NO331745B1 - Blandinger av syklosporin-analoger og bruk av disse som immunmodulerende forbindelser - Google Patents
Blandinger av syklosporin-analoger og bruk av disse som immunmodulerende forbindelser Download PDFInfo
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- NO331745B1 NO331745B1 NO20042029A NO20042029A NO331745B1 NO 331745 B1 NO331745 B1 NO 331745B1 NO 20042029 A NO20042029 A NO 20042029A NO 20042029 A NO20042029 A NO 20042029A NO 331745 B1 NO331745 B1 NO 331745B1
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- mixture
- isomer
- accordance
- cyclosporine
- isatx247
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US34620101P | 2001-10-19 | 2001-10-19 | |
PCT/CA2002/001560 WO2003033527A2 (en) | 2001-10-19 | 2002-10-17 | Cyclosporine analogue mixtures and their use as immunomodulating agents |
Publications (2)
Publication Number | Publication Date |
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NO20042029L NO20042029L (no) | 2004-05-14 |
NO331745B1 true NO331745B1 (no) | 2012-03-19 |
Family
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Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
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NO20042029A NO331745B1 (no) | 2001-10-19 | 2004-05-14 | Blandinger av syklosporin-analoger og bruk av disse som immunmodulerende forbindelser |
NO2022042C NO2022042I1 (no) | 2001-10-19 | 2022-10-14 | Voclosporin, a calcineurin inhibitor, its salts and esters |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
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NO2022042C NO2022042I1 (no) | 2001-10-19 | 2022-10-14 | Voclosporin, a calcineurin inhibitor, its salts and esters |
Country Status (38)
Country | Link |
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US (2) | US20110092669A1 (ro) |
EP (2) | EP1436322B1 (ro) |
JP (4) | JP2005511538A (ro) |
KR (1) | KR100992850B1 (ro) |
CN (1) | CN100344648C (ro) |
AR (1) | AR036853A1 (ro) |
AT (1) | ATE401339T1 (ro) |
AU (1) | AU2002331510B2 (ro) |
BE (1) | BE2022C547I2 (ro) |
BR (1) | BR0213659A (ro) |
CA (2) | CA2727642C (ro) |
CO (1) | CO5570682A2 (ro) |
CY (2) | CY1108410T1 (ro) |
DE (1) | DE60227686D1 (ro) |
DK (1) | DK1436322T3 (ro) |
EC (3) | ECSP045059A (ro) |
ES (1) | ES2310604T3 (ro) |
FI (1) | FIC20220041I1 (ro) |
FR (1) | FR22C1051I2 (ro) |
HK (1) | HK1062567A1 (ro) |
HR (1) | HRP20040353B1 (ro) |
IL (2) | IL160762A0 (ro) |
LT (1) | LTC1436322I2 (ro) |
MA (1) | MA26337A1 (ro) |
ME (1) | ME00487B (ro) |
MX (1) | MXPA04003624A (ro) |
MY (1) | MY187182A (ro) |
NL (1) | NL301200I2 (ro) |
NO (2) | NO331745B1 (ro) |
NZ (1) | NZ531945A (ro) |
PL (1) | PL210697B1 (ro) |
PT (1) | PT1436322E (ro) |
RU (1) | RU2337106C2 (ro) |
SI (1) | SI1436322T1 (ro) |
TN (1) | TNSN04069A1 (ro) |
UY (1) | UY27502A1 (ro) |
WO (1) | WO2003033527A2 (ro) |
ZA (1) | ZA200402270B (ro) |
Families Citing this family (22)
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MY187182A (en) * | 2001-10-19 | 2021-09-08 | Isotechnika Inc | Cyclosporine analogue mixtures and their use as immunomodulating agents |
NZ531944A (en) | 2001-10-19 | 2006-03-31 | Isotechnika Inc | Synthesis of cyclosporin analogs |
TW200505946A (en) * | 2003-04-08 | 2005-02-16 | Hoffmann La Roche | Process for preparation of cyclosporin a analog |
WO2006063470A1 (en) * | 2004-12-17 | 2006-06-22 | Isotechnika Inc. | Metabolites of cyclosporin analogs |
US7696165B2 (en) | 2006-03-28 | 2010-04-13 | Albany Molecular Research, Inc. | Use of cyclosporin alkyne analogues for preventing or treating viral-induced disorders |
US7696166B2 (en) | 2006-03-28 | 2010-04-13 | Albany Molecular Research, Inc. | Use of cyclosporin alkyne/alkene analogues for preventing or treating viral-induced disorders |
AU2008310956B2 (en) | 2007-10-08 | 2014-08-07 | Aurinia Pharmaceuticals Inc. | Ophthalmic compositions comprising calcineurin inhibitors or mTOR inhibitors |
