NO333679B1 - Forbindelse eller farmasoytisk salt derav, samt anvendelser og fremgangsmate for fremstilling av samme - Google Patents
Forbindelse eller farmasoytisk salt derav, samt anvendelser og fremgangsmate for fremstilling av samme Download PDFInfo
- Publication number
- NO333679B1 NO333679B1 NO20060219A NO20060219A NO333679B1 NO 333679 B1 NO333679 B1 NO 333679B1 NO 20060219 A NO20060219 A NO 20060219A NO 20060219 A NO20060219 A NO 20060219A NO 333679 B1 NO333679 B1 NO 333679B1
- Authority
- NO
- Norway
- Prior art keywords
- group
- alkoxy
- compound
- alkyl group
- alkyl
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Classifications
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- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H5/00—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
- C07H5/04—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium to nitrogen
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Diabetes (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Obesity (AREA)
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- Endocrinology (AREA)
- Urology & Nephrology (AREA)
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- Child & Adolescent Psychology (AREA)
- Ophthalmology & Optometry (AREA)
- Neurosurgery (AREA)
- Vascular Medicine (AREA)
- Neurology (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49152303P | 2003-08-01 | 2003-08-01 | |
| PCT/JP2004/011311 WO2005012321A1 (en) | 2003-08-01 | 2004-07-30 | Novel compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20060219L NO20060219L (no) | 2006-04-28 |
| NO333679B1 true NO333679B1 (no) | 2013-08-05 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20060219A NO333679B1 (no) | 2003-08-01 | 2006-01-16 | Forbindelse eller farmasoytisk salt derav, samt anvendelser og fremgangsmate for fremstilling av samme |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7521430B2 (pt) |
| EP (1) | EP1654269B1 (pt) |
| JP (1) | JP4717811B2 (pt) |
| KR (1) | KR101101500B1 (pt) |
| CN (2) | CN102060888A (pt) |
| AU (1) | AU2004260760B2 (pt) |
| BR (1) | BRPI0413233A (pt) |
| CA (1) | CA2534022C (pt) |
| EA (1) | EA011025B1 (pt) |
| ES (1) | ES2527053T3 (pt) |
| IL (1) | IL173051A (pt) |
| MX (1) | MXPA06001273A (pt) |
| NO (1) | NO333679B1 (pt) |
| NZ (1) | NZ545305A (pt) |
| TW (1) | TWI377209B (pt) |
| UA (5) | UA86042C2 (pt) |
| WO (1) | WO2005012321A1 (pt) |
| ZA (2) | ZA200601686B (pt) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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| DK2488515T3 (en) * | 2009-10-14 | 2017-02-27 | Janssen Pharmaceutica Nv | PROCEDURE FOR THE PREPARATION OF COMPOUNDS USED AS INHIBITORS OF SGLT2 |
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| HUE029853T2 (en) | 2010-05-11 | 2017-04-28 | Janssen Pharmaceutica Nv | Pharmaceutical formulations containing 1- (beta-D-Glucopyranosyl) -2-thienylmethylbenzene derivatives as SGLT inhibitors |
| CA2832938C (en) | 2011-04-13 | 2019-09-03 | Janssen Pharmaceutica Nv | Process for the preparation of compounds useful as inhibitors of sglt2 |
| US9035044B2 (en) | 2011-05-09 | 2015-05-19 | Janssen Pharmaceutica Nv | L-proline and citric acid co-crystals of (2S, 3R, 4R, 5S,6R)-2-(3-((5-(4-fluorophenyl)thiopen-2-yl)methyl)4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol |
| ES2835828T3 (es) * | 2013-02-26 | 2021-06-23 | Mitsubishi Tanabe Pharma Corp | Procedimiento para producir a-halo-tetraacilglucosa |
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| US6683056B2 (en) | 2000-03-30 | 2004-01-27 | Bristol-Myers Squibb Company | O-aryl glucoside SGLT2 inhibitors and method |
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| CA2429833A1 (en) * | 2000-11-30 | 2002-06-06 | Kissei Pharmaceutical Co., Ltd. | Glucopyranosyloxybenzylbenzene derivatives, medicinal compositions containing the same and intermediates in the production thereof |
| PL209375B1 (pl) | 2000-12-28 | 2011-08-31 | Kissei Pharmaceutical | Pochodne glukopiranozyloksypirazolu, kompozycja farmaceutyczna zawierająca takie pochodne i zastosowanie tych pochodnych do wytwarzania kompozycji farmaceutycznej |
| TWI255817B (en) * | 2001-02-14 | 2006-06-01 | Kissei Pharmaceutical | Glucopyranosyloxybenzylbenzene derivatives and medicinal use thereof |
| EP1432720A1 (en) * | 2001-09-05 | 2004-06-30 | Bristol-Myers Squibb Company | O-pyrazole glucoside sglt2 inhibitors and method of use |
| DE102004048388A1 (de) * | 2004-10-01 | 2006-04-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | D-Pyranosyl-substituierte Phenyle, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung |
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- 2004-07-30 BR BRPI0413233-5A patent/BRPI0413233A/pt not_active IP Right Cessation
- 2004-07-30 CA CA2534022A patent/CA2534022C/en not_active Expired - Fee Related
- 2004-07-30 KR KR1020067002158A patent/KR101101500B1/ko not_active IP Right Cessation
- 2004-07-30 EP EP04771313.6A patent/EP1654269B1/en not_active Expired - Lifetime
- 2004-07-30 WO PCT/JP2004/011311 patent/WO2005012321A1/en active Application Filing
- 2004-07-30 MX MXPA06001273A patent/MXPA06001273A/es active IP Right Grant
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|---|---|
| WO2005012321A1 (en) | 2005-02-10 |
| IL173051A (en) | 2012-06-28 |
| EP1654269A1 (en) | 2006-05-10 |
| UA86042C2 (en) | 2009-03-25 |
| NZ545305A (en) | 2008-11-28 |
| CN1829728A (zh) | 2006-09-06 |
| AU2004260760A1 (en) | 2005-02-10 |
| UA83377C2 (uk) | 2008-07-10 |
| UA86599C2 (en) | 2009-05-12 |
| CN102060888A (zh) | 2011-05-18 |
| ZA200603880B (en) | 2010-01-27 |
| TWI377209B (en) | 2012-11-21 |
| US20070060545A1 (en) | 2007-03-15 |
| BRPI0413233A (pt) | 2006-10-03 |
| ES2527053T3 (es) | 2015-01-20 |
| JP4717811B2 (ja) | 2011-07-06 |
| UA87991C2 (en) | 2009-09-10 |
| EA011025B1 (ru) | 2008-12-30 |
| NO20060219L (no) | 2006-04-28 |
| KR20060132539A (ko) | 2006-12-21 |
| CA2534022C (en) | 2012-10-02 |
| CA2534022A1 (en) | 2005-02-10 |
| ZA200601686B (en) | 2007-05-30 |
| EA200600348A1 (ru) | 2006-08-25 |
| UA85569C2 (ru) | 2009-02-10 |
| KR101101500B1 (ko) | 2012-01-03 |
| IL173051A0 (en) | 2006-06-11 |
| EP1654269B1 (en) | 2014-10-15 |
| US7521430B2 (en) | 2009-04-21 |
| MXPA06001273A (es) | 2006-04-11 |
| JP2007518682A (ja) | 2007-07-12 |
| TW200510440A (en) | 2005-03-16 |
| AU2004260760B2 (en) | 2009-08-13 |
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Owner name: MITSUBISHI TANABE PHARMA CORP, JP |
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| MM1K | Lapsed by not paying the annual fees |