und Pilzen
US4017631A (en) * 1974-11-19 1977-04-12 Janssen Pharmaceutica N.V. Imidazolium salts
DE2531031C3 (de) * 1975-07-11 1978-03-16 Schuelke & Mayr Gmbh, 2000 Norderstedt 1 -Benzyl-3-alkyI-imidazoliumsalze
DE2643563A1 (de) * 1976-09-28 1978-03-30 Bayer Ag Alpha-(4-biphenylyl)-benzyl-azolium- salze, verfahren zu ihrer herstellung sowie ihre verwendung zur bekaempfung von mikroorganismen
DE2714290A1 (de) * 1977-03-31 1978-10-05 Bayer Ag Fungizide mittel
US4267179A (en) * 1978-06-23 1981-05-12 Janssen Pharmaceutica, N.V. Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
US4402957A (en) * 1979-04-04 1983-09-06 Janssen Pharmaceutica N.V. Heterocyclic derivatives of [4-(piperazin-1-ylphenyloxymethyl)-1,3-dioxolan-2-ylmethyl]-1H-imidazoles and 1H-1,2,4-triazoles
FR2486079A1 (fr) * 1980-07-07 1982-01-08 Rhone Poulenc Agrochimie Sels quaternaires d'alcoyl-1-imidazolium de l'acide phosphoreux ou ses monoesters, procedes pour les preparer et compositions fongicides les contenant
US4490530A (en) * 1981-01-14 1984-12-25 Janssen Pharmaceutica N.V. Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)-methyl-1H-imidazoles and 1H-1,2,4-triazoles
EP0069442B1 (en) * 1981-06-06 1985-02-20 Pfizer Limited Antifungal agents, processes for their preparation, and pharmaceutical compositions containing them
DE3217963A1 (de) * 1982-05-13 1983-11-17 Basf Ag, 6700 Ludwigshafen Dibenzofuranoxyalkyl-imidazoliumsalze, verfahren zu ihrer herstellung und ihre verwendung als mikrozide
US4861879A (en) * 1983-02-28 1989-08-29 Janssen Pharmaceutica N.V. [[4-[4-Phenyl-1-piperazinyl)phenoxymethyl]-1-3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles
DE3319845A1 (de) * 1983-06-01 1984-12-06 Basf Ag, 6700 Ludwigshafen Arylalkylimidazolium- und -triazoliumsalze, verfahren zu ihrer herstellung und ihre verwendung als mikrozide
US5128351A (en) * 1990-05-04 1992-07-07 American Cyanamid Company Bis-aryl amide and urea antagonists of platelet activating factor
WO1995019983A1 (en) * 1994-01-24 1995-07-27 Janssen Pharmaceutica N.V. Watersoluble azole antifungals
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions

Also Published As

Publication number Publication date
JP2965532B2 (ja) 1999-10-18
AU3685097A (en) 1998-03-12
HU9701479D0 (en) 1997-10-28
KR100252433B1 (ko) 2000-08-01
US5900486A (en) 1999-05-04
CN1182739A (zh) 1998-05-27
NZ328607A (en) 1999-08-30
CA2214669A1 (en) 1998-03-09
US5962686A (en) 1999-10-05
HUP9701479A3 (en) 2001-02-28
MA26440A1 (fr) 2004-12-20
CZ282897A3 (cs) 1998-06-17
JPH10114758A (ja) 1998-05-06
HUP9701479A2 (hu) 1999-02-01
IL121691A0 (en) 1998-02-22
NO974125D0 (no) 1997-09-08
KR19980024429A (ko) 1998-07-06

Similar Documents

Publication Publication Date Title
CA2396738A1 (en) Thiazole derivatives as active superoxide radical inhibitors
IL135537A0 (en) Substituted fused heterocyclic compounds
YU25299A (sh) Paraziticidni pirazoli
ES8708230A1 (es) Un procedimiento para preparar derivados de piridina
MX9800718A (es) Derivados de 2-(4-substituidos)-bencilamino-2-metil- propanamida.
MX9701685A (es) Nuevos derivados de bencimidazol que tienen la actividad de inhibicion de la fosfodiestearasa cgmp.
ATE271045T1 (de) Sauerstoffhaltige heterocyclische verbindungen
NO974125L (no) N-benzylazoliumderivater
AU629048B2 (en) N-(-4-(phenyl)-1,2-dihydro-3-quinolyl)-N'-(phenyl) urea derivatives and their use
HK1031867A1 (en) 2-phenoxyaniline derivatives
EP0829478A3 (en) N-Benzylimidazolium and N-benzyltriazolium derivatives, their preparation and their use as antifungal and antimycotic agents
NZ304438A (en) Substituted triazole derivatives and antifungal compositions
NZ296285A (en) Inhibiting physiological conditions associated with bradykinin using a benzothiophene such as raloxifene
ES2168062A1 (es) Composiciones para control de cucarachas
EP0795326A4 (ja)
EP0291247A3 (en) Novel cinnamoylamide derivatives
SG50820A1 (en) Novel thiouracil derivatives and metal surface- treating agent comprising thereof
NZ335975A (en) Heterocyclic substituted pyrrolidine amide derivatives useful in treating respiratory diseases
NO963307L (no) Karbamoylmetylureaderivater
TW334426B (en) Piperazine derivatives
ECSP972249A (es) Derivados de n-bencilazolio
EP0782988A4 (en) INDOL DERIVATIVES
IL126548A0 (en) Use of aspirochlorine or derivatives thereof as immunosuppressive agents
DE60009301D1 (en) Benzimidazolverbindungen
EP0878475A3 (en) 5-(4-Piperidinyl)dibenzothiazepine derivatives and 5-(4-piperidinyl)dibenzoxazepine derivatives, and antiarrhythmic agents

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application