NO341949B1 - Triazolylfenylbenzensulfonamider - Google Patents

Triazolylfenylbenzensulfonamider Download PDF

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Publication number
NO341949B1
NO341949B1 NO20090662A NO20090662A NO341949B1 NO 341949 B1 NO341949 B1 NO 341949B1 NO 20090662 A NO20090662 A NO 20090662A NO 20090662 A NO20090662 A NO 20090662A NO 341949 B1 NO341949 B1 NO 341949B1
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NO
Norway
Prior art keywords
triazol
chloro
tert
benzenesulfonamide
butyl
Prior art date
Application number
NO20090662A
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English (en)
Norwegian (no)
Swedish (sv)
Other versions
NO20090662L (no
Inventor
Trevor T Charvat
Cheng Hu
Anita Melikian
Aaron Novack
Andrew M K Pennell
Edward J Sullivan
Xuefei Tan
William D Thomas
Solomon Ungashe
Yibin Zeng
Sreenivas Punna
Original Assignee
Chemocentryx Inc
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Application filed by Chemocentryx Inc filed Critical Chemocentryx Inc
Publication of NO20090662L publication Critical patent/NO20090662L/no
Publication of NO341949B1 publication Critical patent/NO341949B1/no

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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Animal Behavior & Ethology (AREA)
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  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Immunology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
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  • Dermatology (AREA)
  • Obesity (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
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NO20090662A 2006-07-14 2009-02-11 Triazolylfenylbenzensulfonamider NO341949B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US83104206P 2006-07-14 2006-07-14
US94583907P 2007-06-22 2007-06-22
PCT/US2007/015808 WO2008010934A2 (en) 2006-07-14 2007-07-10 Triazolyl phenyl benzenesulfonamides

Publications (2)

Publication Number Publication Date
NO20090662L NO20090662L (no) 2009-03-26
NO341949B1 true NO341949B1 (no) 2018-02-26

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ID=38896161

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20090662A NO341949B1 (no) 2006-07-14 2009-02-11 Triazolylfenylbenzensulfonamider

Country Status (21)

Country Link
EP (1) EP2046762B1 (enExample)
JP (1) JP5266219B2 (enExample)
KR (1) KR101433392B1 (enExample)
AT (1) ATE498615T1 (enExample)
AU (1) AU2007275873B2 (enExample)
BR (1) BRPI0714407A2 (enExample)
CA (1) CA2657776C (enExample)
CO (1) CO6180465A2 (enExample)
DE (1) DE602007012552D1 (enExample)
DK (1) DK2046762T3 (enExample)
EA (1) EA015710B1 (enExample)
IL (1) IL196409A (enExample)
MA (1) MA30690B1 (enExample)
MX (1) MX2009000395A (enExample)
NO (1) NO341949B1 (enExample)
NZ (1) NZ574759A (enExample)
PL (1) PL2046762T3 (enExample)
PT (1) PT2046762E (enExample)
UA (1) UA98304C2 (enExample)
WO (1) WO2008010934A2 (enExample)
ZA (1) ZA200900281B (enExample)

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US7683176B2 (en) 2006-07-14 2010-03-23 Chemocentryx, Inc. Triazolyl pyridyl benzenesulfonamides
CA2677481C (en) 2007-02-08 2015-07-07 Synta Pharmaceuticals Corp. Triazole compounds that modulate hsp90 activity
TWI490214B (zh) * 2008-05-30 2015-07-01 艾德克 上野股份有限公司 苯或噻吩衍生物及該等作為ｖａｐ－１抑制劑之用途
WO2010005922A1 (en) * 2008-07-07 2010-01-14 Fasgen, Inc. Novel compounds, pharmaceutical compositions containing same, methods of use for same, and methods for preparing same
US8343977B2 (en) 2009-12-30 2013-01-01 Arqule, Inc. Substituted triazolo-pyrimidine compounds
SG192126A1 (en) * 2011-01-25 2013-09-30 Univ Michigan Bcl-2/bcl-xl inhibitors and therapeutic methods using the same
WO2013016155A1 (en) * 2011-07-22 2013-01-31 Glaxo Group Limited Polymorphic forms of the sodium salt of 4-tert-butyl-n-[4-chloro-2-(1-oxy-pyridine-4-carbonyl)-phenyl]-benzenesulfonamide
HUE032747T2 (en) * 2011-07-22 2017-10-30 Chemocentryx Inc Crystalline form of the sodium salt of 4-tert-butyl-N- [4-chloro-2- (1-oxypyridine-4-carbonyl) phenyl] benzenesulfonamide
JP6166721B2 (ja) * 2011-07-22 2017-07-19 ケモセントリックス， インコーポレイテッド ４−ｔｅｒｔ−ブチル−Ｎ−［４−クロロ−２−（１−オキシ−ピリジン−４−カルボニル）−フェニル］−ベンゼンスルホンアミドのナトリウム塩の多形
US20140329809A1 (en) 2011-10-28 2014-11-06 Galderma Research & Development New leukocyte infiltrate markers for rosacea and uses thereof
CA2865714C (en) * 2012-02-29 2021-06-15 Chemocentryx, Inc. Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists
EP2820010B1 (en) * 2012-03-01 2018-05-09 Allergan, Inc. Benzofuran-2-sulfonamide derivatives as chemokine receptor modulators
ES2735360T3 (es) * 2013-12-02 2019-12-18 Chemocentryx Inc Compuestos CCR6
EP3087074A1 (en) 2013-12-23 2016-11-02 Norgine BV Benzene sulfonamides as ccr9 inhibitors
EP3087069B1 (en) 2013-12-23 2019-01-30 Norgine B.V. Compounds useful as ccr9 modulators
US10000458B2 (en) * 2016-03-31 2018-06-19 Sumitomo Chemical Company, Limited Production method of 1, 2, 4-triazole compound
CA3136279A1 (en) 2019-05-09 2020-11-12 Grey Wolf Therapeutics Limited Phenyl-sulfamoyl.benzoyc acids as erap1 modulators
EP3996711A4 (en) 2019-07-10 2023-08-16 ChemoCentryx, Inc. Indanes as pd-l1 inhibitors
KR20220084119A (ko) 2019-10-16 2022-06-21 케모센트릭스, 인크. Pd-l1 질환의 치료를 위한 헤테로아릴-바이페닐 아미드
US11866429B2 (en) 2019-10-16 2024-01-09 Chemocentryx, Inc. Heteroaryl-biphenyl amines for the treatment of PD-L1 diseases
CN115477626B (zh) * 2021-06-16 2024-08-02 上海璃道医药科技有限公司 N-取代苯基磺酰胺类化合物及其用途
JP2024534799A (ja) * 2021-08-20 2024-09-26 エナンタ ファーマシューティカルズ インコーポレイテッド １７－ベータ－ヒドロキシステロイドデヒドロゲナーゼ１３型阻害剤及びその使用方法

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WO2008010934A3 (en) 2008-03-27
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