NO924612L - Fremgangsmaate for fremstilling av 3-amino-2-aryl-kinuklidiner - Google Patents

Fremgangsmaate for fremstilling av 3-amino-2-aryl-kinuklidiner

Info

Publication number
NO924612L
NO924612L NO92924612A NO924612A NO924612L NO 924612 L NO924612 L NO 924612L NO 92924612 A NO92924612 A NO 92924612A NO 924612 A NO924612 A NO 924612A NO 924612 L NO924612 L NO 924612L
Authority
NO
Norway
Prior art keywords
pct
alkyl
compounds
date dec
furyl
Prior art date
Application number
NO92924612A
Other languages
English (en)
Norwegian (no)
Other versions
NO924612D0 (no
Inventor
Iii John A Lowe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO924612D0 publication Critical patent/NO924612D0/no
Publication of NO924612L publication Critical patent/NO924612L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO92924612A 1990-06-01 1992-11-30 Fremgangsmaate for fremstilling av 3-amino-2-aryl-kinuklidiner NO924612L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53252590A 1990-06-01 1990-06-01
PCT/US1991/002853 WO1991018899A1 (en) 1990-06-01 1991-04-25 3-amino-2-aryl quinuclidines, process for their preparation and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
NO924612D0 NO924612D0 (no) 1992-11-30
NO924612L true NO924612L (no) 1992-11-30

Family

ID=24122165

Family Applications (1)

Application Number Title Priority Date Filing Date
NO92924612A NO924612L (no) 1990-06-01 1992-11-30 Fremgangsmaate for fremstilling av 3-amino-2-aryl-kinuklidiner

Country Status (18)

Country Link
US (1) US5451586A (sv)
EP (1) EP0532527B1 (sv)
JP (1) JPH072740B2 (sv)
KR (1) KR930700499A (sv)
AT (1) ATE113947T1 (sv)
AU (1) AU648317B2 (sv)
CA (1) CA2084193C (sv)
DE (1) DE69105131T2 (sv)
DK (1) DK0532527T3 (sv)
ES (1) ES2063507T3 (sv)
FI (1) FI113654B (sv)
HU (1) HUT62891A (sv)
IE (1) IE911856A1 (sv)
IL (1) IL98259A0 (sv)
NO (1) NO924612L (sv)
PT (1) PT97771A (sv)
WO (1) WO1991018899A1 (sv)
ZA (1) ZA914134B (sv)

Families Citing this family (91)

* Cited by examiner, † Cited by third party
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US5750542A (en) * 1993-09-28 1998-05-12 Pfizer Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors
WO1992020661A1 (en) * 1991-05-22 1992-11-26 Merck & Co., Inc. N, n-diacylpiperazines
US5716965A (en) * 1991-05-22 1998-02-10 Pfizer Inc. Substituted 3-aminoquinuclidines
DK0587723T3 (da) * 1991-05-31 1996-04-01 Pfizer Quinuclidinderivater
UA39168C2 (uk) * 1991-06-20 2001-06-15 Пфайзер, Інк. Фторалкоксифенільні похідні піперидину або хінуклідину, що є антагоністами речовини p і фармацевтична композиція на їх основі
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ATE161821T1 (de) * 1991-11-12 1998-01-15 Pfizer Azyklische ethylendiaminderivate als 'substance p rezeptor' antagonisten
FR2688219B1 (fr) 1992-03-03 1994-07-08 Sanofi Elf Sels d'ammonium quaternaires de composes aromatiques amines, leur preparation et compositions pharmaceutiques les contenant.
CA2134964C (en) * 1992-05-18 1997-12-30 Manoj C. Desai Bridged aza-bicyclic derivatives as substance p antagonists
US5637699A (en) * 1992-06-29 1997-06-10 Merck & Co., Inc. Process for preparing morpholine tachykinin receptor antagonists
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US5387595A (en) * 1992-08-26 1995-02-07 Merck & Co., Inc. Alicyclic compounds as tachykinin receptor antagonists
US5837711A (en) * 1992-10-28 1998-11-17 Pfizer Inc. Substituted quinuclidines as substance P antagonists
DE69307340T2 (de) * 1992-11-12 1997-04-24 Pfizer Chinuclidin derivat als substanz p antagonist
US5344830A (en) * 1992-12-10 1994-09-06 Merck & Co., Inc. N,N-diacylpiperazine tachykinin antagonists
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TW385308B (en) * 1994-03-04 2000-03-21 Merck & Co Inc Prodrugs of morpholine tachykinin receptor antagonists
US6203803B1 (en) 1994-12-14 2001-03-20 Societe L'oreal S.A. Use of a substance P antagonist in a cosmetic composition, and the composition thus obtained
FR2719476B1 (fr) * 1994-05-05 1997-05-23 Oreal Utilisation d'un antagoniste de substance P dans une composition cosmétique et composition obtenue.
FR2719474B1 (fr) 1994-05-05 1996-05-31 Oreal Utilisation d'un antagoniste de substance P dans une composition cosmétique et composition obtenue.
TW397825B (en) * 1994-10-14 2000-07-11 Novartis Ag Aroyl-piperidine derivatives
FR2725900B1 (fr) * 1994-10-21 1997-07-18 Sanofi Sa Utilisation d'antagonistes des recepteurs nk1 pour la preparation de medicaments a action cardioregulatrice
IL116249A (en) * 1994-12-12 2003-07-06 Pfizer Nk-1 receptor antagonists for the treatment of neuronal damage and stroke
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2729954B1 (fr) 1995-01-30 1997-08-01 Sanofi Sa Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
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Also Published As

Publication number Publication date
CA2084193C (en) 1998-04-07
HU9203777D0 (en) 1993-03-29
PT97771A (pt) 1992-03-31
EP0532527A1 (en) 1993-03-24
JPH05506243A (ja) 1993-09-16
NO924612D0 (no) 1992-11-30
DK0532527T3 (da) 1995-01-02
KR930700499A (ko) 1993-03-15
ATE113947T1 (de) 1994-11-15
FI925443A0 (fi) 1992-11-30
DE69105131T2 (de) 1995-03-23
AU7860291A (en) 1991-12-31
CA2084193A1 (en) 1991-12-02
ZA914134B (en) 1993-01-27
US5451586A (en) 1995-09-19
FI113654B (sv) 2004-05-31
IL98259A0 (en) 1992-06-21
JPH072740B2 (ja) 1995-01-18
ES2063507T3 (es) 1995-01-01
DE69105131D1 (de) 1994-12-15
FI925443A (fi) 1992-11-30
IE911856A1 (en) 1991-12-04
HUT62891A (en) 1993-06-28
EP0532527B1 (en) 1994-11-09
AU648317B2 (en) 1994-04-21
WO1991018899A1 (en) 1991-12-12

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