US9017725B2 (en) | 2009-06-09 | 2015-04-28 | Aurinia Pharmaceuticals Inc. | Topical drug delivery systems for ophthalmic use |
GB0912584D0 (en) * | 2009-07-20 | 2009-08-26 | Ucl Business Plc | Cyclosporin conjugates |
HUE042490T2 (hu) | 2010-12-15 | 2019-07-29 | Contravir Pharmaceuticals Inc | 1-es és 3-as aminosav-pozícióban módosított ciklosporin analóg molekulák |
GB201222455D0 (en) * | 2012-12-13 | 2013-01-30 | Perioc Ltd | Novel pharmaceutical formulations and their use in the treatment of periodontaldisease |
JP2020510249A (ja) * | 2016-11-30 | 2020-04-02 | シュレーディンガー インコーポレイテッドSchrodinger,Inc. | 化学の遷移状態を計算するためのグラフィカルユーザインタフェース |
EP3551046B1 (en) | 2016-12-07 | 2023-07-19 | Biora Therapeutics, Inc. | Gastrointestinal tract detection methods, devices and systems |
WO2018106928A1 (en) | 2016-12-08 | 2018-06-14 | Contravir Pharmaceuticals, Inc. | Treatment and prevention of hbv diseases by cyclosporine analogue molecules modified at amino acides 1 and 3 |
US11523772B2 (en) | 2016-12-14 | 2022-12-13 | Biora Therapeutics, Inc. | Treatment of a disease of the gastrointestinal tract with an immunosuppressant |
US20190224275A1 (en) | 2017-05-12 | 2019-07-25 | Aurinia Pharmaceuticals Inc. | Protocol for treatment of lupus nephritis |
US10286036B2 (en) * | 2017-05-12 | 2019-05-14 | Aurinia Pharmaceuticals Inc. | Protocol for treatment of lupus nephritis |
WO2019246312A1 (en) | 2018-06-20 | 2019-12-26 | Progenity, Inc. | Treatment of a disease of the gastrointestinal tract with an immunomodulator |
EP4201952A1 (en) | 2021-12-21 | 2023-06-28 | Curia Spain, S.A.U. | Process for the controlled synthesis of voclosporin |
WO2024052941A1 (en) * | 2022-09-09 | 2024-03-14 | Dr. Reddy's Laboratories Limited | Improved process for the preparation of voclosporin |
WO2024157132A1 (en) * | 2023-01-25 | 2024-08-02 | Indena S.P.A. | Process for the preparation of an intermediate useful for the synthesis of voclosporin |
WO2024157186A1 (en) * | 2023-01-25 | 2024-08-02 | Procos S.P.A. | New process for the preparation of amorphous voclosporin |
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US4278545A (en) * | 1979-09-12 | 1981-07-14 | The Bendix Corporation | Apparatus for separating solids and liquid components |
CH670644A5 (ro) * | 1986-12-18 | 1989-06-30 | Lonza Ag | |
US5162540A (en) * | 1986-12-18 | 1992-11-10 | Lonza Ltd. | Process for the production of (+) biotin |
ES2059558T3 (es) * | 1987-06-17 | 1994-11-16 | Sandoz Ag | Ciclosporins y su uso como productos farmaceuticos. |
US5972630A (en) * | 1991-08-19 | 1999-10-26 | Dade Behring Marburg Gmbh | Homogeneous immunoassays using enzyme inhibitors |
US5750510A (en) * | 1997-04-04 | 1998-05-12 | Abbott Laboratories | 3-descladinose-2,3-anhydroerythromycin derivatives |
US5939406A (en) * | 1997-07-21 | 1999-08-17 | Wisconsin Alumni Research Foundation | 18-substituted-19-nor-vitamin D compounds |
KR100585348B1 (ko) * | 1997-10-08 | 2006-06-01 | 이소테크니카 인코포레이티드 | 중수소화된 시클로스포린 유사체 및 면역조절제로서 그의용도 |
MY187182A (en) * | 2001-10-19 | 2021-09-08 | Isotechnika Inc | Cyclosporine analogue mixtures and their use as immunomodulating agents |
NZ531944A (en) * | 2001-10-19 | 2006-03-31 | Isotechnika Inc | Synthesis of cyclosporin analogs |
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CHAD | Change of the owner's name or address (par. 44 patent law, par. patentforskriften) |
Owner name: AURINIA PHARMACEUTICALS INC, CA |
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Representative=s name: ACAPO AS, POSTBOKS 1880 NORDNES, 5817 BERGEN, NORG |
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Free format text: PRODUCT NAME: VOCLOSPORIN, A CALCINEURIN INHIBITOR, ITS SALTS AND ESTERS; NAT. REG. NO/DATE: EU/1/22/1678 20220920; FIRST REG. NO/DATE: EU/1/22/1678/001 20220915 Spc suppl protection certif: 2022042 Filing date: 20221014 |
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